Total properties:
62
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Patent #:
|
|
Issue Dt:
|
11/08/2005
|
Application #:
|
10392195
|
Filing Dt:
|
03/19/2003
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Publication #:
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|
Pub Dt:
|
10/02/2003
| | | | |
Title:
|
(+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE: METHODS OF USING AND COMPOSITIONS THEREOF
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Patent #:
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Issue Dt:
|
02/06/2007
|
Application #:
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10748085
|
Filing Dt:
|
12/29/2003
|
Publication #:
|
|
Pub Dt:
|
10/14/2004
| | | | |
Title:
|
FLUOROALKOXY-SUBSTITUTED 1,3-DIHYDRO-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES
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Patent #:
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Issue Dt:
|
06/28/2005
|
Application #:
|
10798372
|
Filing Dt:
|
03/12/2004
|
Publication #:
|
|
Pub Dt:
|
12/23/2004
| | | | |
Title:
|
N-ALKYL-HYDROXAMIC ACID-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES
|
|
|
Patent #:
|
|
Issue Dt:
|
07/17/2007
|
Application #:
|
10900270
|
Filing Dt:
|
07/28/2004
|
Publication #:
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Pub Dt:
|
04/20/2006
| | | | |
Title:
|
ISOINDOLINE COMPOUNDS AND METHODS OF MAKING AND USING THE SAME
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|
Patent #:
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|
Issue Dt:
|
07/29/2008
|
Application #:
|
10900332
|
Filing Dt:
|
07/28/2004
|
Publication #:
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|
Pub Dt:
|
02/02/2006
| | | | |
Title:
|
ISOINDOLINE COMPOUNDS AND METHODS OF THEIR USE
|
|
|
Patent #:
|
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Issue Dt:
|
09/23/2008
|
Application #:
|
11106142
|
Filing Dt:
|
04/13/2005
|
Publication #:
|
|
Pub Dt:
|
09/01/2005
| | | | |
Title:
|
(+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE:, AND METHODS OF SYNTHESIS AND COMPOSITIONS THEREOF
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Patent #:
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Issue Dt:
|
02/16/2010
|
Application #:
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11124280
|
Filing Dt:
|
05/09/2005
|
Publication #:
|
|
Pub Dt:
|
09/15/2005
| | | | |
Title:
|
METHODS OF USING N-ALKYL-HYDROXAMIC ACID-ISOINDOLYL COMPOUNDS
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Patent #:
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Issue Dt:
|
04/15/2008
|
Application #:
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11170308
|
Filing Dt:
|
06/28/2005
|
Publication #:
|
|
Pub Dt:
|
12/01/2005
| | | | |
Title:
|
METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4 ACETYLAMINOISOINDOLINE 1,3-DIONE
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Patent #:
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Issue Dt:
|
04/24/2007
|
Application #:
|
11392845
|
Filing Dt:
|
03/28/2006
|
Publication #:
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|
Pub Dt:
|
08/17/2006
| | | | |
Title:
|
METHODS OF THE TREATMENT OF PSORIATIC ARTHRITIS USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
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Patent #:
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Issue Dt:
|
10/02/2007
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Application #:
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11392846
|
Filing Dt:
|
03/28/2006
|
Publication #:
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|
Pub Dt:
|
08/17/2006
| | | | |
Title:
|
METHODS OF THE TREATMENT OR PREVENTION OF EXERCISE-INDUCED ASTHMA USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
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Patent #:
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Issue Dt:
|
03/17/2009
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Application #:
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11601355
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Filing Dt:
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11/16/2006
|
Publication #:
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|
Pub Dt:
|
03/29/2007
| | | | |
Title:
|
FLUOROALKOXY-SUBSTITUTED 1,3-DIHYDRO-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES
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|
Patent #:
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Issue Dt:
|
02/24/2009
|
Application #:
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11820788
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Filing Dt:
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06/19/2007
|
Publication #:
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Pub Dt:
|
10/18/2007
| | | | |
Title:
|
ISOINDOLINE COMPOUNDS AND METHODS OF MAKING AND USING THE SAME
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Patent #:
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Issue Dt:
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03/24/2009
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Application #:
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11824523
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Filing Dt:
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06/29/2007
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Publication #:
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|
Pub Dt:
|
01/31/2008
| | | | |
Title:
|
METHODS OF USING(+)-2-[1-(3-ETHOXY-4METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3,-DIONE
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Patent #:
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Issue Dt:
|
02/09/2010
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Application #:
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12069282
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Filing Dt:
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02/08/2008
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Publication #:
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Pub Dt:
|
08/28/2008
| | | | |
Title:
|
METHODS OF USING (+)-2-[1-(3-ETHOXY-4 METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4 ACETYLAMINOISOINDOLINE 1,3-DIONE
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Patent #:
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Issue Dt:
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08/04/2009
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Application #:
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12070322
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Filing Dt:
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02/15/2008
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Publication #:
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Pub Dt:
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06/19/2008
| | | | |
Title:
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ISOINDOLINE COMPOUNDS AND METHODS OF THEIR USE
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Patent #:
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Issue Dt:
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02/22/2011
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Application #:
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12079615
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Filing Dt:
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03/27/2008
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Publication #:
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Pub Dt:
|
09/25/2008
| | | | |
Title:
|
SOLID FORMS COMPRISING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2- METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE, COMPOSITIONS THEREOF, AND USES THEREOF
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Patent #:
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Issue Dt:
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02/09/2010
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Application #:
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12098379
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Filing Dt:
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04/04/2008
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Publication #:
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Pub Dt:
|
10/02/2008
| | | | |
Title:
|
METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE- 1,3-DIONE
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Patent #:
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Issue Dt:
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02/22/2011
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Application #:
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12363664
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Filing Dt:
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01/30/2009
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Publication #:
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Pub Dt:
|
06/04/2009
| | | | |
Title:
|
FLUOROALKOXY-SUBSTITUTED 1,3-DIHYDRO-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES
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Patent #:
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Issue Dt:
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09/27/2011
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Application #:
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12368245
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Filing Dt:
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02/09/2009
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Publication #:
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Pub Dt:
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06/11/2009
| | | | |
Title:
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ISOINDOLINE COMPOUNDS AND METHODS OF MAKING AND USING THE SAME
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Patent #:
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Issue Dt:
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10/19/2010
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Application #:
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12535642
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Filing Dt:
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08/04/2009
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Publication #:
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Pub Dt:
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11/26/2009
| | | | |
Title:
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ISOINDOLINE COMPOUNDS AND METHODS OF THEIR USE
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Patent #:
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Issue Dt:
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08/14/2012
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12556479
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Filing Dt:
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09/09/2009
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Publication #:
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Pub Dt:
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07/01/2010
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Title:
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PROCESSES FOR THE PREPARATION OF AMINOSULFONE COMPOUNDS
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Patent #:
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06/04/2013
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12630788
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12/03/2009
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Publication #:
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Pub Dt:
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06/24/2010
| | | | |
Title:
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METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE 1,3-DIONE
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Patent #:
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12/13/2011
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12705527
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02/12/2010
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Publication #:
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Pub Dt:
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10/21/2010
| | | | |
Title:
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N-ALKYL-HYDROXAMIC ACID-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES
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Patent #:
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Issue Dt:
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05/05/2015
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Application #:
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12942930
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Filing Dt:
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11/09/2010
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05/26/2011
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Title:
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Nanosuspension of a Poorly Soluble Drug via Microfluidization Process
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01/10/2012
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12945800
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11/12/2010
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Publication #:
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Pub Dt:
|
05/12/2011
| | | | |
Title:
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SOLID FORMS COMPRISING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE, COMPOSITIONS THEREOF, AND USES THEREOF
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Patent #:
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04/17/2012
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13010738
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01/20/2011
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Publication #:
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Pub Dt:
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05/26/2011
| | | | |
Title:
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FLUOROALKOXY-SUBSTITUTED 1,3-DIHYDRO-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES
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Patent #:
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NONE
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Application #:
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13161201
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Filing Dt:
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06/15/2011
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Publication #:
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Pub Dt:
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12/29/2011
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Title:
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BIOMARKERS FOR THE TREATMENT OF PSORIASIS
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01/14/2014
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13300458
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11/18/2011
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Pub Dt:
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04/26/2012
| | | | |
Title:
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SOLID FORMS COMPRISING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE, COMPOSITIONS THEREOF, AND USES THEREOF
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Patent #:
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10/07/2014
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13346455
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01/09/2012
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07/12/2012
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Title:
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PHENETHYLSULFONE ISOINDOLINE DERIVATIVES AND THEIR USE
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Patent #:
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Issue Dt:
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03/01/2016
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13458896
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04/27/2012
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Pub Dt:
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11/01/2012
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Title:
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METHODS AND COMPOSITIONS USING PDE4 INHIBITORS FOR THE TREATMENT AND MANAGEMENT OF AUTOIMMUNE AND INFLAMMATORY DISEASES
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Patent #:
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Issue Dt:
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08/09/2016
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13639848
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01/04/2013
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Pub Dt:
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05/30/2013
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Title:
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METHODS FOR TREATING RESPIRATORY VIRAL INFECTION
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08/12/2014
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13682652
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11/20/2012
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Pub Dt:
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01/23/2014
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Title:
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METHODS OF TREATING ARTHRITIC CONDITIONS USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE 1,3-DIONE
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Patent #:
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NONE
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13727366
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12/26/2012
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Pub Dt:
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06/27/2013
| | | | |
Title:
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FORMULATIONS OF (+)-2-[1-(3-ETHOXY-4-METHOXY-PHENYL)-2-METHANESULFONYL-ETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
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Patent #:
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11/17/2015
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13771164
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02/20/2013
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Publication #:
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Pub Dt:
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08/22/2013
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Title:
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PROCESSES FOR THE PREPARATION OF (S)-1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHANESULFONYLETHYLAMINE
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Patent #:
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Issue Dt:
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09/08/2015
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13772242
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Filing Dt:
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02/20/2013
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Pub Dt:
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08/22/2013
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Title:
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ASYMMETRIC SYNTHETIC PROCESSES FOR THE PREPARATION OF AMINOSULFONE COMPOUNDS
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09/12/2017
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13978869
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12/19/2013
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Publication #:
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Pub Dt:
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04/03/2014
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Title:
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ORAL DOSAGE FORMS OF CYCLOPROPANECARBOXYLIC ACID {2-[(1S)-1-(3-ETHOXY-4-METHOXY-PHENYL)-2-METHANESULFONYL-ETHYL]-3-OXO-2,3-DIHYDRO-1H-ISOINDOL-4-YL}-AMIDE
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Patent #:
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06/02/2015
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13979602
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02/26/2014
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Publication #:
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Pub Dt:
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07/10/2014
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Title:
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ISOTOPOLOGUES OF ISOINDOLE DERIVATIVES
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Patent #:
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NONE
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13993046
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Filing Dt:
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10/02/2013
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Publication #:
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Pub Dt:
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01/16/2014
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Title:
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CONTROLLED RELEASE ORAL DOSAGE FORMS OF POORLY SOLUBLE DRUGS AND USES THEREOF
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07/12/2016
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14003750
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02/19/2014
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Pub Dt:
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07/03/2014
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Title:
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METHODS FOR TREATING DISEASES USING ISOINDOLINE COMPOUNDS
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03/17/2015
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14026794
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09/13/2013
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Publication #:
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Pub Dt:
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03/20/2014
| | | | |
Title:
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PROCESSES FOR THE PREPARATION OF ISOINDOLE COMPOUNDS AND ISOTOPOLOGUES THEREOF
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Patent #:
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Issue Dt:
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04/28/2015
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Application #:
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14102407
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Filing Dt:
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12/10/2013
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Publication #:
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Pub Dt:
|
04/10/2014
| | | | |
Title:
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SOLID FORMS COMPRISING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE, COMPOSITIONS THEREOF, AND USES THEREOF
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Patent #:
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Issue Dt:
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01/23/2018
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14209874
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03/13/2014
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Pub Dt:
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06/25/2015
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Title:
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METHODS FOR THE TREATMENT OF PSORIATIC ARTHRITIS USING APREMILAST
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Patent #:
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10/18/2016
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14305082
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06/16/2014
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Pub Dt:
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12/18/2014
| | | | |
Title:
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FORMULATIONS OF (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
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03/15/2016
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14316160
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06/26/2014
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Pub Dt:
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12/18/2014
| | | | |
Title:
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METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE 1,3-DIONE
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Patent #:
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02/06/2018
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14344870
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01/20/2015
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07/09/2015
| | | | |
Title:
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FORMULATIONS OF CYCLOPROPANECARBOXYLIC ACID {2-[(1S)-1-(3-ETHOXY-4-METHOXY-PHENYL)-2-METHANESULFONYL-ETHYL]-3-OXO-2,3-DIHYDRO-1H-ISOINDOL-4-YL}-AMIDE
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NONE
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14603128
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01/22/2015
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07/30/2015
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Title:
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METHODS FOR THE TREATMENT OF OBESITY USING APREMILAST
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09/06/2016
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14642511
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03/09/2015
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Publication #:
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Pub Dt:
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07/02/2015
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Title:
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PROCESSES FOR THE PREPARATION OF ISOINDOLE COMPOUNDS AND ISOTOPOLOGUES THEREOF
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Patent #:
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Issue Dt:
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09/06/2016
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14670336
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03/26/2015
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Publication #:
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Pub Dt:
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07/16/2015
| | | | |
Title:
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SOLID FORMS COMPRISING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4- ACETYLAMINOISOINDOLINE-1,3-DIONE, COMPOSITIONS THEREOF, AND USES THEREOF
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Patent #:
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04/11/2017
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14676709
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04/01/2015
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Pub Dt:
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09/24/2015
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Title:
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NANOSUSPENSION OF A POORLY SOLUBLE DRUG VIA MICROFLUIDIZATION PROCESS
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Patent #:
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11/01/2016
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14712595
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05/14/2015
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Pub Dt:
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11/19/2015
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Title:
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USE OF PDE4 INHIBITORS AND COMBINATIONS THEREOF FOR THE TREATMENT OF CYSTIC FIBROSIS
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05/09/2017
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14726287
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05/29/2015
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Pub Dt:
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09/17/2015
| | | | |
Title:
|
ISOTOPOLOGUES OF ISOINDOLE DERIVATIVES
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|
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Patent #:
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Issue Dt:
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10/09/2018
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Application #:
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14826027
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Filing Dt:
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08/13/2015
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Publication #:
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Pub Dt:
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02/18/2016
| | | | |
Title:
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METHODS FOR THE TREATMENT OF DISEASES AMELIORATED BY PDE4 INHIBITION USING DOSAGE TITRATION OF APREMILAST
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Patent #:
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Issue Dt:
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03/07/2017
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Application #:
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14882564
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Filing Dt:
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10/14/2015
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Publication #:
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Pub Dt:
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02/04/2016
| | | | |
Title:
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PROCESSES FOR THE PREPARATION OF (S)-1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHANESULFONYLETHYLAMINE
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Patent #:
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Issue Dt:
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01/03/2017
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Application #:
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14938714
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Filing Dt:
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11/11/2015
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Publication #:
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Pub Dt:
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05/12/2016
| | | | |
Title:
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CONTROLLED RELEASE ORAL DOSAGE FORMS OF POORLY SOLUBLE DRUGS AND USES THEREOF
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|
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Patent #:
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Issue Dt:
|
08/08/2017
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Application #:
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15016856
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Filing Dt:
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02/05/2016
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Publication #:
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|
Pub Dt:
|
06/02/2016
| | | | |
Title:
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METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
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Patent #:
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NONE
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Issue Dt:
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|
Application #:
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15311153
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Filing Dt:
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11/14/2016
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Publication #:
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Pub Dt:
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03/30/2017
| | | | |
Title:
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COMPOSITIONS AND METHODS FOR THE TREATMENT OF ATHEROSCLEROTIC CARDIOVASCULAR DISEASES WITH PDE4 MODULATORS
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|
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Patent #:
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|
Issue Dt:
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05/28/2019
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Application #:
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15321718
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Filing Dt:
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12/22/2016
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Publication #:
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Pub Dt:
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05/25/2017
| | | | |
Title:
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APREMILAST FOR THE TREATMENT OF A LIVER DISEASE OR A LIVER FUNCTION ABNORMALITY
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|
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Patent #:
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Issue Dt:
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06/27/2017
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Application #:
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15414782
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Filing Dt:
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01/25/2017
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Publication #:
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|
Pub Dt:
|
05/11/2017
| | | | |
Title:
|
PROCESSES FOR THE PREPARATION OF (S)-1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHANESULFONYLETHYLAMINE
|
|
|
Patent #:
|
|
Issue Dt:
|
10/09/2018
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Application #:
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15629678
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Filing Dt:
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06/21/2017
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Publication #:
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|
Pub Dt:
|
10/05/2017
| | | | |
Title:
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METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
|
|
|
Patent #:
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NONE
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Issue Dt:
|
|
Application #:
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16109634
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Filing Dt:
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08/22/2018
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Publication #:
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|
Pub Dt:
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12/20/2018
| | | | |
Title:
|
METHODS FOR THE TREATMENT OF DISEASES AMELIORATED BY PDE4 INHIBITION USING DOSAGE TITRATION OF APREMILAST
|
|
|
Patent #:
|
|
Issue Dt:
|
04/07/2020
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Application #:
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16125571
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Filing Dt:
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09/07/2018
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Publication #:
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Pub Dt:
|
01/03/2019
| | | | |
Title:
|
METHODS OF USING (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE
|
|
|
Patent #:
|
|
Issue Dt:
|
07/28/2015
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Application #:
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29425538
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Filing Dt:
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06/25/2012
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Title:
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PHARMACEUTICAL TABLET
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|