Total properties:
945
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7
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10
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Patent #:
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Issue Dt:
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08/28/2012
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Application #:
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12977222
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Filing Dt:
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12/23/2010
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Publication #:
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Pub Dt:
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01/12/2012
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Title:
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PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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02/19/2013
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Application #:
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12982209
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Filing Dt:
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12/30/2010
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Publication #:
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Pub Dt:
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09/01/2011
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Title:
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PREPARATION OF PROTECTED ALPHA-KETO BETA-AMINO ESTERS AND AMIDES
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Patent #:
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Issue Dt:
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06/30/2015
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Application #:
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13014505
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Filing Dt:
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01/26/2011
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Publication #:
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Pub Dt:
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03/22/2012
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Title:
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PYRAZOLOPYRIDINE KINASE INHIBITORS
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Patent #:
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Issue Dt:
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08/28/2012
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Application #:
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13018908
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Filing Dt:
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02/01/2011
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Publication #:
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Pub Dt:
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05/19/2011
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Title:
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SODIUM CHANNEL PROTEIN TYPE III ALPHA-SUBUNIT SPLICE VARIANT
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Patent #:
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Issue Dt:
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02/19/2013
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Application #:
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13020947
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Filing Dt:
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02/04/2011
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Publication #:
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Pub Dt:
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07/28/2011
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Title:
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AMINOPYRIDINE KINASE INHIBITORS
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Patent #:
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Issue Dt:
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01/10/2012
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Application #:
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13022820
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Filing Dt:
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02/08/2011
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Publication #:
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Pub Dt:
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06/02/2011
| | | | |
Title:
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CASPASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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03/19/2013
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Application #:
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13033872
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Filing Dt:
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02/24/2011
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Publication #:
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Pub Dt:
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11/24/2011
| | | | |
Title:
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THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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09/24/2013
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Application #:
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13034039
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Filing Dt:
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02/24/2011
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Publication #:
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Pub Dt:
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09/29/2011
| | | | |
Title:
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CO-CRYSTALS AND PHARMACEUTICAL FORMULATIONS COMPRISING THE SAME
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Patent #:
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Issue Dt:
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05/14/2013
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Application #:
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13036930
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Filing Dt:
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02/28/2011
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Publication #:
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Pub Dt:
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07/07/2011
| | | | |
Title:
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INHIBITORS OF SERINE PROTEASES
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Patent #:
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Issue Dt:
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06/25/2013
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Application #:
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13053172
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Filing Dt:
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03/21/2011
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Publication #:
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Pub Dt:
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09/22/2011
| | | | |
Title:
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SOLID FORMS OF N-[2,4-BIS(1,1-DIMETHYLETHYL)-5-HYDROXYPHENYL]-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXAMIDE
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Patent #:
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Issue Dt:
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12/04/2012
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Application #:
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13069889
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Filing Dt:
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03/23/2011
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Publication #:
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Pub Dt:
|
07/14/2011
| | | | |
Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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NONE
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Issue Dt:
|
|
Application #:
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13072380
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Filing Dt:
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03/25/2011
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Publication #:
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Pub Dt:
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10/13/2011
| | | | |
Title:
|
SOLID FORMS OF (R)-1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2-YL)-1H-INDOL-5-YL) CYCLOPROPANECARBOXAMIDE
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Patent #:
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Issue Dt:
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02/12/2013
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Application #:
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13074772
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Filing Dt:
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03/29/2011
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Publication #:
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Pub Dt:
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07/28/2011
| | | | |
Title:
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INHIBITORS OF SERINE PROTEASES
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|
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Patent #:
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Issue Dt:
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10/08/2013
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Application #:
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13081750
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Filing Dt:
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04/07/2011
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Publication #:
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Pub Dt:
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10/20/2011
| | | | |
Title:
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PHARMACEUTICAL COMPOSITIONS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACID AND ADMINISTRATION THEREOF
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Patent #:
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Issue Dt:
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08/13/2013
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Application #:
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13082156
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Filing Dt:
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04/07/2011
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Publication #:
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Pub Dt:
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10/27/2011
| | | | |
Title:
|
SOLID FORMS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACID
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Patent #:
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Issue Dt:
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08/27/2013
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Application #:
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13090563
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Filing Dt:
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04/20/2011
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Publication #:
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Pub Dt:
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06/28/2012
| | | | |
Title:
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C-MET PROTEIN KINASE INHIBITORS
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Patent #:
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NONE
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Issue Dt:
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Application #:
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13092838
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Filing Dt:
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04/22/2011
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Publication #:
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Pub Dt:
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10/20/2011
| | | | |
Title:
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Modulators of Cystic Fibrosis Transmembrane Conductance Regulator
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Patent #:
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Issue Dt:
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01/21/2014
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Application #:
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13094183
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Filing Dt:
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04/26/2011
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Publication #:
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Pub Dt:
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03/22/2012
| | | | |
Title:
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TRIAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
|
01/01/2013
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Application #:
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13099643
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Filing Dt:
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05/03/2011
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Publication #:
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Pub Dt:
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08/25/2011
| | | | |
Title:
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TRIAZOLOTHIADIAZOLE INHIBITOR OF C-MET PROTEIN KINASE
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Patent #:
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Issue Dt:
|
12/03/2013
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Application #:
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13102335
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Filing Dt:
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05/06/2011
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Publication #:
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Pub Dt:
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12/15/2011
| | | | |
Title:
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HETEROCYCLIC CHROMENE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS
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Patent #:
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Issue Dt:
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04/02/2013
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Application #:
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13104291
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Filing Dt:
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10/27/2011
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Publication #:
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Pub Dt:
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02/16/2012
| | | | |
Title:
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COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
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|
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Patent #:
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|
Issue Dt:
|
03/03/2015
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Application #:
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13106167
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Filing Dt:
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05/12/2011
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Publication #:
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Pub Dt:
|
07/12/2012
| | | | |
Title:
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COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
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|
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Patent #:
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|
Issue Dt:
|
02/24/2015
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Application #:
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13106173
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Filing Dt:
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05/12/2011
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Publication #:
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Pub Dt:
|
02/09/2012
| | | | |
Title:
|
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
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|
|
Patent #:
|
|
Issue Dt:
|
08/04/2015
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Application #:
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13106178
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Filing Dt:
|
05/12/2011
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Publication #:
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|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
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|
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Patent #:
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|
Issue Dt:
|
05/10/2016
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Application #:
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13106184
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Filing Dt:
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05/12/2011
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Publication #:
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Pub Dt:
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05/17/2012
| | | | |
Title:
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COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
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|
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Patent #:
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|
Issue Dt:
|
06/23/2015
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Application #:
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13106337
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Filing Dt:
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05/12/2011
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Publication #:
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Pub Dt:
|
02/09/2012
| | | | |
Title:
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COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
|
|
|
Patent #:
|
|
Issue Dt:
|
04/25/2017
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Application #:
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13106476
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Filing Dt:
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05/12/2011
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Publication #:
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Pub Dt:
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02/02/2012
| | | | |
Title:
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COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
|
|
|
Patent #:
|
|
Issue Dt:
|
12/25/2012
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Application #:
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13107802
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Filing Dt:
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05/13/2011
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Publication #:
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Pub Dt:
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11/17/2011
| | | | |
Title:
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INHIBITORS OF P38
|
|
|
Patent #:
|
|
Issue Dt:
|
11/27/2012
|
Application #:
|
13108077
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Filing Dt:
|
05/16/2011
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Publication #:
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|
Pub Dt:
|
12/22/2011
| | | | |
Title:
|
MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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|
|
Patent #:
|
|
Issue Dt:
|
09/24/2013
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Application #:
|
13112115
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Filing Dt:
|
05/20/2011
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Publication #:
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|
Pub Dt:
|
12/15/2011
| | | | |
Title:
|
MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/26/2013
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Application #:
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13112868
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Filing Dt:
|
05/20/2011
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Publication #:
|
|
Pub Dt:
|
11/24/2011
| | | | |
Title:
|
Processes for Producing Modulators of Cystic Fibrosis Transmembrane Conductance Regulator
|
|
|
Patent #:
|
|
Issue Dt:
|
09/11/2012
|
Application #:
|
13114215
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Filing Dt:
|
05/24/2011
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Publication #:
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|
Pub Dt:
|
12/01/2011
| | | | |
Title:
|
AMINOPYRAZOLE TRIAZOLOTHIADIAZOLE INHIBITOR OF C-MET PROTEIN KINASE
|
|
|
Patent #:
|
|
Issue Dt:
|
03/04/2014
|
Application #:
|
13153199
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Filing Dt:
|
06/03/2011
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Publication #:
|
|
Pub Dt:
|
02/23/2012
| | | | |
Title:
|
TREATMENT OF HEPATITIS C VIRUS WITH TELAPREVIR (VX-950) IN PATIENTS NON-RESPONSIVE TO TREATMENT WITH PEGYLATED INTERFERON-ALPHA 2A/2B AND RIBAVIRIN
|
|
|
Patent #:
|
|
Issue Dt:
|
10/22/2013
|
Application #:
|
13155420
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Filing Dt:
|
06/08/2011
|
Publication #:
|
|
Pub Dt:
|
01/19/2012
| | | | |
Title:
|
FORMULATIONS OF (R)-1-(2,2-DIFLUOROBENZO[D] [1,3] DIOXOL-5-YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2-YL)-1H-INDOL-5-YL)CYCLOPROPANECARBOXAMIDE
|
|
|
Patent #:
|
|
Issue Dt:
|
01/07/2014
|
Application #:
|
13167654
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Filing Dt:
|
06/23/2011
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Publication #:
|
|
Pub Dt:
|
02/23/2012
| | | | |
Title:
|
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
|
|
|
Patent #:
|
|
Issue Dt:
|
11/06/2012
|
Application #:
|
13171652
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Filing Dt:
|
06/29/2011
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Publication #:
|
|
Pub Dt:
|
08/02/2012
| | | | |
Title:
|
MODULATORS OF MUSCARINIC RECEPTORS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/30/2013
|
Application #:
|
13174844
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Filing Dt:
|
07/01/2011
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Publication #:
|
|
Pub Dt:
|
01/05/2012
| | | | |
Title:
|
MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/19/2013
|
Application #:
|
13178677
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Filing Dt:
|
07/08/2011
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Publication #:
|
|
Pub Dt:
|
01/12/2012
| | | | |
Title:
|
MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
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|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
13182695
|
Filing Dt:
|
07/14/2011
|
Publication #:
|
|
Pub Dt:
|
01/19/2012
| | | | |
Title:
|
PALATABLE PHARMACEUTICAL COMPOSITION
|
|
|
Patent #:
|
|
Issue Dt:
|
03/25/2014
|
Application #:
|
13186985
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Filing Dt:
|
07/20/2011
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Publication #:
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|
Pub Dt:
|
05/24/2012
| | | | |
Title:
|
METHODS FOR AMPLIFYING HEPATITIS C VIRUS NUCLEIC ACIDS
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|
|
Patent #:
|
|
Issue Dt:
|
03/03/2015
|
Application #:
|
13187416
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Filing Dt:
|
07/20/2011
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Publication #:
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|
Pub Dt:
|
01/24/2013
| | | | |
Title:
|
DEVICE TO COLLECT AND SEGREGATE TISSUE SAMPLES SECTIONED ON A MICROTOME
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|
|
Patent #:
|
|
Issue Dt:
|
05/21/2013
|
Application #:
|
13193739
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Filing Dt:
|
07/29/2011
|
Publication #:
|
|
Pub Dt:
|
06/28/2012
| | | | |
Title:
|
AZAINDAZOLES USEFUL AS INHIBITORS OF KINASES
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|
|
Patent #:
|
|
Issue Dt:
|
10/16/2012
|
Application #:
|
13205291
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Filing Dt:
|
08/08/2011
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Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
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|
|
Patent #:
|
|
Issue Dt:
|
03/12/2013
|
Application #:
|
13206638
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Filing Dt:
|
08/10/2011
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Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
DIHYDRODIAZEPINES USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
13206954
|
Filing Dt:
|
08/10/2011
|
Publication #:
|
|
Pub Dt:
|
12/08/2011
| | | | |
Title:
|
TRIAZOLOTHIADIAZOLE INHIBITOR OF C-MET PROTEIN KINASE
|
|
|
Patent #:
|
|
Issue Dt:
|
12/11/2012
|
Application #:
|
13210712
|
Filing Dt:
|
08/16/2011
|
Publication #:
|
|
Pub Dt:
|
12/08/2011
| | | | |
Title:
|
PRODRUG OF AN ICE INHIBITOR
|
|
|
Patent #:
|
|
Issue Dt:
|
09/03/2013
|
Application #:
|
13211502
|
Filing Dt:
|
08/17/2011
|
Publication #:
|
|
Pub Dt:
|
02/16/2012
| | | | |
Title:
|
TETRAHYDROTHIAZOLOPYRIDINE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
13214419
|
Filing Dt:
|
08/22/2011
|
Publication #:
|
|
Pub Dt:
|
02/23/2012
| | | | |
Title:
|
PHARMACEUTICAL COMPOSITIONS OF (R)-1-(2,2-DIFLUOROBENZO[D] [1,3]DIOXOL-5-YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2-YL)-1H-INDOL-5-YL) CYCLOPROPANECARBOXAMIDE AND ADMINISTRATION THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
04/01/2014
|
Application #:
|
13216530
|
Filing Dt:
|
08/24/2011
|
Publication #:
|
|
Pub Dt:
|
06/21/2012
| | | | |
Title:
|
PROCESSES FOR THE FACILE SYNTHESIS OF DIARYL AMINES AND ANALOGUES THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
09/18/2012
|
Application #:
|
13216606
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Filing Dt:
|
08/24/2011
|
Publication #:
|
|
Pub Dt:
|
03/01/2012
| | | | |
Title:
|
TRI-CYCLIC PYRAZOLOPYRIDINE KINASE INHIBITORS
|
|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
13219590
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Filing Dt:
|
08/26/2011
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Publication #:
|
|
Pub Dt:
|
03/15/2012
| | | | |
Title:
|
PHARMACEUTICAL COMPOSITION AND ADMINISTRATIONS THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
07/09/2013
|
Application #:
|
13234332
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Filing Dt:
|
09/16/2011
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Publication #:
|
|
Pub Dt:
|
06/28/2012
| | | | |
Title:
|
THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
03/26/2013
|
Application #:
|
13234634
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Filing Dt:
|
09/16/2011
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Publication #:
|
|
Pub Dt:
|
01/12/2012
| | | | |
Title:
|
Gyrase Inhibitors and Uses Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
12/24/2013
|
Application #:
|
13237303
|
Filing Dt:
|
09/20/2011
|
Publication #:
|
|
Pub Dt:
|
03/22/2012
| | | | |
Title:
|
MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
|
|
|
Patent #:
|
|
Issue Dt:
|
12/31/2013
|
Application #:
|
13238386
|
Filing Dt:
|
09/21/2011
|
Publication #:
|
|
Pub Dt:
|
01/19/2012
| | | | |
Title:
|
INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASES
|
|
|
Patent #:
|
|
Issue Dt:
|
09/03/2013
|
Application #:
|
13253196
|
Filing Dt:
|
10/05/2011
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Publication #:
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Pub Dt:
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11/01/2012
| | | | |
Title:
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[1,2,4]TRIAZOLO[4,3-f]PTERIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
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Patent #:
|
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Issue Dt:
|
10/02/2012
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Application #:
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13253322
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Filing Dt:
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10/05/2011
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Publication #:
|
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Pub Dt:
|
03/15/2012
| | | | |
Title:
|
C-MET PROTEIN KINASE INHIBITORS
|
|
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Patent #:
|
|
Issue Dt:
|
02/05/2013
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Application #:
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13275551
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Filing Dt:
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10/18/2011
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Publication #:
|
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Pub Dt:
|
06/14/2012
| | | | |
Title:
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KINASE INHIBITORS
|
|
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Patent #:
|
|
Issue Dt:
|
04/01/2014
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Application #:
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13280670
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Filing Dt:
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10/25/2011
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Publication #:
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Pub Dt:
|
06/21/2012
| | | | |
Title:
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COMPOUNDS USEFUL AS INHIBITORS OF JANUS KINASES
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Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
13289300
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Filing Dt:
|
11/04/2011
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Publication #:
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Pub Dt:
|
07/05/2012
| | | | |
Title:
|
4 SUBSTITUTED PYRAZOLOPYRIMIDINES
|
|
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Patent #:
|
|
Issue Dt:
|
09/24/2013
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Application #:
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13289320
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Filing Dt:
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11/04/2011
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Publication #:
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Pub Dt:
|
07/12/2012
| | | | |
Title:
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PYRAZOLOPYRIDINES
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Patent #:
|
|
Issue Dt:
|
08/06/2013
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Application #:
|
13294635
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Filing Dt:
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11/11/2011
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Publication #:
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Pub Dt:
|
03/08/2012
| | | | |
Title:
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METHOD FOR IDENTIFYING PROTEASE INHIBITORS
|
|
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Patent #:
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|
Issue Dt:
|
09/22/2015
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Application #:
|
13308609
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Filing Dt:
|
12/01/2011
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Publication #:
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Pub Dt:
|
07/19/2012
| | | | |
Title:
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PYRAZOLOPYRIDINE KINASE INHIBITORS
|
|
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Patent #:
|
|
Issue Dt:
|
10/22/2013
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Application #:
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13308612
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Filing Dt:
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12/01/2011
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Publication #:
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Pub Dt:
|
07/19/2012
| | | | |
Title:
|
TRI-CYCLIC PYRAZOLOPYRIDINE KINASE INHIBITORS
|
|
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Patent #:
|
|
Issue Dt:
|
10/16/2012
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Application #:
|
13309117
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Filing Dt:
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12/01/2011
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Publication #:
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Pub Dt:
|
03/29/2012
| | | | |
Title:
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CASPASE INHIBITORS AND USES THEREOF
|
|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
13322006
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Filing Dt:
|
02/08/2012
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Publication #:
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|
Pub Dt:
|
05/24/2012
| | | | |
Title:
|
METHOD OF MONITORING ERYTHROPOIESIS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/25/2012
|
Application #:
|
13325089
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Filing Dt:
|
12/14/2011
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Publication #:
|
|
Pub Dt:
|
07/26/2012
| | | | |
Title:
|
PYRIDONES USEFUL AS INHIBITORS OF KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
12/03/2013
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Application #:
|
13347926
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Filing Dt:
|
01/11/2012
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Publication #:
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|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3,4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
07/09/2013
|
Application #:
|
13349789
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Filing Dt:
|
01/13/2012
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Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
GYRASE AND TOPOISOMERASE IV INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/09/2013
|
Application #:
|
13349845
|
Filing Dt:
|
01/13/2012
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Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
SOLID FORMS OF GYRASE INHIBITOR (R)-1-ETHYL-3-[5-[2-(1-HYDROXY-1-METHYL-ETHYL)PYRIMIDIN-5-YL]-7-(TETRAHYDROFURAN-2-YL)-1H-BENZIMIDAZOL-2-YL]UREA
|
|
|
Patent #:
|
|
Issue Dt:
|
06/18/2013
|
Application #:
|
13349868
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Filing Dt:
|
01/13/2012
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Publication #:
|
|
Pub Dt:
|
08/09/2012
| | | | |
Title:
|
ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE
|
|
|
Patent #:
|
|
Issue Dt:
|
06/25/2013
|
Application #:
|
13349884
|
Filing Dt:
|
01/13/2012
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Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
PROCESS OF MAKING GYRASE AND TOPOISOMERASE IV INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/02/2013
|
Application #:
|
13349984
|
Filing Dt:
|
01/13/2012
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Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
SOLID FORMS OF GYRASE INHIBITOR (R)-1-ETHYL-3-[6-FLUORO-5-[2-(1-HYDROXY-1-METHYL-ETHYL)PYRIMIDIN-5-YL]-7-(TETRAHYDROFURAN-2-YL)-1H-BENZIMIDAZOL-2-YL]UREA
|
|
|
Patent #:
|
|
Issue Dt:
|
11/26/2013
|
Application #:
|
13351573
|
Filing Dt:
|
01/17/2012
|
Publication #:
|
|
Pub Dt:
|
07/26/2012
| | | | |
Title:
|
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/15/2013
|
Application #:
|
13356924
|
Filing Dt:
|
01/24/2012
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/02/2013
|
Application #:
|
13358778
|
Filing Dt:
|
01/26/2012
|
Publication #:
|
|
Pub Dt:
|
08/23/2012
| | | | |
Title:
|
SOLID FORMS OF N-[2,4-BIS(1,1-DIMETHYLETHYL)-5-HYDROXYPHENYL]-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXAMIDE
|
|
|
Patent #:
|
|
Issue Dt:
|
12/23/2014
|
Application #:
|
13364586
|
Filing Dt:
|
02/02/2012
|
Publication #:
|
|
Pub Dt:
|
08/02/2012
| | | | |
Title:
|
PYRROLOPYRAZINE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
08/20/2019
|
Application #:
|
13398184
|
Filing Dt:
|
02/16/2012
|
Publication #:
|
|
Pub Dt:
|
09/27/2012
| | | | |
Title:
|
CHROMAN-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/01/2013
|
Application #:
|
13402519
|
Filing Dt:
|
02/22/2012
|
Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
HETEROCYCLIC DERIVATIVES AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
13403169
|
Filing Dt:
|
02/23/2012
|
Publication #:
|
|
Pub Dt:
|
12/13/2012
| | | | |
Title:
|
DEAZAPURINES USEFUL AS INHIBITORS OF JANUS KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
05/28/2013
|
Application #:
|
13409702
|
Filing Dt:
|
03/01/2012
|
Publication #:
|
|
Pub Dt:
|
06/28/2012
| | | | |
Title:
|
AZAINDOLES USEFUL AS INHIBITORS OF JANUS KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
01/29/2013
|
Application #:
|
13413327
|
Filing Dt:
|
03/06/2012
|
Publication #:
|
|
Pub Dt:
|
06/28/2012
| | | | |
Title:
|
SOLID FORMS OF N-[2,4-BIS(1,1-DIMETHYLETHYL)-5-HYDROXYPHENYL]-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXAMIDE
|
|
|
Patent #:
|
|
Issue Dt:
|
06/11/2013
|
Application #:
|
13416157
|
Filing Dt:
|
03/09/2012
|
Publication #:
|
|
Pub Dt:
|
10/11/2012
| | | | |
Title:
|
Process for Preparing Azabicyclic Compounds
|
|
|
Patent #:
|
|
Issue Dt:
|
09/09/2014
|
Application #:
|
13418737
|
Filing Dt:
|
03/13/2012
|
Publication #:
|
|
Pub Dt:
|
10/18/2012
| | | | |
Title:
|
MORPHOLINE-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
13418927
|
Filing Dt:
|
03/13/2012
|
Publication #:
|
|
Pub Dt:
|
10/11/2012
| | | | |
Title:
|
Pharmaceutical Composition and Administrations Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
11/13/2012
|
Application #:
|
13419936
|
Filing Dt:
|
03/14/2012
|
Publication #:
|
|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
PIPERIDINE AND PIPERAZINE PHENYL SULPHONAMIDES AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/28/2014
|
Application #:
|
13424736
|
Filing Dt:
|
03/20/2012
|
Publication #:
|
|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
METHODS FOR PREPARING PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/03/2013
|
Application #:
|
13439379
|
Filing Dt:
|
04/04/2012
|
Publication #:
|
|
Pub Dt:
|
08/16/2012
| | | | |
Title:
|
MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
|
|
|
Patent #:
|
|
Issue Dt:
|
11/04/2014
|
Application #:
|
13440981
|
Filing Dt:
|
09/04/2012
|
Publication #:
|
|
Pub Dt:
|
04/18/2013
| | | | |
Title:
|
AMINOPYRAZINES AS ATR KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
08/06/2013
|
Application #:
|
13441287
|
Filing Dt:
|
04/06/2012
|
Publication #:
|
|
Pub Dt:
|
10/11/2012
| | | | |
Title:
|
AZAINDOLES USEFUL AS INHIBITORS OF JAK AND OTHER PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
06/03/2014
|
Application #:
|
13442244
|
Filing Dt:
|
04/09/2012
|
Publication #:
|
|
Pub Dt:
|
08/23/2012
| | | | |
Title:
|
KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/19/2013
|
Application #:
|
13450303
|
Filing Dt:
|
04/18/2012
|
Publication #:
|
|
Pub Dt:
|
08/09/2012
| | | | |
Title:
|
MODULAR TEST TUBE RACK
|
|
|
Patent #:
|
|
Issue Dt:
|
06/11/2013
|
Application #:
|
13450805
|
Filing Dt:
|
04/19/2012
|
Publication #:
|
|
Pub Dt:
|
08/09/2012
| | | | |
Title:
|
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/18/2014
|
Application #:
|
13452758
|
Filing Dt:
|
04/20/2012
|
Publication #:
|
|
Pub Dt:
|
10/24/2013
| | | | |
Title:
|
Solid Forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide
|
|
|
Patent #:
|
|
Issue Dt:
|
04/02/2013
|
Application #:
|
13453193
|
Filing Dt:
|
04/23/2012
|
Publication #:
|
|
Pub Dt:
|
01/17/2013
| | | | |
Title:
|
MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
|
|
|
Patent #:
|
|
Issue Dt:
|
11/11/2014
|
Application #:
|
13457855
|
Filing Dt:
|
04/27/2012
|
Publication #:
|
|
Pub Dt:
|
08/16/2012
| | | | |
Title:
|
ION CHANNEL MODULATORS AND METHODS OF USE
|
|
|
Patent #:
|
|
Issue Dt:
|
02/18/2014
|
Application #:
|
13467185
|
Filing Dt:
|
05/09/2012
|
Publication #:
|
|
Pub Dt:
|
11/01/2012
| | | | |
Title:
|
SOLID FORMS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACID
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
13475388
|
Filing Dt:
|
05/18/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
Modulators of ATP-Binding Cassette Transporters
|
|
|
Patent #:
|
|
Issue Dt:
|
09/10/2013
|
Application #:
|
13477663
|
Filing Dt:
|
05/22/2012
|
Publication #:
|
|
Pub Dt:
|
12/06/2012
| | | | |
Title:
|
5-CYANO-4- (PYRROLO [2,3B] PYRIDINE-3-YL) -PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/13/2012
|
Application #:
|
13478538
|
Filing Dt:
|
05/23/2012
|
Publication #:
|
|
Pub Dt:
|
09/20/2012
| | | | |
Title:
|
COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
|
|