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Patent #:
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Issue Dt:
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02/09/1999
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Application #:
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08935274
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Filing Dt:
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09/22/1997
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Title:
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2,3-DIHYDRO-1H-ISOINDOL DERIVATIVES
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Patent #:
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Issue Dt:
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02/09/1999
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Application #:
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08935275
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Filing Dt:
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09/22/1997
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Title:
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2,3-DIHYDRO-1H-ISOINDOLE DERIVATIVES AND THEIR USE AS SEROTONIN REUPTAKE INHIBITORS
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Patent #:
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Issue Dt:
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02/23/1999
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Application #:
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08935279
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Filing Dt:
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09/22/1997
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Title:
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2,3-DIHYDRO-1H-ISOINDOLE DERIVATIVES AND THEIR USE AS SEROTONIN REUPTAKE INHIBITORS
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Patent #:
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Issue Dt:
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02/23/1999
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Application #:
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08935280
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Filing Dt:
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09/22/1997
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Title:
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2,3-DIHYDRO-1H-ISOINDOLEDERIVATIVES
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Patent #:
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Issue Dt:
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01/05/1999
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Application #:
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08943460
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Filing Dt:
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10/03/1997
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Title:
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PHARMACEUTICAL COMPOSITIONS FOR PIPERIDINALKANOL COMPOUNDS
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Patent #:
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Issue Dt:
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08/03/1999
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Application #:
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08948005
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Filing Dt:
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10/09/1997
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Title:
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PHARMACEUTICAL COMPOSITION FOR PIPERIDINOALKANOL COMPOUNDS
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Patent #:
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Issue Dt:
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12/21/1999
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Application #:
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08959789
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Filing Dt:
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10/29/1997
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Title:
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N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS
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Patent #:
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Issue Dt:
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09/07/1999
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Application #:
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08961298
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Filing Dt:
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10/30/1997
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Title:
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PYRIDINIMINYL-1,2-BENZISOXAZOLES AND -BENZISOTHIAZOLES
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Patent #:
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Issue Dt:
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01/12/1999
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Application #:
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08966837
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Filing Dt:
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11/10/1997
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Title:
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PROCESSES FOR PREPARING INTERMEDIATES OF INHIBITORS OF ENKEPHALINASE AND ANGIOTENSIN CONVERTING ENZYME AND INTERMEDIATES THEREOF
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Patent #:
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Issue Dt:
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02/16/1999
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Application #:
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08966838
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Filing Dt:
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11/10/1997
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Title:
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PROCESS FOR PREPARING INTERMEDIATES OF INHIBITORS OF ENKEPHALINASE AND ANGIOTENSIN CONVERTING ENZYME AND INTERMEDIATES THEREOF
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Patent #:
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Issue Dt:
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12/15/1998
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Application #:
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08967075
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Filing Dt:
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11/10/1997
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Title:
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PROCESSES FOR PREPARING INTERMEDIATES OF INHIBITORS OF ENKEPHALINASE AND ANGIOTENSIN CONVERTING ENZYME AND INTERMEDIATES THEREOF
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Patent #:
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Issue Dt:
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11/02/1999
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Application #:
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08971891
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Filing Dt:
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11/17/1997
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Title:
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NOVEL CARBOXYSUBSTITUTED CYCLIC CARBOXAMIDE DERIVATIVES
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Patent #:
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Issue Dt:
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09/05/2000
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Application #:
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08974112
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Filing Dt:
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11/19/1997
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Title:
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SUBSTITUTED PHENOLS AND THIOPHENOLS USEFUL AS ANTIOXIDANT AGENTS
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Patent #:
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Issue Dt:
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06/29/1999
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Application #:
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08975086
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Filing Dt:
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11/20/1997
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Title:
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TRANS CYCLOPENTANYL DEAZAADENYL ANALOGS USEFUL AS IMMUNOSUPPRESSANTS
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Patent #:
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Issue Dt:
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07/27/1999
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Application #:
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08975088
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Filing Dt:
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11/20/1997
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Title:
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NOVEL TRANS CYCLOPENTANYL AZAADENYL ANALOGS USEFUL AS IMMUNOSUPRESSANT S
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Patent #:
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Issue Dt:
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05/18/1999
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Application #:
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08975552
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Filing Dt:
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11/20/1997
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Title:
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TRANS CYCLOPENTANYL DEAZAADENYL ANALOGS USEFUL AS IMMUNOSUPRESSANTS
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Patent #:
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Issue Dt:
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03/07/2000
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Application #:
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08978567
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Filing Dt:
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11/26/1997
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Title:
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PROCESS FOR CONVERTING HYDROXY HETEROAROMATICS TO ARYLAMINES
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Patent #:
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Issue Dt:
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01/19/1999
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Application #:
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08990672
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Filing Dt:
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12/15/1997
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Title:
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NOVEL HETEROCYCLIC SUBSTITUTED PYRROLIDINE AMIDE DERIVATIVES
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Patent #:
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Issue Dt:
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11/09/1999
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Application #:
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08990673
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Filing Dt:
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12/15/1997
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Title:
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HETEROCYCLE SUBSTITUTED PROPENOIC ACID DERIVATIVES AS NMDA ANTAGONIST
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Patent #:
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Issue Dt:
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12/21/1999
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Application #:
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09010720
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Filing Dt:
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01/22/1998
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Title:
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4-PIPERIDINYL) H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS
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Patent #:
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Issue Dt:
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02/08/2000
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Application #:
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09026323
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Filing Dt:
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02/19/1998
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Title:
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USE OF (+)-A-(2,3-DIMETHOXYPHENYL-1-{2-(4-FLUOROPHENYL)ETHYL}-4- PIPERIDINEMETHANOL IN TREATING DEPRESSIVE DISORDERS AND BIPOLAR DISORDERS
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Patent #:
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Issue Dt:
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12/30/2003
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Application #:
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09027258
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Filing Dt:
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02/20/1998
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Title:
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IMPROVED ASSAYS FOR BETA-AMYLOID PROCESSING
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Patent #:
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Issue Dt:
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11/16/1999
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Application #:
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09035276
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Filing Dt:
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03/09/1998
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Title:
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SPIRO[CYCLOPENT[B]INDOLE-PIPERIDINES]
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Patent #:
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Issue Dt:
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01/26/1999
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Application #:
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09067386
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Filing Dt:
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04/27/1998
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Title:
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HETEROCYCLIC SUBSTIUED PIPERAZINONE DERIVATIVES
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Patent #:
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Issue Dt:
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12/21/1999
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Application #:
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09076433
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Filing Dt:
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05/12/1998
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Title:
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NOVEL TRIPTOLIDE DERIVATIVES USEFUL IN THE TREATMENT OF AUTOIMMUNE DISEASES
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Patent #:
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Issue Dt:
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10/26/1999
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Application #:
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09076591
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Filing Dt:
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05/12/1998
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Title:
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NOVEL TRIPTOLIDE DERIVATIVES USEFUL IN THE TREATMENT OF AUTOIMMUNE DISEASES
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Patent #:
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Issue Dt:
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09/28/1999
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Application #:
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09079331
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Filing Dt:
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05/14/1998
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Title:
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PROCESS FOR PREPARING 6-O-MONOESTERS OF CASTANOSPERMINE
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Patent #:
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Issue Dt:
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03/29/2005
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Application #:
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09082038
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Filing Dt:
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05/20/1998
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Publication #:
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Pub Dt:
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04/10/2003
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Title:
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THREE-DIMENSIONAL ARRAY OF SUPPORTS FOR SOLID-PHASE PARALLEL SYNTHESIS AND METHOD OF USE
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Patent #:
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Issue Dt:
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10/17/2000
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Application #:
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09103215
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Filing Dt:
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06/23/1998
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Title:
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2,6-DI-T-BUTYL-4-[DIMETHYL-4-METHOXYPHENYLSILYL)-METHYL-OXY]PHENOL AND 2,6-DI-T-BUTYL-4-[DIMETHYL-2-METHOXY-PHENYLSILYL)METHYLOXY]PHENOL
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Patent #:
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Issue Dt:
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03/21/2000
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Application #:
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09127478
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Filing Dt:
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07/31/1998
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Title:
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PHARMACEUTICAL COMPOSITION FOR COMBINAITON OF PIPERIDINOALKANOL-DECONGESTANT
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Patent #:
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Issue Dt:
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09/05/2000
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Application #:
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09157841
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Filing Dt:
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09/21/1998
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Title:
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PHARMACEUTICAL COMPOSITION FOR PIPERIDINOALKANOL COMPOUNDS
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Patent #:
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Issue Dt:
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07/02/2002
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Application #:
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09247052
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Filing Dt:
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02/09/1999
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Title:
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6,9,-DISUBSTITUTED 2-[TRANS-(4-AMINOCYCLOHEXYL) AMINO] PURINES
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Patent #:
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Issue Dt:
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11/12/2002
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Application #:
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09247053
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Filing Dt:
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02/09/1999
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Title:
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6,9-DISUBSTITUTED 2-[TRANS-(4-AMINOCYCLOHEXYL)AMINO] PURINES
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Patent #:
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Issue Dt:
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12/28/1999
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Application #:
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09288388
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Filing Dt:
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04/08/1999
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Title:
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ANTIPSYCHOTIC AGENTS, COMPOSITIONS AND METHOD OF USE
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Patent #:
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Issue Dt:
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09/11/2001
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Application #:
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09314534
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Filing Dt:
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05/19/1999
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Title:
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PROFILE SEARCHING IN NUCLEIC ACID SEQUENCES USING THE FAST FOURIER TRANSFORMATION
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Patent #:
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Issue Dt:
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12/05/2000
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Application #:
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09333372
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Filing Dt:
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06/15/1999
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Title:
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SPIRO(CYCLOPENT(B)INDOLE-PIPERIDINES)
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Patent #:
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Issue Dt:
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05/16/2000
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Application #:
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09337957
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Filing Dt:
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06/22/1999
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Title:
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ESTERS OF (+)-A-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL)ETHYL)-4-PIPERIDINEME THANOL
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Patent #:
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Issue Dt:
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01/30/2001
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Application #:
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09363305
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Filing Dt:
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07/28/1999
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Title:
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HETEROCYCLE SUBSTITUTED PROPENOIC ACID DERIVATIVES AS NMDA ANTAGONIST
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Patent #:
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Issue Dt:
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08/21/2001
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Application #:
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09382932
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Filing Dt:
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08/25/1999
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Title:
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USE OF R (+)-ALPHA-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL) ETHYL]-4-PIPERIDINEMETHANOL FOR THE TREATMENT OF SLEEP DISORDERS
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Patent #:
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Issue Dt:
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04/01/2003
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Application #:
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09449222
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Filing Dt:
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11/24/1999
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Title:
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APPARATUS AND METHOD FOR SYNTHESIZING COMBINATIONAL LIBRARIES
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Patent #:
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Issue Dt:
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09/24/2002
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Application #:
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09454555
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Filing Dt:
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12/07/1999
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Title:
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BIODEGRADABLE POLYMER ENCAPSULATED PHARMACEUTICAL COMPOSITIONS AND METHOD FOR PREPARING THE SAME
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Patent #:
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Issue Dt:
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11/12/2002
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Application #:
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09459046
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Filing Dt:
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12/10/1999
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Title:
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AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS
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Patent #:
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Issue Dt:
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12/11/2001
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Application #:
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09464907
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Filing Dt:
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12/17/1999
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Title:
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AMIDOMALONAMIDES USEFUL AS INHIBITORS OF MMP OF MATRIX METALLOPROTEINASE
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Patent #:
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Issue Dt:
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03/05/2002
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Application #:
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09464908
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Filing Dt:
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12/17/1999
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Title:
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SELECTIVE INHIBITORS OF MMP-12
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Patent #:
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Issue Dt:
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02/27/2001
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Application #:
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09513847
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Filing Dt:
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10/29/1997
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Title:
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NOVEL SUBSTITUTED 4-(1H-BENZIMIDAZOL-2YL)[1,4]DIAZEPANES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASE
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Patent #:
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Issue Dt:
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12/31/2002
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Application #:
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09577634
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Filing Dt:
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05/24/2000
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Title:
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MATHEMATICAL ANALYSIS FOR THE ESTIMATION OF CHANGES IN THE LEVEL OF GENE EXPRESSION
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Patent #:
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Issue Dt:
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04/29/2003
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Application #:
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09589462
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Filing Dt:
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06/07/2000
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Title:
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SCREENING METHODS FOR ALTERING CIRCADIAN RHYTHMS AND FOR HUMAN CASEIN KINASE I D AND/OR E PHOSPHORYLATION OF HUMAN CLOCK PROTEINS, PERIOD 1, -2 AND -3
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Patent #:
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Issue Dt:
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10/15/2002
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Application #:
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09615246
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Filing Dt:
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07/13/2000
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Title:
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SULFURIC ACID MONO-[3({1-[2-(4-FLUORO-PHENYL)-ETHYL]-PIPERIDIN
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Patent #:
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Issue Dt:
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05/08/2001
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Application #:
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09624477
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Filing Dt:
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07/24/2000
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Title:
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Spiro[cyclopent[b]indole-piperidines]
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Patent #:
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Issue Dt:
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11/13/2001
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Application #:
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09648005
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Filing Dt:
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05/06/1999
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Title:
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Novel carboxy substituted acylic carboxamide derivatives
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Patent #:
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Issue Dt:
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04/30/2002
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Application #:
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09699647
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Filing Dt:
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10/30/2000
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Title:
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USE OF (+) -ALPHA- (2, 3-DIMETHOXYPHENYL) - 1 - [ 2 - ( 4 - FLUOROPHENYL) ETHYL ] -4 - PIPERIDINEMETHANOL IN TREATING DEPRESSIVE DISORDERS AND BIPOLAR DISORDERS
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Patent #:
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Issue Dt:
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07/18/2006
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Application #:
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09712129
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Filing Dt:
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11/15/2000
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Title:
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HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS
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Patent #:
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Issue Dt:
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07/18/2006
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Application #:
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09712129
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Filing Dt:
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11/15/2000
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Title:
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HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS
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Patent #:
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Issue Dt:
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02/17/2004
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Application #:
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09741536
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Filing Dt:
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12/20/2000
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Publication #:
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Pub Dt:
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05/22/2003
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Title:
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NOVEL ELASTASE INHIBITORS
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Patent #:
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Issue Dt:
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06/10/2003
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Application #:
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09760589
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Filing Dt:
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01/16/2001
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Publication #:
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Pub Dt:
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03/06/2003
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Title:
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PSEUDOPOLYMORPH OF ( - ) -CIS -2-(2 -CHLOROPHENYL) -5, 7-DIHYDROXY-8 [4R- ( 3S-HYDROXY -1-METHYL)PIPERIDINYL ] -4H -1 -BENZOPYRAN-4-ONE
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11/23/2004
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09760590
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Filing Dt:
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01/16/2001
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Publication #:
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Pub Dt:
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12/13/2001
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Title:
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ETHANOL SOLVATE OF (-)-CIS-2- (2-CHLOROPHENYL)-5, 7-DIHYDROXY-8 [4R-(3S-HYDROXY-1-M ETHYL) PIPERIDINYL} -4H-1-BENZOPYRAN-4-ONE
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11/12/2002
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09768666
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01/24/2001
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01/10/2002
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Title:
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SPIRO[CYCLOPENT[B]INDOLE-PIPERIDINES]
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Issue Dt:
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11/26/2002
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Application #:
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09815868
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03/23/2001
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Publication #:
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Pub Dt:
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03/28/2002
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Title:
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3-SUBSTITUTED PYRROLIDINES USEFUL AS INHIBITORS OF MATRIX METALLOPROTEINASES
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Patent #:
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Issue Dt:
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09/02/2003
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Application #:
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09886424
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Filing Dt:
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06/21/2001
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Publication #:
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Pub Dt:
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11/15/2001
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Title:
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THE USE OF R (+)-ALPHA- (2,3-DIMETHOXYPHENYL) -1- [ 2- (4-FLUOROPHENYL) ETHYL] -4-PIPER IDINEMETHANOL FOR THE TREATMENT OF SLEEP DISORDERS
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Patent #:
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01/11/2005
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Application #:
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09950931
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09/12/2001
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Publication #:
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Pub Dt:
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02/21/2002
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Title:
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PROFILE SEARCHING IN NUCLEIC ACID SEQUENCES USING THE FAST FOURIER TRANSFORMATION
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Patent #:
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Issue Dt:
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09/19/2006
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Application #:
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10031922
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Filing Dt:
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05/13/2002
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Title:
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PRESERVED PHARMACEUTICAL FORMULATIONS
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Patent #:
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Issue Dt:
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03/30/2004
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Application #:
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10043498
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Filing Dt:
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01/11/2002
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Publication #:
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Pub Dt:
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10/17/2002
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Title:
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NOVEL PROCESSES FOR THE PREPARATION OR (R)-ALPHA-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL)ETHYL]-4-PIPERIDINEMETHANOL
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Patent #:
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Issue Dt:
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10/24/2006
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Application #:
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10088250
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Filing Dt:
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12/23/2002
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Title:
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THIENOISOXAZOLYL-AND THIENYLPYRRAZOLYL-PHENOXY SUBSTITUTED PROPYL DERIVATIVES USEFUL AS D4 ANTAGONISTS
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Patent #:
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Issue Dt:
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08/15/2006
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Application #:
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10088369
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Filing Dt:
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12/23/2002
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Title:
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THIENOISOXAZOLE PHENOXY UNSUBSTITUTED ETHYL AND PROPYL DERIVATIVES USEFUL AS D4 ANTAGONISTS
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Issue Dt:
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08/16/2005
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10104097
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03/22/2002
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Publication #:
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Pub Dt:
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08/15/2002
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Title:
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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Patent #:
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Issue Dt:
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05/04/2004
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Application #:
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10104149
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Filing Dt:
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03/22/2002
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Publication #:
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Pub Dt:
|
07/25/2002
| | | | |
Title:
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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|
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Patent #:
|
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Issue Dt:
|
01/06/2004
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Application #:
|
10104277
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Filing Dt:
|
03/22/2002
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Publication #:
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Pub Dt:
|
07/25/2002
| | | | |
Title:
|
NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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|
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Patent #:
|
|
Issue Dt:
|
03/02/2004
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Application #:
|
10104311
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Filing Dt:
|
03/22/2002
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Publication #:
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|
Pub Dt:
|
07/25/2002
| | | | |
Title:
|
NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
|
|
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Patent #:
|
|
Issue Dt:
|
02/10/2004
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Application #:
|
10104783
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Filing Dt:
|
03/22/2002
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Publication #:
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Pub Dt:
|
07/25/2002
| | | | |
Title:
|
NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
11/14/2006
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Application #:
|
10160883
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Filing Dt:
|
06/03/2002
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Publication #:
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Pub Dt:
|
12/19/2002
| | | | |
Title:
|
PROCESSES FOR PREPARING ANHYDROUS AND HYDRATE FORMS OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES, POLYMORPHS AND PSEUDOMORPHS THEREOF
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|
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Patent #:
|
|
Issue Dt:
|
11/21/2006
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Application #:
|
10162011
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Filing Dt:
|
06/03/2002
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Publication #:
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Pub Dt:
|
12/19/2002
| | | | |
Title:
|
PROCESSES FOR PREPARING ANHYDROUS AND HYDRATE FORMS OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES, POLYMORPHS AND PSEUDOMORPHS THEREOF
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|
|
Patent #:
|
|
Issue Dt:
|
01/27/2004
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Application #:
|
10170050
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Filing Dt:
|
06/12/2002
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Publication #:
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Pub Dt:
|
01/30/2003
| | | | |
Title:
|
NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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|
|
Patent #:
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|
Issue Dt:
|
11/04/2003
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Application #:
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10178494
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Filing Dt:
|
06/24/2002
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Publication #:
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Pub Dt:
|
06/05/2003
| | | | |
Title:
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6,9-DISUBSTITUTED 2-[TRANS-(4-AMINOCYCLOHEXYL) AMINO] PURINES
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Patent #:
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Issue Dt:
|
04/06/2004
|
Application #:
|
10200821
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Filing Dt:
|
07/22/2002
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Publication #:
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|
Pub Dt:
|
05/08/2003
| | | | |
Title:
|
SULFURIC ACID MONO-[ 3- ( {1- [ 2- (4-FLUORO-PHENYL ) -ETHYL ] -PIPERIDIN-4-YL} -HYDROXY-METHYL) -2-METHOXY-PHENYL ] ESTER
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Patent #:
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Issue Dt:
|
10/17/2006
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Application #:
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10316353
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Filing Dt:
|
12/11/2002
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Publication #:
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|
Pub Dt:
|
10/23/2003
| | | | |
Title:
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APPARATUS AND METHOD FOR SYNTHESIZING COMBINATORIAL LIBRARIES
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Patent #:
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Issue Dt:
|
09/06/2005
|
Application #:
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10609751
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Filing Dt:
|
06/30/2003
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Publication #:
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Pub Dt:
|
01/01/2004
| | | | |
Title:
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Use of R (+)-alpha-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol for the treatment of substance induced insomnia
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Patent #:
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Issue Dt:
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03/31/2009
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Application #:
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11459068
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Filing Dt:
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07/21/2006
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Publication #:
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Pub Dt:
|
01/04/2007
| | | | |
Title:
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THIENOISOXAZOLYL-AND THIENYLPYRRAZOLYL PHENOXY SUBSTITUTED PROPYL DERIVATIVES USEFUL AS D4 ANTAGONISTS
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Patent #:
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Issue Dt:
|
02/23/2010
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Application #:
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11534828
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Filing Dt:
|
09/25/2006
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Publication #:
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Pub Dt:
|
01/25/2007
| | | | |
Title:
|
METHODS OF TREATING ALLERGIC REACTIONS USING HYDRATED FORMS OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES
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Patent #:
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Issue Dt:
|
02/16/2010
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Application #:
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11534839
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Filing Dt:
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09/25/2006
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Publication #:
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Pub Dt:
|
01/25/2007
| | | | |
Title:
|
METHODS OF TREATING ALLERGIC REACTIONS USING AN ANHYDROUS FORM OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES
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|
Patent #:
|
NONE
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Issue Dt:
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Application #:
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11553751
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Filing Dt:
|
10/27/2006
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Publication #:
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Pub Dt:
|
06/07/2007
| | | | |
Title:
|
PROCESSES FOR PREPARING ANHYDROUS AND HYDRATE FORMS OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES, POLYMORPHS AND PSEUDOMORPHS THEREOF
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Patent #:
|
NONE
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Issue Dt:
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Application #:
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11972749
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Filing Dt:
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01/11/2008
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Publication #:
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Pub Dt:
|
05/08/2008
| | | | |
Title:
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Ethanol Solvate of (-)-cis-2-(2-chlorophenyl)-5,7-dihydroxy-8-[4R-(3S-hydroxy-1-methyl)piperidinyl]-4H-1-benzopyran-4-one
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Patent #:
|
NONE
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Issue Dt:
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Application #:
|
11978669
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Filing Dt:
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10/30/2007
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Publication #:
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Pub Dt:
|
07/10/2008
| | | | |
Title:
|
A HYDRATED FORM OF AN ANTHISTAMINIC PIPERIDINE DERIVATIVE AND METHODS OF MAKING A HYDRATED FORM OF AN ANTHIHISTAMINIC PIPERIDINE DERIVATIVE
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Patent #:
|
NONE
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Issue Dt:
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Application #:
|
11978670
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Filing Dt:
|
10/30/2007
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Publication #:
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Pub Dt:
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07/10/2008
| | | | |
Title:
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Processes for preparing anhydrous and hydrate forms of antihistaminic piperidine derivatives, polymorphs and pseudomorphs thereof
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Patent #:
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Issue Dt:
|
03/06/2012
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Application #:
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12565410
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Filing Dt:
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09/23/2009
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Publication #:
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Pub Dt:
|
01/28/2010
| | | | |
Title:
|
PHARMACEUTICAL COMPOSITION FOR PIPERIDINOALKANOL COMPOUNDS
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