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Patent #:
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Issue Dt:
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10/03/1989
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Application #:
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07247797
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Filing Dt:
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09/22/1988
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Title:
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SUBSTITUTED IMIDAZO(2,1-B)QUINAZOLIN-5(3H)-ONES AND RELATED TRICYCLIC COMPOUNDS AND USE AS BRONCHODILATORS
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Patent #:
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Issue Dt:
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09/26/1989
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Application #:
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07254208
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Filing Dt:
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10/11/1988
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Title:
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1,4-DISUBSTITUTED-PIPERIDINYL COMPOUNDS USEFUL AS ANALGESIS AND MUSCLE RELAXANTS
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Patent #:
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Issue Dt:
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03/13/1990
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Application #:
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07299913
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Filing Dt:
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01/19/1989
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Title:
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USE OF 1,4-DISUBSTITUTED-PIPERIDINYL COMPOUNDS IN THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF INSOMNIA
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Patent #:
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Issue Dt:
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03/05/1991
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Application #:
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07380068
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Filing Dt:
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07/14/1989
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Title:
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5'-DEOXY-5',5'-DIHALO-ADENOSINES AND PURINE ANALOGUES
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Patent #:
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Issue Dt:
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04/30/1991
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Application #:
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07527676
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Filing Dt:
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05/16/1990
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Title:
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MEDICAMENT COMPOSITIONS DERIVED FROM QUINOLIZINE AND QUINOLIZINONE AND USE THEREOF
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Patent #:
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Issue Dt:
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12/20/1994
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Application #:
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07759568
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Filing Dt:
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09/13/1991
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Title:
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AMINO ACID SEQUENCE FOR A FUNCTIONAL HUMAN INTERLEUKIN-8 RECEPTOR
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Patent #:
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Issue Dt:
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05/04/1993
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Application #:
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07905494
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Filing Dt:
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06/25/1992
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Title:
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NOVEL AMINO AND NITRO CONTAINING TRICYCLIC COMPOUNDS USEFUL AS INHIBITORS OF ACE
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Patent #:
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Issue Dt:
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11/30/1993
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Application #:
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07922130
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Filing Dt:
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07/29/1992
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Title:
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SUGAR-FREE DRY MIX CELLULOSE ETHER COMPOSITIONS AS BULK LAXATIVES
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Patent #:
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Issue Dt:
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11/15/1994
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Application #:
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07969383
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Filing Dt:
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10/30/1992
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Title:
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HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALETICS
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Patent #:
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Issue Dt:
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11/28/1995
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Application #:
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08068947
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Filing Dt:
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05/28/1993
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Title:
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PEPTIDE SEQUENCING USING MASS SPECTROMETRY
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Patent #:
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Issue Dt:
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10/25/1994
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Application #:
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08106311
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Filing Dt:
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08/13/1993
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Title:
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SULFONIC ACID DERIVATIVES IN THE TREATMENT OF VIRAL DISEASES
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Patent #:
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Issue Dt:
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11/27/2001
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Application #:
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08137440
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Filing Dt:
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10/15/1993
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Title:
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GALANTHAMINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS
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Patent #:
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Issue Dt:
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11/27/2001
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Application #:
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08137443
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Filing Dt:
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10/15/1993
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Title:
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GALANTHAMINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS
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Patent #:
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Issue Dt:
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11/13/2001
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Application #:
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08137444
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Filing Dt:
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10/15/1993
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Title:
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GALANTHAMINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS
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Patent #:
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Issue Dt:
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04/18/1995
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Application #:
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08194137
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Filing Dt:
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02/09/1994
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Title:
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ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS
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Patent #:
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Issue Dt:
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10/17/1995
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Application #:
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08242395
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Filing Dt:
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05/13/1994
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Title:
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PREPARATION OF N-ALKYL-N-PYRIDINYL-1H-INDOL-1-AMINES
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Patent #:
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Issue Dt:
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11/24/1998
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Application #:
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08249830
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Filing Dt:
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05/26/1994
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Title:
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TOPOLOGICALLY SEGREGATED, ENCODED SOLID PHASE LIBRARIES
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Patent #:
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Issue Dt:
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06/03/1997
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Application #:
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08263289
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Filing Dt:
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06/21/1994
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Title:
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SELECTIVELY CLEAVABLE LINKERS BASED ON IMINODIACETIC ACID ESTERS FOR SOLID PHASE PEPTIDE SYNTHESIS
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Patent #:
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Issue Dt:
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07/29/1997
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Application #:
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08273090
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Filing Dt:
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07/11/1994
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Title:
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APPARATUS AND METHOD FOR RANDOM POLYMER SYNTHESIS
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Patent #:
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Issue Dt:
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08/19/1997
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Application #:
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08309395
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Filing Dt:
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09/20/1994
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Title:
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HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS
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Patent #:
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Issue Dt:
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07/07/1998
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Application #:
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08329000
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Filing Dt:
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10/25/1994
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Title:
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3-(HETEROARYL)-1-[(2,3-DIHYDRO-1H-ISOINDOL-2-YL)ALKYL]PYRROLIDINES AND 3-(HETEROARYL)-1-[(2,3-DIHYDRO-1H-INDOL-1-YL)ALKYL]PYRROLIDINES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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11/18/1997
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Application #:
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08354199
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Filing Dt:
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12/12/1994
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Title:
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COMBINATORIAL LIBRARIES HAVING A PREDETERMINED FREQUENCY OF EACH SPECIES OF TEST COMPOUND
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Patent #:
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Issue Dt:
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03/14/2000
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Application #:
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08397542
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Filing Dt:
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03/02/1995
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Title:
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METHOD OF PROVIDING AND ANTHIHISTAMINIC EFFECT IN A HEPATICALLY IMPAIRED PATIENT
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Patent #:
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Issue Dt:
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07/02/2002
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Application #:
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08435079
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Filing Dt:
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05/08/1995
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Title:
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[1-INDANON-2-YL]METHYLPIPERIDINES
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Patent #:
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Issue Dt:
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07/01/1997
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Application #:
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08455468
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Filing Dt:
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05/31/1995
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Title:
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PREPARATION OF N-ALKYL-N-PYRIDINYL-1H-INDOL-1-AMINES
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Patent #:
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Issue Dt:
|
01/28/2003
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Application #:
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08455469
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Filing Dt:
|
05/31/1995
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Title:
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PREPARATION OF N-ALKYL-N-PYRIDINYL-1H-INDOL-1-AMINES
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Patent #:
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Issue Dt:
|
11/02/1999
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Application #:
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08465863
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Filing Dt:
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06/06/1995
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Title:
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N-[4-HETEROARYL-1-PIPERIDINYL)ALKYL]PHTHALIMIDES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
|
11/02/1999
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Application #:
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08466241
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Filing Dt:
|
06/06/1995
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Title:
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4-HETEROARYL-1-PIPERAZINEALKYLAMINES AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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12/14/1999
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Application #:
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08466252
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Filing Dt:
|
06/06/1995
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Title:
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[(4-HETEROARYL-1-PIPERAZINYL)-ALKOXY]-3,4-DIHYDOR-1(2H)NAPHTHALENONES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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03/04/1997
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Application #:
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08466821
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Filing Dt:
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06/06/1995
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Title:
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HETEROARYLPIPERIDINES, AND THEIR USE AS ANTIPSYCHOTICS AND ANALGESICO
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Patent #:
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Issue Dt:
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03/30/1999
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Application #:
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08467133
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Filing Dt:
|
06/06/1995
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Title:
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1-(ARYLTHIOALKYL, ARYLAMINOALKYL OR ARYLMETHYLENEALKYL)-3-(HETEROARYL)PYRROLIDINES AND RELATED COMPOUNDS USEFUL AS ANTIPSYCHOTICS AND ANALGESICS
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Patent #:
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Issue Dt:
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03/28/2000
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Application #:
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08467401
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Filing Dt:
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06/06/1995
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Title:
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3-HETEROARYL-1-PYRROLIDINEALKYLAMINES AND DERIVATIVES THEREOF AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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12/07/1999
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Application #:
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08468065
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Filing Dt:
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06/06/1995
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Title:
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N-[(4-HETEROARYL-1-PIPERAZINYL)ALKYL]PHTHALIMIDES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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07/06/1999
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Application #:
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08468075
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Filing Dt:
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06/06/1995
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Title:
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4-HETEROARYL-1-PIPERIDINEALKANOLS AND DERIVATIVES THEREOF AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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10/31/2000
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Application #:
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08468611
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Filing Dt:
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06/06/1995
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Title:
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1-(ARYLOXYALKYL)-4-(HETEROARYL)PIPERIDINES AND RELATED COMPOUNDS USEFUL AS ANTIPSYCHOTICS AND ANALGESICS
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Patent #:
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Issue Dt:
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09/22/1998
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Application #:
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08468991
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Filing Dt:
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06/06/1995
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Title:
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2-[(4-HETEROARYL-1-PIPERIDINYL)ALKYL]-1,3-DIOXANES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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03/25/1997
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Application #:
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08469000
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Filing Dt:
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06/06/1995
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Title:
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1-(ARYLOXYALKYL)-3- (HETEROARYL) PYRROLIDINES AND RELATED COMPOUNDS USEFUL AS ANTIPSYCHOTICS AND ANALGESICS
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Patent #:
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Issue Dt:
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01/07/1997
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Application #:
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08469365
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Filing Dt:
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06/06/1995
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Title:
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HETEROARYLPIPERIDINES AND THEIR USE AS ANTIPSYCHOTICS AND ANAGESICS
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Patent #:
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Issue Dt:
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11/12/1996
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Application #:
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08469392
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Filing Dt:
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06/06/1995
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Title:
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ORAL PHARMACEUTICAL COMPOSITION OF PIPERIDINOALKANOL COMPOUNDS IN SOLUTION FORM
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Patent #:
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Issue Dt:
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02/23/1999
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Application #:
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08470039
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Filing Dt:
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06/06/1995
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Title:
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4-HETEROARYL-1-PIPERAZINEALKANOLS AND DERIVATIVES THEREOF AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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09/02/1997
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Application #:
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08470059
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Filing Dt:
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06/06/1995
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Title:
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INTERMEDIATE COMPOUNDS IN THE SYNTHESIS OF HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES
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Patent #:
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Issue Dt:
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08/29/2000
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Application #:
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08471032
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Filing Dt:
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06/06/1995
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Title:
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1-(ARYLTHIOALKYL, ARYLAMINOALKYL OR ARYLMETHYLENEALKYL)-4-(HETEROARYL) PIPERIDINES AND RELATED COMPOUNDS USEFUL AS ANTIPSYCHOTICS AND ANALGESICS
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Patent #:
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Issue Dt:
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04/04/2000
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Application #:
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08471197
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Filing Dt:
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06/06/1995
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Title:
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SUBSTITUTED 3-(AMINOALKYLAMINO)-1,2-BENZISOXAZOLES AND RELATED COMPOUNDS
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Issue Dt:
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03/30/1999
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Application #:
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08471393
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Filing Dt:
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06/06/1995
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Title:
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4-HETEROARYL-1-PIPERAZINEALKYLTHIOLS AND DERIVATIVES THEREOF AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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10/12/1999
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Application #:
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08471512
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Filing Dt:
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06/06/1995
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Title:
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1-[(2-PYRIMIDINYLOXY)ALKYL]4-(HETEROARYL)PIPERAZINES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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Issue Dt:
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09/22/1998
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Application #:
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08471754
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Filing Dt:
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06/06/1995
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Title:
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1[(2-PYRIMIDINYLOXY)ALKYL]-4-(HETEROARYL)PIPERIDINES AND RELATED COMPOUNDS AND THEIR THERAPEUTIC UTILITY
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04/14/1998
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08742166
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11/01/1996
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Title:
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PHARMACEUTICAL COMPOSITION FOR PIPERIDINOALKANOL COMPOUNDS
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12/08/1998
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08754878
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11/22/1996
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Title:
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MOTIF LIBRARIES
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04/02/2002
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08798258
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Filing Dt:
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02/11/1997
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Title:
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4-AZA STEROIDS
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08/08/2000
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Application #:
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08806012
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Filing Dt:
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02/24/1997
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Title:
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ISATIN DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS AND ANALGESICS
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Patent #:
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Issue Dt:
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10/11/2005
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Application #:
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08893080
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07/15/1997
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Title:
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3-MERCAPTOACETYLAMINO-1,5-SUBSTITUTED-2-OXO-AZEPAN DERIVATIVES USEFUL AS INHIBITORS OF MATRIX METALLOPROTEINASE
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01/05/1999
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Application #:
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08943460
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10/03/1997
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Title:
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PHARMACEUTICAL COMPOSITIONS FOR PIPERIDINALKANOL COMPOUNDS
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08/03/1999
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Application #:
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08948005
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10/09/1997
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Title:
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PHARMACEUTICAL COMPOSITION FOR PIPERIDINOALKANOL COMPOUNDS
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10/03/2000
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08971775
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11/17/1997
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Title:
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METHOD FOR PRODUCING COMBINATORIAL LIBRARIES HAVING A PREDETERMINED FREQUENCY OF EACH SPECIES OF TEST COMPOUND
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08/20/2002
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08975212
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11/20/1997
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Title:
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NOVEL TRANS CYCLOPENTANYL PURINE ANALOGS USEFUL AS IMMUNOSUPPRESSANTS
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02/08/2000
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09026323
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02/19/1998
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Title:
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USE OF (+)-A-(2,3-DIMETHOXYPHENYL-1-{2-(4-FLUOROPHENYL)ETHYL}-4- PIPERIDINEMETHANOL IN TREATING DEPRESSIVE DISORDERS AND BIPOLAR DISORDERS
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12/30/2003
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09027258
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02/20/1998
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Title:
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IMPROVED ASSAYS FOR BETA-AMYLOID PROCESSING
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03/29/2005
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09082038
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05/20/1998
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Publication #:
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04/10/2003
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Title:
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THREE-DIMENSIONAL ARRAY OF SUPPORTS FOR SOLID-PHASE PARALLEL SYNTHESIS AND METHOD OF USE
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03/21/2000
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09127478
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07/31/1998
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Title:
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PHARMACEUTICAL COMPOSITION FOR COMBINAITON OF PIPERIDINOALKANOL-DECONGESTANT
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09/05/2000
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09157841
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09/21/1998
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Title:
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PHARMACEUTICAL COMPOSITION FOR PIPERIDINOALKANOL COMPOUNDS
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12/31/2002
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09237689
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01/26/1999
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1-ALKYL-,1-ALKENYL-,AND 1-ALKYNYLARYL-2-AMINO-1,3-PROPANEDIOLS AND RELATED COMPOUNDS
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06/04/2002
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09240842
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Filing Dt:
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02/03/1999
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Title:
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4-HETEROARYL-1-PIPERIDINEALKYLAMINES AND DERIVATIVES THEREOF AND THEIR THERAPEUTIC UTILITY
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Patent #:
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Issue Dt:
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07/02/2002
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Application #:
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09247052
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Filing Dt:
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02/09/1999
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Title:
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6,9,-DISUBSTITUTED 2-[TRANS-(4-AMINOCYCLOHEXYL) AMINO] PURINES
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Patent #:
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Issue Dt:
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11/12/2002
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Application #:
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09247053
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Filing Dt:
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02/09/1999
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Title:
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6,9-DISUBSTITUTED 2-[TRANS-(4-AMINOCYCLOHEXYL)AMINO] PURINES
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Patent #:
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Issue Dt:
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09/11/2001
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Application #:
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09314534
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Filing Dt:
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05/19/1999
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Title:
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PROFILE SEARCHING IN NUCLEIC ACID SEQUENCES USING THE FAST FOURIER TRANSFORMATION
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01/30/2001
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Application #:
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09363305
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Filing Dt:
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07/28/1999
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Title:
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HETEROCYCLE SUBSTITUTED PROPENOIC ACID DERIVATIVES AS NMDA ANTAGONIST
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Issue Dt:
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08/21/2001
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Application #:
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09382932
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Filing Dt:
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08/25/1999
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Title:
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USE OF R (+)-ALPHA-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL) ETHYL]-4-PIPERIDINEMETHANOL FOR THE TREATMENT OF SLEEP DISORDERS
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Patent #:
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04/01/2003
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Application #:
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09449222
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11/24/1999
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Title:
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APPARATUS AND METHOD FOR SYNTHESIZING COMBINATIONAL LIBRARIES
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Issue Dt:
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09/24/2002
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12/07/1999
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Title:
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11/12/2002
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12/10/1999
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12/11/2001
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12/17/1999
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Title:
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03/05/2002
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Title:
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08/03/2004
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12/17/1999
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Title:
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07/17/2001
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12/17/1999
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Title:
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12/31/2002
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04/29/2003
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Title:
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11/16/2004
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06/16/2000
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Title:
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10/15/2002
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07/13/2000
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Title:
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11/13/2001
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05/06/1999
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Novel carboxy substituted acylic carboxamide derivatives
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04/30/2002
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09699647
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10/30/2000
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Title:
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02/17/2004
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05/22/2003
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06/10/2003
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01/16/2001
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03/06/2003
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11/23/2004
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01/16/2001
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12/13/2001
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11/12/2002
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01/24/2001
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01/10/2002
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SPIRO[CYCLOPENT[B]INDOLE-PIPERIDINES]
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11/26/2002
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03/23/2001
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03/28/2002
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09/02/2003
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09886424
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06/21/2001
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11/15/2001
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01/11/2005
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09/12/2001
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02/21/2002
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09/19/2006
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05/13/2002
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03/30/2004
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10043498
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01/11/2002
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10/17/2002
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NOVEL PROCESSES FOR THE PREPARATION OR (R)-ALPHA-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL)ETHYL]-4-PIPERIDINEMETHANOL
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10/24/2006
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12/23/2002
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08/15/2006
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12/23/2002
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08/16/2005
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03/22/2002
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08/15/2002
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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05/04/2004
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10104149
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03/22/2002
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07/25/2002
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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01/06/2004
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07/25/2002
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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03/02/2004
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07/25/2002
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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02/10/2004
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07/25/2002
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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11/14/2006
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12/19/2002
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11/21/2006
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NOVEL ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF
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