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Reel/Frame:022024/0105   Pages: 9
Recorded: 12/23/2008
Attorney Dkt #:20595.001
Conveyance: CERTIFICATE OF MERGER OF GRANITE ACQUISITION, INC. WITH AND INTO GUILFORD PHARMACEUTICALS INC.
Total properties: 47
1
Patent #:
Issue Dt:
09/08/1998
Application #:
08665775
Filing Dt:
06/17/1996
Title:
METHODS OF CANCER TREATMENT USING NAALADASE INHIBITORS
2
Patent #:
Issue Dt:
09/30/1997
Application #:
08665776
Filing Dt:
06/17/1996
Title:
CERTAIN PHOSPHONOMETHYL-PENTANEDIOIC ACID DERIVATIVES THEREOF
3
Patent #:
Issue Dt:
10/20/1998
Application #:
08718703
Filing Dt:
09/27/1996
Title:
TREATMENT OF GLOBAL AND FOCAL ISCHEMIA USING NAALADASE INHIBITORS
4
Patent #:
Issue Dt:
08/18/1998
Application #:
08775586
Filing Dt:
12/31/1996
Title:
INHIBITORS OF NAALADASE ENZYME ACTIVITY
5
Patent #:
Issue Dt:
01/26/1999
Application #:
08778733
Filing Dt:
12/31/1996
Title:
PHOSPHORAMIDATE DERIVATIVES
6
Patent #:
Issue Dt:
10/05/1999
Application #:
08825997
Filing Dt:
04/04/1997
Title:
HYDROXAMIC ACID DERIVATIVES
7
Patent #:
Issue Dt:
10/19/1999
Application #:
08833628
Filing Dt:
04/08/1997
Title:
NAALADASE INHIBITORS
8
Patent #:
Issue Dt:
03/09/1999
Application #:
08833646
Filing Dt:
04/08/1997
Title:
NAALADASE INHIBITORS
9
Patent #:
Issue Dt:
05/11/1999
Application #:
08835572
Filing Dt:
04/09/1997
Title:
CERTAIN SULFOXIDE AND SULFONE DERIVATIVES
10
Patent #:
Issue Dt:
04/25/2000
Application #:
08842360
Filing Dt:
04/24/1997
Title:
PHOSPHONIC ACID DERIVATIVES
11
Patent #:
Issue Dt:
04/04/2000
Application #:
08863624
Filing Dt:
05/27/1997
Title:
NAALADASE INHIBITORS
12
Patent #:
Issue Dt:
01/04/2000
Application #:
08864545
Filing Dt:
05/28/1997
Title:
METHODS OF CANCER TREATMENT USING NAALADASE INHIBITORS
13
Patent #:
Issue Dt:
01/25/2000
Application #:
08884479
Filing Dt:
06/27/1997
Title:
PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING A GLUTAMATE ABNORMALITY AND EFFECTING A NEURONAL ACTIVITY IN AN ANIMAL USING NAALADASE INHIBITORS
14
Patent #:
Issue Dt:
12/21/1999
Application #:
08889358
Filing Dt:
07/08/1997
Title:
TREATMENT OF GLOBAL AND FOCAL ISCHEMIA USING NAALADASE INHIBITORS
15
Patent #:
Issue Dt:
11/02/1999
Application #:
08899319
Filing Dt:
07/23/1997
Title:
PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING COMPULSIVE DISORDERS USING NAALADASE INHIBITORS
16
Patent #:
Issue Dt:
02/15/2000
Application #:
08900194
Filing Dt:
07/25/1997
Title:
INHIBITORS OF NAALADASE ENZYME ACTIVITY
17
Patent #:
Issue Dt:
11/16/1999
Application #:
08974975
Filing Dt:
11/20/1997
Title:
TREATMENT OF GLOBAL AND FOCAL ISCHEMIA USING NAALADASE INHIBITORS
18
Patent #:
Issue Dt:
11/09/1999
Application #:
08985121
Filing Dt:
12/04/1997
Title:
USE OF NAALADASE ACTIVITY TO IDENTIFY PROSTATE CANCER AND BENIGN PROSTATIC HYPERPLASIA
19
Patent #:
Issue Dt:
05/07/2002
Application #:
09001667
Filing Dt:
12/31/1997
Title:
PRODRUGS OF NAALADASE INHIBITORS
20
Patent #:
Issue Dt:
02/22/2000
Application #:
09002146
Filing Dt:
12/31/1997
Title:
ASYMMETRIC SYNTHESES AND INTERMEDIATES FOR PREPARING ENANTIOMER- ENRICHED HYDROXYPHOSPHINYL DERIVATIVES
21
Patent #:
Issue Dt:
06/06/2000
Application #:
09002147
Filing Dt:
12/31/1997
Title:
PHOSPHINIC ALKANOIC ACID DERIVATIVES
22
Patent #:
Issue Dt:
09/19/2000
Application #:
09050009
Filing Dt:
03/30/1998
Title:
PHOSPHINIC ACID DERIVATIVES
23
Patent #:
Issue Dt:
05/28/2002
Application #:
09110262
Filing Dt:
07/06/1998
Title:
PHARMACEUTICAL COMPOSITIONS AND METHODS OF INHIBITING ANGIOGENESIS USING NAALADASE INHIBITORS
24
Patent #:
Issue Dt:
07/24/2001
Application #:
09228391
Filing Dt:
01/12/1999
Title:
THIO-SUBSTITUTED PENTANEDIOIC ACID DERIVATIVES
25
Patent #:
Issue Dt:
09/11/2001
Application #:
09298866
Filing Dt:
04/26/1999
Title:
PHOSPHONIC ACID DERIVATIVES
26
Patent #:
Issue Dt:
08/07/2001
Application #:
09322688
Filing Dt:
06/01/1999
Title:
HYDROXAMIC ACID DERIVATIVES
27
Patent #:
Issue Dt:
05/08/2001
Application #:
09345782
Filing Dt:
07/01/1999
Title:
METHODS FOR TREATING ANXIETY, ANXIETY DISORDERS AND MEMORY IMPAIRMENT USING NAALADASE INHIBITORS
28
Patent #:
Issue Dt:
10/01/2002
Application #:
09346711
Filing Dt:
07/02/1999
Title:
NAALADASE INHIBITORS USEFUL AS PHARMACEUTICAL COMPOUNDS AND COMPOSITIONS
29
Patent #:
Issue Dt:
11/06/2001
Application #:
09378443
Filing Dt:
08/20/1999
Title:
METABOTROPIC GLUTAMATE RECEPTOR LIGAND DERIVATIVES AS NAALADASE INHIBITORS
30
Patent #:
Issue Dt:
07/02/2002
Application #:
09388442
Filing Dt:
09/02/1999
Title:
PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING A GLUTAMATE ABNORMALITY AND EFFECTING A NEURONAL ACTIVITY IN AN ANIMAL USING NAALADASE INHIBITORS
31
Patent #:
Issue Dt:
04/16/2002
Application #:
09405842
Filing Dt:
09/27/1999
Title:
METHODS OF CANCER TREATMENT USING NAALADASE INHIBITORS
32
Patent #:
Issue Dt:
09/03/2002
Application #:
09425197
Filing Dt:
10/22/1999
Title:
METHODS FOR TREATING CERTAIN DISEASES USING NAALADASE INHIBITORS
33
Patent #:
Issue Dt:
02/19/2002
Application #:
09446110
Filing Dt:
02/14/2000
Title:
SULFONAMIDE COMPOUNDS AND MEDICINAL USE THEREOF
34
Patent #:
Issue Dt:
11/12/2002
Application #:
09466059
Filing Dt:
12/17/1999
Title:
NAALADASE INHIBITORS
35
Patent #:
Issue Dt:
04/23/2002
Application #:
09741169
Filing Dt:
12/21/2000
Title:
PHARMACEUTICAL COMPOSITIONS AND METHODS FOR TREATING ANXIETY, ANXIETY DISORDERS AND MEMORY IMPAIRMENT USING NAALADASE INHIBITORS
36
Patent #:
Issue Dt:
09/17/2002
Application #:
09866758
Filing Dt:
05/30/2001
Publication #:
Pub Dt:
02/14/2002
Title:
BENZENEDICARBOXYLIC ACID DERIVATIVES
37
Patent #:
Issue Dt:
05/22/2007
Application #:
09866961
Filing Dt:
05/30/2001
Publication #:
Pub Dt:
02/20/2003
Title:
NAALADASE INHIBITORS FOR TREATING RETINAL DISORDERS AND GLAUCOMA
38
Patent #:
Issue Dt:
07/01/2003
Application #:
10046917
Filing Dt:
01/17/2002
Publication #:
Pub Dt:
06/05/2003
Title:
THIOL-BASED NAALADASE INHIBITORS
39
Patent #:
Issue Dt:
04/26/2005
Application #:
10141818
Filing Dt:
05/10/2002
Publication #:
Pub Dt:
05/08/2003
Title:
HYDROXAMIC ACIDS AND ACYL HYDROXAMINES AS NAALADASE INHIBITORS
40
Patent #:
Issue Dt:
05/25/2004
Application #:
10156880
Filing Dt:
05/30/2002
Publication #:
Pub Dt:
05/29/2003
Title:
THIOLALKYL BENZOIC ACID DERIVATIVES
41
Patent #:
Issue Dt:
02/08/2005
Application #:
10176046
Filing Dt:
06/21/2002
Publication #:
Pub Dt:
05/01/2003
Title:
BENZENEDICARBOXYLIC ACID DERIVATIVES
42
Patent #:
Issue Dt:
10/19/2004
Application #:
10209011
Filing Dt:
08/01/2002
Publication #:
Pub Dt:
01/23/2003
Title:
METHODS FOR TREATING CERTAIN DISEASES USING NAALADASE INHIBITORS
43
Patent #:
Issue Dt:
11/02/2004
Application #:
10431462
Filing Dt:
05/08/2003
Publication #:
Pub Dt:
11/20/2003
Title:
THIOL-BASED NAALADASE INHIBITORS
44
Patent #:
Issue Dt:
12/12/2006
Application #:
10500319
Filing Dt:
11/22/2004
Publication #:
Pub Dt:
04/14/2005
Title:
INDOLES AS NAALADASE INHIBITORS
45
Patent #:
Issue Dt:
10/24/2006
Application #:
10791278
Filing Dt:
03/03/2004
Publication #:
Pub Dt:
01/06/2005
Title:
THIOLACTONES
46
Patent #:
Issue Dt:
11/21/2006
Application #:
10819146
Filing Dt:
04/07/2004
Publication #:
Pub Dt:
10/07/2004
Title:
THIOLALKYL BENZOIC ACID DERIVATIVES
47
Patent #:
Issue Dt:
01/31/2006
Application #:
10959199
Filing Dt:
10/07/2004
Publication #:
Pub Dt:
04/21/2005
Title:
THIOL-BASED NAALADASE INHIBITORS
Assignors
1
Exec Dt:
10/03/2005
2
Exec Dt:
10/03/2005
Assignee
1
5775 WEST OLD SHAKOPEE ROAD
SUITE 100
BLOOMINGTON, MINNESOTA 55437
Correspondence name and address
SUET CHONG
ARNOLD & PORTER LLP
555 12TH ST, NW, ATTN: IP DOCKETING DEPT
WASHINGTON, DC 20004-1206

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