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Patent #:
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Issue Dt:
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11/11/2014
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Application #:
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11811909
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Filing Dt:
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06/12/2007
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Publication #:
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Pub Dt:
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12/13/2007
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Title:
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Thienopyrimidines useful as modulators of ion channels
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Patent #:
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Issue Dt:
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11/16/2010
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Application #:
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11818224
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Filing Dt:
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06/13/2007
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Publication #:
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Pub Dt:
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01/03/2008
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Title:
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CGRP RECEPTOR ANTAGONISTS
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Patent #:
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Issue Dt:
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12/28/2010
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Application #:
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11823762
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Filing Dt:
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06/28/2007
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Pub Dt:
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02/07/2008
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Title:
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MODULATORS OF MUSCARINIC RECEPTORS
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Patent #:
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Issue Dt:
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03/02/2010
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Application #:
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11824606
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Filing Dt:
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06/29/2007
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Pub Dt:
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01/10/2008
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Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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11/30/2010
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Application #:
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11841233
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Filing Dt:
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08/20/2007
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Pub Dt:
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02/19/2009
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Title:
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INDAZOLINONE COMPOSITIONS USEFUL AS KINASE INHIBITORS
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Patent #:
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Issue Dt:
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09/09/2014
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Application #:
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11841646
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Filing Dt:
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08/20/2007
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Publication #:
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Pub Dt:
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03/20/2008
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Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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04/13/2010
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Application #:
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11893245
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Filing Dt:
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08/15/2007
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Pub Dt:
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07/24/2008
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Title:
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MODULATORS OF MUSCARINIC RECEPTORS
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Patent #:
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Issue Dt:
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08/31/2010
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Application #:
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11894092
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Filing Dt:
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08/20/2007
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Publication #:
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Pub Dt:
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03/11/2010
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Title:
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MODULATORS OF MUSCARINIC RECEPTORS
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Patent #:
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Issue Dt:
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04/27/2010
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Application #:
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11933724
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Filing Dt:
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11/01/2007
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Publication #:
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Pub Dt:
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12/11/2008
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Title:
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BENZIMIDAZOLES USEFUL AS MODULATORS OF ION CHANNELS
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Patent #:
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Issue Dt:
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04/24/2012
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Application #:
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11955874
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Filing Dt:
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12/13/2007
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Publication #:
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Pub Dt:
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07/09/2009
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Title:
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CGRP RECEPTOR ANTAGONISTS
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Patent #:
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Issue Dt:
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01/12/2010
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Application #:
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11975297
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Filing Dt:
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10/18/2007
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Publication #:
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Pub Dt:
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05/21/2009
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Title:
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INDOLE DERIVATIVES AS CFTR MODULATORS
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Patent #:
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Issue Dt:
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04/08/2014
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Application #:
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12009829
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Filing Dt:
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01/22/2008
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Publication #:
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Pub Dt:
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02/19/2009
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Title:
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Inhibitors of caspases
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Patent #:
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Issue Dt:
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03/15/2011
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Application #:
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12026705
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Filing Dt:
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02/06/2008
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Publication #:
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Pub Dt:
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05/29/2008
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Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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Patent #:
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Issue Dt:
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11/20/2012
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Application #:
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12031486
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Filing Dt:
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02/14/2008
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Publication #:
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Pub Dt:
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06/04/2009
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Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HEPATITIS C VIRUS NS3 PROTEASE
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Patent #:
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Issue Dt:
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08/19/2014
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Application #:
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12050289
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Filing Dt:
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03/18/2008
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Publication #:
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Pub Dt:
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07/10/2008
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Title:
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QUINAZOLINES USEFUL AS MODULATORS OF VOLTAGE GATED ION CHANNELS
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Patent #:
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Issue Dt:
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05/31/2011
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Application #:
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12062495
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Filing Dt:
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04/03/2008
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Publication #:
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Pub Dt:
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08/13/2009
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Title:
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INHIBITORS OF P38
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Patent #:
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Issue Dt:
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11/16/2010
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Application #:
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12074983
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Filing Dt:
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03/07/2008
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Publication #:
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Pub Dt:
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02/19/2009
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Title:
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PROCESSES AND INTERMEDIATES
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Patent #:
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Issue Dt:
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02/23/2010
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Application #:
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12079917
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Filing Dt:
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03/28/2008
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Publication #:
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Pub Dt:
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10/23/2008
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Title:
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INHIBITORS OF GSK-3 AND CRYSTAL STRUCTURES OF GSK-3BETA PROTEIN AND PROTEIN COMPLEXES
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Patent #:
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Issue Dt:
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06/29/2010
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Application #:
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12082668
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Filing Dt:
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04/10/2008
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Publication #:
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Pub Dt:
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12/18/2008
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Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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Patent #:
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Issue Dt:
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11/06/2012
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Application #:
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12109598
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Filing Dt:
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04/25/2008
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Publication #:
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Pub Dt:
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11/20/2008
| | | | |
Title:
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PYRAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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03/31/2015
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Application #:
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12114935
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Filing Dt:
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05/05/2008
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Publication #:
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Pub Dt:
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12/11/2008
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Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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03/03/2015
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Application #:
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12117941
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Filing Dt:
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05/09/2008
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Publication #:
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Pub Dt:
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01/29/2015
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Title:
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MODULATORS OF CFTR
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Patent #:
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Issue Dt:
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07/13/2010
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Application #:
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12117948
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Filing Dt:
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05/09/2008
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Publication #:
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Pub Dt:
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11/20/2008
| | | | |
Title:
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MODULATORS OF CFTR
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Patent #:
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Issue Dt:
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06/05/2012
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Application #:
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12124303
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Filing Dt:
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05/21/2008
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Publication #:
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Pub Dt:
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11/27/2008
| | | | |
Title:
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ION CHANNEL MODULATORS AND METHODS OF USE
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Patent #:
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Issue Dt:
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06/14/2011
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Application #:
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12140497
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Filing Dt:
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06/17/2008
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Publication #:
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Pub Dt:
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04/09/2009
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Title:
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CASPASE INHIBITORS AND USES THEREOF
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Patent #:
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NONE
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12147861
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06/27/2008
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Pub Dt:
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10/01/2009
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Title:
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COMPOUNDS USEFUL IN CFTR ASSAYS AND METHODS THEREWITH
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Patent #:
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Issue Dt:
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09/20/2011
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12165838
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Filing Dt:
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07/01/2008
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Publication #:
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Pub Dt:
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01/08/2009
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Title:
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PRODRUG OF AN ICE INHIBITOR
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Patent #:
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Issue Dt:
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12/07/2010
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Application #:
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12183580
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Filing Dt:
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07/31/2008
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Publication #:
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Pub Dt:
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01/15/2009
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Title:
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THIAZOLES AND OXAZOLES USEFUL AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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05/29/2012
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Application #:
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12187909
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08/07/2008
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Publication #:
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Pub Dt:
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05/14/2009
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Title:
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AMINO SUBSTITUTED PYRIDINES AS POTENT KINASE INHIBITORS
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Patent #:
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Issue Dt:
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08/09/2011
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12212063
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09/17/2008
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Publication #:
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Pub Dt:
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04/23/2009
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Title:
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PYRIDYL SULFONAMIDES AS MODULATORS OF ION CHANNELS
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Patent #:
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04/05/2011
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12217517
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07/02/2008
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Pub Dt:
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02/12/2009
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Title:
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INHIBITORS OF ASPARTYL PROTEASE
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Patent #:
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09/18/2012
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Application #:
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12221921
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Filing Dt:
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08/07/2008
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Publication #:
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Pub Dt:
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01/29/2009
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Title:
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INHIBITORS OF IMPDH ENZYME
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Patent #:
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09/11/2012
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12224270
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02/16/2009
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09/10/2009
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Title:
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MODULATORS OF MUSCARINIC RECEPTORS
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08/17/2010
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12228164
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08/07/2008
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04/09/2009
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Title:
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PRODRUGS OF CARBAMATE INHIBITORS OF IMPDH
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08/28/2012
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12231982
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09/08/2008
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06/03/2010
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Title:
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PEPTIDOMIMETIC PROTEASE INHIBITORS
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01/25/2011
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12235820
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09/23/2008
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08/27/2009
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Title:
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CASPASE INHIBITORS AND USES THEREOF
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05/29/2012
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12246778
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10/07/2008
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07/09/2009
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Title:
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GYRASE INHIBITORS AND USES THEREOF
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Patent #:
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08/27/2013
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12249230
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10/10/2008
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Pub Dt:
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04/16/2009
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Title:
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HETEROARYL AMIDES USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
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Patent #:
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03/05/2013
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12249251
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10/10/2008
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Pub Dt:
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05/07/2009
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Title:
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AMIDES USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
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07/15/2014
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12249270
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10/10/2008
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Pub Dt:
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05/07/2009
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Title:
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ARYL AMIDES USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
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Patent #:
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05/08/2012
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Application #:
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12262459
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10/31/2008
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11/26/2009
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Title:
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KINASE INHIBITORS
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04/23/2013
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12265125
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11/05/2008
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Publication #:
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Pub Dt:
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11/26/2009
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Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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08/09/2011
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12269108
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11/12/2008
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Pub Dt:
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05/21/2009
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Title:
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PYRROLIDINONE BENZENESULFONAMIDE DERIVATIVES AS MODULATORS OF ION CHANNELS FOR THE TREATMENT OF PAIN
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01/17/2012
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12269109
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11/12/2008
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Publication #:
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Pub Dt:
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05/14/2009
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Title:
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HETEROCYCLIC DERIVATIVES AS MODULATORS OF ION CHANNELS
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04/05/2011
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12269429
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11/12/2008
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07/09/2009
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Title:
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INHIBITORS OF TACE
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08/13/2013
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12271088
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11/14/2008
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06/04/2009
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Title:
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MODULATORS OF ATP-BINDING CASSETTE-TRANSPORTERS
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02/08/2011
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12272425
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11/17/2008
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Pub Dt:
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07/30/2009
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Title:
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HCV NS3-NS4 PROTEASE RESISTANCE MUTANTS
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05/29/2012
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12273799
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11/19/2008
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Pub Dt:
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07/09/2009
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Title:
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AZAINDOLES USEFUL AS INHIBITORS OF JAK AND OTHER PROTEIN KINASES
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04/24/2012
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12283702
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09/15/2008
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Pub Dt:
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04/16/2009
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Title:
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SOLID FORMS OF N-[2,4-BIS(1,1-DIMETHYLETHYL)-5-HYDROXYPHENYL]-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXAMIDE
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07/05/2011
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12287055
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10/03/2008
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Pub Dt:
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04/16/2009
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Title:
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MODULATORS OF MUSCARINIC RECEPTORS
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NONE
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12298353
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07/01/2009
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02/04/2010
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Title:
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HEPATITIS C VIRUS INFECTION BIOMARKERS
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08/13/2013
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12327902
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12/04/2008
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Publication #:
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Pub Dt:
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07/02/2009
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Title:
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SOLID FORMS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACID
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02/28/2012
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12327915
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12/04/2008
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Pub Dt:
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07/09/2009
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Title:
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PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
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Patent #:
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NONE
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Application #:
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12327922
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Filing Dt:
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12/04/2008
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Publication #:
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Pub Dt:
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07/09/2009
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Title:
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FORMULATIONS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACID
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Patent #:
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07/10/2012
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Application #:
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12329179
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Filing Dt:
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12/05/2008
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Publication #:
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Pub Dt:
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03/11/2010
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Title:
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SOLID FORMS OF 1-ETHYL-3-(5-(5-FLUOROPYRIDIN-3-YL)-7-(PYRIMIDIN-2-YL)-1H-BENZO[D]IMIDAZOL-2-YL)UREA
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Patent #:
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01/18/2011
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12338129
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Filing Dt:
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12/18/2008
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Publication #:
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Pub Dt:
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05/07/2009
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Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF GSK-3
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Patent #:
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Issue Dt:
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01/24/2012
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Application #:
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12351401
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Filing Dt:
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01/09/2009
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Publication #:
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Pub Dt:
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09/10/2009
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Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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12/04/2012
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Application #:
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12351447
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Filing Dt:
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01/09/2009
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Publication #:
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Pub Dt:
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12/03/2009
| | | | |
Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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01/24/2012
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Application #:
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12355880
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Filing Dt:
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01/19/2009
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Publication #:
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Pub Dt:
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09/30/2010
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Title:
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DUAL EXPRESSION VECTOR SYSTEM AND SCREENING METHODS
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Patent #:
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Issue Dt:
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11/30/2010
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Application #:
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12356745
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Filing Dt:
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01/21/2009
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Publication #:
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Pub Dt:
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07/23/2009
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Title:
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CGRP RECEPTOR ANTAGONISTS
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Patent #:
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Issue Dt:
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03/15/2011
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Application #:
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12359749
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Filing Dt:
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01/26/2009
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Publication #:
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Pub Dt:
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05/21/2009
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Title:
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CASPASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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11/09/2010
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Application #:
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12365424
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Filing Dt:
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02/04/2009
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Publication #:
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Pub Dt:
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07/02/2009
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Title:
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POLYMORPHIC FORMS OF (S)-1-CYANOBUTAN-2-YL (S)-1-(3-(3-(3-METHOXY-4-(OXAZOL-5-YL)PHENYL)URIEDO)PHENYL)ETHYLCARBAMATE
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Patent #:
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Issue Dt:
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06/04/2013
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Application #:
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12370175
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Filing Dt:
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02/12/2009
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Publication #:
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Pub Dt:
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11/05/2009
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Title:
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INHIBITORS OF ASPARTYL PROTEASE
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Patent #:
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Issue Dt:
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10/30/2012
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Application #:
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12392298
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Filing Dt:
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02/25/2009
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Publication #:
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Pub Dt:
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09/03/2009
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Title:
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HETEROARYL DERIVATIVES AS CFTR MODULATORS
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Patent #:
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Issue Dt:
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03/06/2012
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Application #:
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12410553
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Filing Dt:
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03/25/2009
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Publication #:
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Pub Dt:
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07/16/2009
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Title:
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AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS
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Patent #:
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Issue Dt:
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07/24/2012
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Application #:
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12410725
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Filing Dt:
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03/25/2009
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Publication #:
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Pub Dt:
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10/01/2009
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Title:
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PYRIDYL DERIVATIVES AS CFTR MODULATORS
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Patent #:
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Issue Dt:
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03/29/2011
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Application #:
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12416777
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Filing Dt:
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04/01/2009
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Publication #:
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Pub Dt:
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10/22/2009
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Title:
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SODIUM CHANNEL PROTEIN TYPE III ALPHA-SUBUNIT SPLICE VARIANT
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Patent #:
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Issue Dt:
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10/22/2013
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Application #:
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12422496
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Filing Dt:
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04/13/2009
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Publication #:
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Pub Dt:
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10/08/2009
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Title:
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AZAINDOLE DERIVATIVES AS CFTR MODULATORS
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Patent #:
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Issue Dt:
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02/15/2011
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Application #:
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12424883
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Filing Dt:
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04/16/2009
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Publication #:
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Pub Dt:
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10/08/2009
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Title:
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HETEROCYCLIC DERIVATIVES FOR MODULATION OF CALCIUM CHANNELS
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Patent #:
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Issue Dt:
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03/19/2013
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Application #:
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12430207
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Filing Dt:
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04/27/2009
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Publication #:
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Pub Dt:
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03/11/2010
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Title:
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PROCESSES AND INTERMEDIATES
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Patent #:
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Issue Dt:
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02/12/2013
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Application #:
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12433998
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Filing Dt:
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05/01/2009
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Publication #:
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Pub Dt:
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01/28/2010
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Title:
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AMINOPYRIDINES AND AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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04/24/2012
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Application #:
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12434154
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Filing Dt:
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05/01/2009
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Publication #:
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Pub Dt:
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04/01/2010
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Title:
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TRICYCLIC HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF JANUS KINASE
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Patent #:
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Issue Dt:
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08/17/2010
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Application #:
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12435646
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Filing Dt:
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05/05/2009
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Publication #:
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Pub Dt:
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09/03/2009
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Title:
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PROCESSES FOR PREPARING BIARYL UREAS AND ANALOGS THEREOF
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Patent #:
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Issue Dt:
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09/18/2012
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Application #:
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12436407
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Filing Dt:
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05/06/2009
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Publication #:
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Pub Dt:
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09/03/2009
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Title:
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SUBSTITUTED PYRIMIDINES USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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09/18/2012
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Application #:
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12438995
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Filing Dt:
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02/05/2010
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Publication #:
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Pub Dt:
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06/10/2010
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Title:
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INHIBITORS OF C-MET AND USES THEREOF
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Patent #:
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Issue Dt:
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07/09/2013
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Application #:
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12441187
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Filing Dt:
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02/12/2010
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Publication #:
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Pub Dt:
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06/10/2010
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Title:
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HETEROCYCLIC INHIBITORS OF C-MET AND USES THEREOF
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Patent #:
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Issue Dt:
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03/06/2012
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Application #:
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12448258
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Filing Dt:
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11/13/2009
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Publication #:
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Pub Dt:
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04/22/2010
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Title:
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SUBSTITUTED 5,6-DIHYDROIMIDAZO[1,5-F]PTERIDINES USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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08/21/2012
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Application #:
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12448489
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Filing Dt:
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11/10/2009
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Publication #:
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Pub Dt:
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07/29/2010
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Title:
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5-CYANO-4- (PYRROLO [2,3B] PYRIDINE-3-YL) -PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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03/06/2012
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Application #:
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12464380
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Filing Dt:
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05/12/2009
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Publication #:
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Pub Dt:
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11/12/2009
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Title:
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CASPASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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11/23/2010
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Application #:
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12466420
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Filing Dt:
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05/15/2009
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Publication #:
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Pub Dt:
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11/12/2009
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Title:
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COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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06/05/2012
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Application #:
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12471896
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05/26/2009
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Publication #:
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Pub Dt:
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01/20/2011
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Title:
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CRYSTAL STRUCTURE OF HUMAN JAK3 KINASE DOMAIN COMPLEX AND BINDING POCKETS THEREOF
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Patent #:
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Issue Dt:
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12/13/2011
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12471950
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Filing Dt:
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05/26/2009
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Publication #:
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Pub Dt:
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03/18/2010
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Title:
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COMPOSITIONS OF N-[2,4-BIS(1,1-DIMETHYLETHYL)-5-HYDROXYPHENYL]-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXAMIDE
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05/15/2012
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12475381
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05/29/2009
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Pub Dt:
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09/24/2009
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Title:
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MODULAR TEST TUBE RACK
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Issue Dt:
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10/11/2011
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12478372
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06/04/2009
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Publication #:
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Pub Dt:
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12/31/2009
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Title:
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GYRASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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10/07/2014
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12481962
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Filing Dt:
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06/10/2009
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Pub Dt:
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10/01/2009
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Title:
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PHARMACEUTICAL COMPOSITIONS
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11/29/2011
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12483312
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06/12/2009
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Publication #:
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Pub Dt:
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12/31/2009
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Title:
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GYRASE INHIBITORS AND USES THEREOF
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06/26/2012
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12483787
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06/12/2009
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12/16/2010
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DEVICES FOR CRYSTALLIZATION BY CONTROLLED EVAPORATION
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04/23/2013
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12486235
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06/17/2009
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Pub Dt:
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01/28/2010
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Title:
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AMINOPYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES
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12/07/2010
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12495880
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07/01/2009
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Pub Dt:
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01/07/2010
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Title:
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HETEROCYCLIC DERIVATIVES AS MODULATORS OF ION CHANNELS
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11/05/2013
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12528952
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04/22/2010
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Pub Dt:
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10/28/2010
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Title:
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Inhibitors of Serine Proteases
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06/24/2014
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12528977
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11/23/2010
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Pub Dt:
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03/10/2011
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Title:
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Co-Crystals and Pharmaceutical Compositions Comprising the Same
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08/07/2012
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12538396
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08/10/2009
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Pub Dt:
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12/10/2009
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Title:
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THIAZOLES, IMIDAZOLES, AND PYRAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES
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NONE
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12540516
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08/13/2009
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Pub Dt:
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04/01/2010
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Title:
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QUINOXALINES USEFUL AS INHIBITORS OF PROTEIN KINASES
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07/19/2011
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12545347
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08/21/2009
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12/17/2009
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Title:
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PYRAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
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04/05/2011
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12550042
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08/28/2009
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Pub Dt:
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12/24/2009
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Title:
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INHIBITORS OF P38
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08/02/2011
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12550649
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08/31/2009
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Publication #:
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Pub Dt:
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12/31/2009
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Title:
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INDANE DERIVATIVES AS MODULATORS OF ION CHANNELS
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Issue Dt:
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02/18/2014
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12552003
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09/01/2009
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Publication #:
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Pub Dt:
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12/31/2009
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Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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06/05/2012
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Application #:
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12552430
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09/02/2009
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03/11/2010
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Title:
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GYRASE INHIBITORS AND USES THEREOF
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Issue Dt:
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04/10/2012
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12555203
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09/08/2009
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Publication #:
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Pub Dt:
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12/31/2009
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Title:
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POLYMORPHIC FORMS OF (S)-1-TETRAHYDROFURAN-3-YL-3-(3-(3-METHOXY-4-(OXAZOL-5-YL)PHENYL)UREIDO)BENZYL CARBAMATE
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Patent #:
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Issue Dt:
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04/10/2012
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Application #:
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12556845
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Filing Dt:
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09/10/2009
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Publication #:
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Pub Dt:
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04/08/2010
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Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
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