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02/25/2010
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02/25/2010
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02/18/2010
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10/06/2011
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08/23/2012
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11/28/2013
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02/20/2014
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04/10/2014
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05/28/2015
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08/13/2015
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09/17/2015
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12/31/2015
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05/12/2016
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05/26/2016
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09/22/2016
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02/23/2017
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08/28/2018
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Publication #:
|
|
Pub Dt:
|
04/25/2019
| | | | |
Title:
|
ANTIOXIDANT INFLAMMATION MODULATORS: OLEANOLIC ACID DERIVATIVES WITH AMINO AND OTHER MODIFICATIONS AT C-17
|
|
|
Patent #:
|
|
Issue Dt:
|
02/27/2024
|
Application #:
|
16130242
|
Filing Dt:
|
09/13/2018
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Publication #:
|
|
Pub Dt:
|
03/14/2019
| | | | |
Title:
|
METHODS OF TREATING OBESITY USING ANTIOXIDANT INFLAMMATION MODULATORS
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|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
16157225
|
Filing Dt:
|
10/11/2018
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Publication #:
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|
Pub Dt:
|
03/28/2019
| | | | |
Title:
|
METHODS OF TREATING AND PREVENTING ENDOTHELIAL DYSFUNCTION USING BARDOXOLONE METHYL OR ANALOGS THEREOF
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|
|
Patent #:
|
|
Issue Dt:
|
09/14/2021
|
Application #:
|
16186051
|
Filing Dt:
|
11/09/2018
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Publication #:
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|
Pub Dt:
|
02/27/2020
| | | | |
Title:
|
2,2-DIFLUOROPROPIONAMIDE DERIVATIVES OF BARDOXOLONE METHYL, POLYMORPHIC FORMS AND METHODS OF USE THEREOF
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|
|
Patent #:
|
|
Issue Dt:
|
07/21/2020
|
Application #:
|
16265256
|
Filing Dt:
|
02/01/2019
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Publication #:
|
|
Pub Dt:
|
08/08/2019
| | | | |
Title:
|
CO-CRYSTAL FORMS OF A NOVOBIOCIN ANALOG AND PROLINE
|
|
|
Patent #:
|
|
Issue Dt:
|
03/23/2021
|
Application #:
|
16315821
|
Filing Dt:
|
01/07/2019
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Publication #:
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|
Pub Dt:
|
11/21/2019
| | | | |
Title:
|
METHODS OF TREATING ALPORT SYNDROME USING BARDOXOLONE METHYL OR ANALOGS THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
04/05/2022
|
Application #:
|
16468054
|
Filing Dt:
|
06/10/2019
|
Publication #:
|
|
Pub Dt:
|
04/30/2020
| | | | |
Title:
|
PYRIMIDINE TRICYCLIC ENONE DERIVATIVES FOR INHIBITION OF ROR-GAMMA AND OTHER USES
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|
|
Patent #:
|
|
Issue Dt:
|
01/26/2021
|
Application #:
|
16527171
|
Filing Dt:
|
07/31/2019
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Publication #:
|
|
Pub Dt:
|
04/30/2020
| | | | |
Title:
|
C17-HETEROARYL DERIVATIVES OF OLEANOLIC ACID AND METHODS OF USE THEREOF
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|
|
Patent #:
|
|
Issue Dt:
|
12/07/2021
|
Application #:
|
16701585
|
Filing Dt:
|
12/03/2019
|
Publication #:
|
|
Pub Dt:
|
07/02/2020
| | | | |
Title:
|
PYRAZOLYL AND PYRIMIDINYL TRICYCLIC ENONES AS ANTIOXIDANT INFLAMMATION MODULATORS
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|
|
Patent #:
|
|
Issue Dt:
|
08/24/2021
|
Application #:
|
16776091
|
Filing Dt:
|
01/29/2020
|
Publication #:
|
|
Pub Dt:
|
08/27/2020
| | | | |
Title:
|
BIPHENYL AMIDES WITH MODIFIED ETHER GROUPS AS HSP90 INHIBITORS AND HSP70 INDUCERS
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|
|
Patent #:
|
|
Issue Dt:
|
01/05/2021
|
Application #:
|
16783025
|
Filing Dt:
|
02/05/2020
|
Publication #:
|
|
Pub Dt:
|
09/10/2020
| | | | |
Title:
|
C-TERMINAL HSP90 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
08/17/2021
|
Application #:
|
16786429
|
Filing Dt:
|
02/10/2020
|
Publication #:
|
|
Pub Dt:
|
07/30/2020
| | | | |
Title:
|
ANTIOXIDANT INFLAMMATION MODULATORS: OLEANOLIC ACID DERIVATIVES WITH AMINO AND OTHER MODIFICATIONS AT C-17
|
|
|
Patent #:
|
|
Issue Dt:
|
08/02/2022
|
Application #:
|
16894461
|
Filing Dt:
|
06/05/2020
|
Publication #:
|
|
Pub Dt:
|
11/05/2020
| | | | |
Title:
|
CO-CRYSTAL FORMS OF A NOVOBIOCIN ANALOG AND PROLINE
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
16933635
|
Filing Dt:
|
07/20/2020
|
Publication #:
|
|
Pub Dt:
|
02/11/2021
| | | | |
Title:
|
C17 POLAR-SUBSTITUTED HETEROAROMATIC SYNTHETIC TRITERPENOIDS AND METHODS OF USE THEREOF
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|
|
Patent #:
|
|
Issue Dt:
|
11/28/2023
|
Application #:
|
17055331
|
Filing Dt:
|
11/13/2020
|
Publication #:
|
|
Pub Dt:
|
08/26/2021
| | | | |
Title:
|
BIARYL AMIDES WITH MODIFIED SUGAR GROUPS FOR TREATMENT OF DISEASES ASSOCIATED WITH HEAT SHOCK PROTEIN PATHWAY
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|
|
Patent #:
|
|
Issue Dt:
|
07/19/2022
|
Application #:
|
17112060
|
Filing Dt:
|
12/04/2020
|
Publication #:
|
|
Pub Dt:
|
06/24/2021
| | | | |
Title:
|
C-TERMINAL HSP90 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
08/09/2022
|
Application #:
|
17135128
|
Filing Dt:
|
12/28/2020
|
Publication #:
|
|
Pub Dt:
|
05/13/2021
| | | | |
Title:
|
C17-HETEROARYL DERIVATIVES OF OLEANOLIC ACID AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
09/20/2022
|
Application #:
|
17173340
|
Filing Dt:
|
02/11/2021
|
Publication #:
|
|
Pub Dt:
|
06/03/2021
| | | | |
Title:
|
METHODS OF TREATING ALPORT SYNDROME USING BARDOXOLONE METHYL OR ANALOGS THEREOF
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|
|
Patent #:
|
NONE
|
Issue Dt:
|
05/28/2024
|
Application #:
|
17251295
|
Filing Dt:
|
12/11/2020
|
Publication #:
|
|
Pub Dt:
|
09/23/2021
| | | | |
Title:
|
PYRAZOLE AND IMIDAZOLE COMPOUNDS FOR INHIBITION OF IL-17 AND RORGAMMA
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|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17252841
|
Filing Dt:
|
12/16/2020
|
Publication #:
|
|
Pub Dt:
|
05/20/2021
| | | | |
Title:
|
CYSTEINE-DEPENDENT INVERSE AGONISTS OF NUCLEAR RECEPTORS ROR-GAMMA/ROR-GAMMA-T AND METHODS OF TREATING DISEASES OR DISORDERS THEREWITH
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|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17304778
|
Filing Dt:
|
06/25/2021
|
Publication #:
|
|
Pub Dt:
|
11/18/2021
| | | | |
Title:
|
2,2-DIFLUOROPROPIONAMIDE DERIVATIVES OF BARDOXOLONE METHYL, POLYMORPHIC FORMS AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
03/05/2024
|
Application #:
|
17305537
|
Filing Dt:
|
07/09/2021
|
Publication #:
|
|
Pub Dt:
|
01/27/2022
| | | | |
Title:
|
ANTIOXIDANT INFLAMMATION MODULATORS: OLEANOLIC ACID DERIVATIVES WITH AMINO AND OTHER MODIFICATIONS AT C-17
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|
|
Patent #:
|
|
Issue Dt:
|
07/25/2023
|
Application #:
|
17375882
|
Filing Dt:
|
07/14/2021
|
Publication #:
|
|
Pub Dt:
|
02/10/2022
| | | | |
Title:
|
BIPHENYL AMIDES WITH MODIFIED ETHER GROUPS AS HSP90 INHIBITORS AND HSP70 INDUCERS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/16/2024
|
Application #:
|
17444594
|
Filing Dt:
|
08/06/2021
|
Publication #:
|
|
Pub Dt:
|
03/10/2022
| | | | |
Title:
|
2,2-DIFLUOROPROPIONAMIDE DERIVATIVES OF BARDOXOLONE METHYL, POLYMORPHIC FORMS AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
11/14/2023
|
Application #:
|
17457808
|
Filing Dt:
|
12/06/2021
|
Publication #:
|
|
Pub Dt:
|
09/08/2022
| | | | |
Title:
|
PYRAZOLYL AND PYRIMIDINYL TRICYCLIC ENONES AS ANTIOXIDANT INFLAMMATION MODULATORS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17577456
|
Filing Dt:
|
01/18/2022
|
Publication #:
|
|
Pub Dt:
|
05/05/2022
| | | | |
Title:
|
PYRIMIDINE TRICYCLIC ENONE DERIVATIVES FOR INHIBITION OF ROR-GAMMA AND OTHER USES
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17757701
|
Filing Dt:
|
06/17/2022
|
Publication #:
|
|
Pub Dt:
|
04/13/2023
| | | | |
Title:
|
SYNTHETIC TRITERPENOIDS WITH NITROGEN-BASED SUBSTITUENTS AT C-17 AND METHODS OF USE THEREOF
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|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17863135
|
Filing Dt:
|
07/12/2022
|
Publication #:
|
|
Pub Dt:
|
03/30/2023
| | | | |
Title:
|
C-TERMINAL HSP90 INHIBITORS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17998291
|
Filing Dt:
|
11/09/2022
|
Publication #:
|
|
Pub Dt:
|
08/17/2023
| | | | |
Title:
|
METHODS OF TREATING COVID-19 USING BARDOXOLONE METHYL OR ANALOGS THEREOF
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
18149696
|
Filing Dt:
|
01/04/2023
|
Publication #:
|
|
Pub Dt:
|
08/10/2023
| | | | |
Title:
|
C4-MODIFIED OLEANOLIC ACID DERIVATIVES FOR INHIBITION OF IL-17 AND OTHER USES
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
18168495
|
Filing Dt:
|
02/13/2023
|
Publication #:
|
|
Pub Dt:
|
02/08/2024
| | | | |
Title:
|
CO-CRYSTAL FORMS OF A NOVOBIOCIN ANALOG AND PROLINE
|
|