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110
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Patent #:
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Issue Dt:
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03/06/1990
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Application #:
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07376172
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Filing Dt:
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06/30/1989
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Title:
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ESTERS OF HEXAHYDRO-8-HYDROXY-2,6-METHANO-2H-QUINOLIZIN-3(4H)-ONE AND RELATED COMPOUNDS
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Patent #:
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Issue Dt:
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10/24/2000
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Application #:
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07622305
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Filing Dt:
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12/05/1990
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Title:
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ISOLATION OF CASTANOSPERMINE AND ITS USE AS AN ANTIDIABETIC AGENT
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Patent #:
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Issue Dt:
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05/04/1993
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Application #:
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07667943
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Filing Dt:
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03/12/1991
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Title:
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8-SUBSTITUTED PURINES AS SELECTIVE ADENOSINE RECEPTOR AGENTS
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Patent #:
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Issue Dt:
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01/11/1994
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Application #:
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07776143
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Filing Dt:
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10/15/1991
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Title:
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NOVEL AZADECALIN AMIDES AND THIOAMIDES AS INHIBITORS OF CHOLESTEROL BIOSYNTHESIS
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Patent #:
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Issue Dt:
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02/23/1993
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Application #:
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07795572
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Filing Dt:
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11/12/1991
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Title:
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3-AMIDOINDOLYL DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF
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Patent #:
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Issue Dt:
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05/16/1995
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Application #:
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07896733
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Filing Dt:
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06/09/1992
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Title:
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S-ADENOSYL METHIONINE DECARBOXYLASE INHIBITORS
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Patent #:
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Issue Dt:
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03/08/1994
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Application #:
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07926109
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Filing Dt:
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08/05/1992
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Title:
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CYCLIC NITRONES, PHARMACEUTICAL COMPOSITONS THEREOF AND THEIR USE IN TREATING SHOCK.
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Patent #:
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Issue Dt:
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06/14/1994
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Application #:
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07995309
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Filing Dt:
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12/22/1992
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Title:
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CONTROLLED RELEASE FORMULATION FOR PHARMACEUTICAL COMPOUNDS
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Patent #:
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Issue Dt:
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03/07/1995
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Application #:
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08032526
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Filing Dt:
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03/15/1993
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Title:
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NEUROPEPTIDE Y AGONISTS AND PARTIAL AGONISTS
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Patent #:
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Issue Dt:
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08/16/1994
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Application #:
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08039539
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Filing Dt:
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03/29/1993
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Title:
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PROCESS FOR THE PRODUCTION OF 2-IMIDAZOLONES
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Patent #:
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Issue Dt:
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05/03/1994
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Application #:
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08046326
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Filing Dt:
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04/12/1993
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Title:
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NOVEL AMINO AND NITRO CONTAINING TRICYCLIC COMPOUNDS USEFUL AS INHIBITORS OF ACE
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Patent #:
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Issue Dt:
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04/19/1994
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Application #:
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08077619
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Filing Dt:
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06/15/1993
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Title:
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NOVEL BIS[4-(2,6-DI-ALKYL)PHENOL]SILANE DERIVATIVES AS ANTIATHEROSCLEROTIC AGENTS
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Patent #:
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Issue Dt:
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09/24/1996
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Application #:
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08081368
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Filing Dt:
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06/30/1993
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Title:
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NOVEL DIFLUORO STATONE ANALOGS
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Patent #:
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Issue Dt:
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10/04/1994
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Application #:
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08097097
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Filing Dt:
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07/26/1993
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Title:
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METHOD FOR PRODUCING AN OREXIGENIC EFFECT
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Patent #:
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Issue Dt:
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01/10/1995
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Application #:
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08108786
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Filing Dt:
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08/17/1993
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Title:
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ANTIALLERGIC COMPOUNDS
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Patent #:
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Issue Dt:
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01/03/1995
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Application #:
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08113505
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Filing Dt:
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08/27/1993
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Title:
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2'-HALOMETHYLIDENE CYTIDINE, URIDINE AND GUANOSINE COMPOUNDS AND THEIR PHARMACEUTICAL COMPOSITIONS
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Patent #:
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Issue Dt:
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07/25/1995
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Application #:
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08119791
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Filing Dt:
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09/15/1993
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Title:
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SEROTONIN RECEPTOR AGENTS
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Patent #:
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Issue Dt:
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06/13/1995
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Application #:
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08119924
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Filing Dt:
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09/10/1993
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Title:
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NOVEL AMINOACETYLMERCAPTO DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
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06/27/1995
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Application #:
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08146646
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Filing Dt:
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11/01/1993
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Title:
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NOVEL 2-SUBSTITUTED INDANE-2-MERCAPTOACETYLAMIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
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07/04/1995
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Application #:
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08149572
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Filing Dt:
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11/09/1993
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Title:
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NOVEL MERCAPTOACETYLAMIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
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03/19/1996
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Application #:
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08154146
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Filing Dt:
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11/17/1993
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Title:
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CALCIUM UPTAKE INHIBITORS
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Patent #:
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Issue Dt:
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11/28/1995
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Application #:
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08159913
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Filing Dt:
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11/30/1993
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Title:
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HETEROCYCLIC-NMDA ANTAGONISTS
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Patent #:
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Issue Dt:
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10/10/1995
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Application #:
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08163235
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Filing Dt:
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12/06/1993
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Title:
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NOVEL 2-SUBSTITUTED INDANE-2-CARBOXYALKYL DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
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01/16/1996
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Application #:
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08165144
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Filing Dt:
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12/10/1993
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Title:
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NMDA ANTAGONISTS
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Patent #:
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Issue Dt:
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11/01/1994
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Application #:
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08187353
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Filing Dt:
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01/25/1994
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Title:
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NMDA ANTAGONISTS
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Patent #:
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Issue Dt:
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12/06/1994
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Application #:
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08201149
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Filing Dt:
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02/24/1994
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Title:
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PIPERIDINYL THIACYCLIC DERIVATIVES
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Patent #:
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Issue Dt:
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07/25/1995
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Application #:
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08201878
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Filing Dt:
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02/25/1994
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Title:
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METHOD OF USING 4-AMINO- STEROIDS IN THE TREATMENT OF BENIGN PROSTATIC HYPERPLASIA
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Patent #:
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Issue Dt:
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04/08/1997
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Application #:
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08209084
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Filing Dt:
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03/09/1994
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Title:
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TREATMENT OF OBSESSIVE-COMPULSIVE DISORDERS WITH 5-HT2 ANTAGONISTS
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Patent #:
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Issue Dt:
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05/07/1996
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Application #:
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08241814
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Filing Dt:
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05/12/1994
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Title:
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CARBOCYCLIC ADENOSINE ANALOGS USEFUL AS IMMUNOSUPPRESSANTS
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Patent #:
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|
Issue Dt:
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03/05/1996
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Application #:
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08248847
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Filing Dt:
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05/25/1994
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Title:
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NOVEL PEPTIDASE INHIBITORS
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Patent #:
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|
Issue Dt:
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06/05/2001
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Application #:
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08275685
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Filing Dt:
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07/14/1994
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Title:
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NOVEL INTERMEDIATES USEFUL FOR THE PREPARATION OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
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12/26/1995
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Application #:
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08279623
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Filing Dt:
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07/22/1994
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Title:
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1-PIPERIDINYL ALKANOYLANYL SULFONAMIDES FOR TREATMENT OF CARDIAC ARRHYTHMIA.
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Patent #:
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Issue Dt:
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04/16/1996
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Application #:
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08290792
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Filing Dt:
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08/16/1994
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Title:
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2,6-METHANO-2H-QUINOLIZIN DERIVATIVE AS 5-HT3-RECEPTOR ANTAGONIST
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Patent #:
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Issue Dt:
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08/29/1995
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Application #:
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08307538
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Filing Dt:
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09/16/1994
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Title:
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1-PHENYL-3-PHENYL-2-PROPYNE-1-ONES AS CALCIUM UPTAKE INHIBITORS
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Patent #:
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Issue Dt:
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03/19/1996
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Application #:
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08313657
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Filing Dt:
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09/27/1994
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Title:
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CARDIOPROTECTIVE TOCOPHEROL ANALOGS
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Patent #:
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Issue Dt:
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08/13/1996
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Application #:
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08318670
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Filing Dt:
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10/06/1994
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Title:
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HYDRAZIDE DERIVATIVES OF 3,4-DIHYDRO-2H-1-BENZOPYRANS
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Patent #:
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Issue Dt:
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04/23/1996
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Application #:
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08318784
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Filing Dt:
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10/05/1994
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Title:
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CARDIOPROTECTIVE AGENTS
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Patent #:
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Issue Dt:
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07/23/1996
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Application #:
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08336703
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Filing Dt:
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11/08/1994
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Title:
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9-PURINYL PHOSPHONIC ACID DERIVATIVES
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Patent #:
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Issue Dt:
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10/01/1996
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Application #:
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08350236
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Filing Dt:
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12/06/1994
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Title:
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NOVEL ANTIDEPRESSANTS
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Patent #:
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|
Issue Dt:
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07/02/1996
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Application #:
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08353736
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Filing Dt:
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12/12/1994
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Title:
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NOVEL 2,6-DI-ALKYL-4-SILY1-PHENOLS AS ANTIATHEROSCLEROTIC AGENTS
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Patent #:
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|
Issue Dt:
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05/20/1997
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Application #:
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08369234
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Filing Dt:
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01/06/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
10/01/1996
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Application #:
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08372694
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Filing Dt:
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01/13/1995
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Title:
|
(+)-ALPHA-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL)ETHYL]-4- PIPERIDINEMETHANOL
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Patent #:
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Issue Dt:
|
02/13/1996
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Application #:
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08372710
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Filing Dt:
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01/13/1995
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Title:
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3-AMIDOINDOLYL DERIVATIVE
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Patent #:
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Issue Dt:
|
07/16/2002
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Application #:
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08372712
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Filing Dt:
|
01/13/1995
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Title:
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NOVEL 9-N-BICYCLIC NUCEOSIDE AGENTS USEFUL AS SELECTIVE INHIBITORS OF PROINFLAMMATORY CYTOKINES
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Patent #:
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Issue Dt:
|
04/16/1996
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Application #:
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08380472
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Filing Dt:
|
01/30/1995
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Title:
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5H-DIBENZO (A,D) CYCLOHEPTENES AS MUSCARINIC RECEPTOR ANYAGONISTS
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Patent #:
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Issue Dt:
|
12/02/1997
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Application #:
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08382941
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Filing Dt:
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01/31/1995
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Title:
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NOVEL ACETYLCHOLINESTERASE INHIBITORS
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Patent #:
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Issue Dt:
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04/01/2003
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Application #:
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08383339
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Filing Dt:
|
02/03/1995
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Publication #:
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|
Pub Dt:
|
01/10/2002
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Title:
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NOVEL CARBOCYCLIC NUCLEOSIDE AGENTS USEFUL AS SELECTIVE INHIBITORS OF PROINFLAMMATORY CYTOKINES
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Patent #:
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|
Issue Dt:
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10/22/1996
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Application #:
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08397304
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Filing Dt:
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03/02/1995
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Title:
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NOVEL 2-SUBSTITUTED INDANE-2-MERCAPTOACETYLAMIDE DISULFIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
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08/05/1997
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Application #:
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08400314
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Filing Dt:
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03/06/1995
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Title:
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NOVEL PROCESSES FOR PREPARING (S)-4-AMINO-HEPTA-5,6-DIENOIC ACID AND INTERMEDIATES THEREOF
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Patent #:
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|
Issue Dt:
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06/03/1997
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Application #:
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08406979
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Filing Dt:
|
04/03/1995
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Title:
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NOVEL MERCAPTOACETYLAMIDE BICYCLIC LACTAM DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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|
Issue Dt:
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06/18/1996
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Application #:
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08417179
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Filing Dt:
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04/05/1995
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Title:
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NOVEL MERCAPTOACETYLAMIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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|
Issue Dt:
|
02/13/1996
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Application #:
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08417424
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Filing Dt:
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04/05/1995
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Title:
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NOVEL MERCAPTOACETYLAMIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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|
Issue Dt:
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01/07/1997
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Application #:
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08423675
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Filing Dt:
|
04/17/1995
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Title:
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NOVEL 2-SUBSTITUTED INDANE-2-CARBOXYALKYL DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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|
Issue Dt:
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05/20/1997
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Application #:
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08427937
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Filing Dt:
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04/26/1995
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Title:
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METHOD OF EFFECTING IMMUNOSUPPRESSION BY ADMINISTERING CARBOCYCLIC ADENOSINE ANALOGS
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Patent #:
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|
Issue Dt:
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10/07/1997
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Application #:
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08431587
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Filing Dt:
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05/01/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
07/01/1997
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Application #:
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08432487
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Filing Dt:
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05/01/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
02/27/1996
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Application #:
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08432617
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Filing Dt:
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05/02/1995
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Title:
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ANTICOAGULANT PEPTIDES
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Patent #:
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|
Issue Dt:
|
04/08/1997
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Application #:
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08432660
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Filing Dt:
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05/02/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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|
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Patent #:
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|
Issue Dt:
|
07/29/1997
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Application #:
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08432731
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Filing Dt:
|
05/02/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
08/05/1997
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Application #:
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08433299
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Filing Dt:
|
05/03/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
07/22/1997
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Application #:
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08433777
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Filing Dt:
|
05/03/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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Issue Dt:
|
09/02/1997
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Application #:
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08434134
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Filing Dt:
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05/02/1995
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Title:
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NOVEL PROCESS FOR PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
04/16/1996
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Application #:
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08439536
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Filing Dt:
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05/11/1995
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Title:
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PROCESS FOR THE PREPARATION OF RIBONUCLEOTIDE REDUCTASE INHIBITORS
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Patent #:
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Issue Dt:
|
05/21/1996
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Application #:
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08441911
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Filing Dt:
|
05/16/1995
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Title:
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3-(INDOL-3-YL)-PROPENOIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF
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Patent #:
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Issue Dt:
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11/14/2000
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Application #:
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08458747
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Filing Dt:
|
06/02/1995
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Title:
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NOVEL INTERMEDIATES USEFUL FOR THE PREPARATION OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES
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Patent #:
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|
Issue Dt:
|
07/30/1996
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Application #:
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08460029
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Filing Dt:
|
06/02/1995
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Title:
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ANTIARRHYTHMIC PIPERIDIN-1-YL-2,2-DIALKYLPROPANONE ARYLSULFONAMIDE DERIVATIVES
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Patent #:
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Issue Dt:
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02/25/1997
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Application #:
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08462406
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Filing Dt:
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06/05/1995
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Title:
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NMDA ANTAGONISTS
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Patent #:
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Issue Dt:
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02/24/1998
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Application #:
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08476538
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Filing Dt:
|
06/07/1995
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Title:
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(+)-ALPHA-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUROPHENYL)ETHYL]-4- PIPERIDINEMETHANOL
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Patent #:
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Issue Dt:
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12/15/1998
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Application #:
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08481666
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Filing Dt:
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06/07/1995
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Title:
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NOVEL PEPTIDASE INHIBITORS
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Patent #:
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Issue Dt:
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12/23/1997
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Application #:
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08485700
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Filing Dt:
|
06/07/1995
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Title:
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(+)-ALPHA_(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL)ETHYL]-4- PIPERIDINEMETHANOL
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Patent #:
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Issue Dt:
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12/23/1997
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Application #:
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08485701
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Filing Dt:
|
06/07/1995
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Title:
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(+)-A-(2,3-DIMETHOXYPHENYL)-1-[2-(4-FLUOROPHENYL)ETHYL]-4- PIPERIDINEMETHANOL
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Patent #:
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Issue Dt:
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08/20/1996
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Application #:
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08502980
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Filing Dt:
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07/17/1995
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Title:
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NMDA ANTAGONISM METHOD
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Patent #:
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Issue Dt:
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10/28/1997
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Application #:
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08502989
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Filing Dt:
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07/17/1995
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Title:
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TRIFUNCTIONAL ANTITHROMBIN AND ANTIPLATELET PEPTIDES
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Patent #:
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Issue Dt:
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12/30/1997
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Application #:
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08554212
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Filing Dt:
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11/06/1995
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Title:
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3-AMINOINDOLYL DERIVATIVES
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Patent #:
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Issue Dt:
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10/07/1997
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Application #:
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08554621
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Filing Dt:
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11/06/1995
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Title:
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3-AMIDOINDOLYL DERIVATIVES
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Patent #:
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Issue Dt:
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09/02/1997
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Application #:
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08557120
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Filing Dt:
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11/21/1995
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Title:
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AROMATIC ACETYLCHOLINESTERASE INHIBITORS
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Patent #:
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Issue Dt:
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02/18/1997
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Application #:
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08571022
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Filing Dt:
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12/12/1995
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Title:
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NOVEL INDANE-2-MERCAPTOACETYLAMIDE DISULFIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE
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Patent #:
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Issue Dt:
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05/13/1997
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Application #:
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08572326
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Filing Dt:
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12/14/1995
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Title:
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NOVEL 2-SUBSTITUTED INDANE-2-MERCAPTOACETYLAMIDE DISULFIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
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02/10/1998
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Application #:
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08578698
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Filing Dt:
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12/18/1995
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Title:
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DIFLUORO STATONE ANALOGS
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Patent #:
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|
Issue Dt:
|
03/02/1999
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Application #:
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08594505
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Filing Dt:
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01/31/1996
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Title:
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NOVEL INDOLE DERIVATIVES USEFUL TO TREAT ESTROGEN-RELATED NEOPLASMS AND DISORDERS
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Patent #:
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Issue Dt:
|
11/25/1997
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Application #:
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08624362
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Filing Dt:
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07/03/1996
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Title:
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STABLE PHARMACEUTICAL COMPOSITION OF TERFENADINE AND IBUPROFEN
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Patent #:
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Issue Dt:
|
11/02/1999
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Application #:
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08624407
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Filing Dt:
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03/28/1996
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Title:
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INHIBITORS OF BETA-AMYLOID PROTEIN PRODUCTION
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Patent #:
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Issue Dt:
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09/16/1997
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Application #:
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08648150
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Filing Dt:
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07/03/1996
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Title:
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HETEROCYCLIC BENZENESULFONYLIMINE DERIVATIVES AS INHIBITORS OF IL-1 ACTION
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Patent #:
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Issue Dt:
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12/16/1997
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Application #:
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08670136
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Filing Dt:
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06/25/1996
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Title:
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ACYLATED ENOL DERIVATIVES AS PRODRUGS OF ELASTASE INHIBITORS
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Patent #:
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Issue Dt:
|
03/24/1998
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Application #:
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08673250
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Filing Dt:
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06/26/1996
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Title:
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NOVEL MERCAPTOACETYLAMIDO 1,3,4,5-TETRAHYDRO-BENZO[C]AZEPIN-3-ONE DISULFIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
|
12/28/1999
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Application #:
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08737905
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Filing Dt:
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11/22/1996
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Title:
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PERFLUOROALKYL KETONE INHIBITORS OF ELASTASE AND PROCESSES FOR MAKING THE SAME
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Patent #:
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Issue Dt:
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05/26/1998
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Application #:
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08781566
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Filing Dt:
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01/09/1997
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Title:
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(S)-4-AMINO-HEPTA-5,6-DIENOIC ACID AND INTERMEDIATES THEROF
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Patent #:
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Issue Dt:
|
02/10/1998
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Application #:
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08788098
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Filing Dt:
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01/23/1997
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Title:
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ANTI-VIRAL COMPOUNDS
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Patent #:
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Issue Dt:
|
01/19/1999
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Application #:
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08795576
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Filing Dt:
|
02/06/1997
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Title:
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SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES
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Patent #:
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Issue Dt:
|
10/20/1998
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Application #:
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08798664
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Filing Dt:
|
02/11/1997
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Title:
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SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES
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Patent #:
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Issue Dt:
|
10/05/1999
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Application #:
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08854647
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Filing Dt:
|
05/12/1997
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Title:
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METHOD OF LOWERING SERUM CHOLESTEROL LEVELS WITH 2,6-DI-ALKYL-4-SILYL-PHENOLS
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Patent #:
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Issue Dt:
|
10/26/1999
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Application #:
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08882764
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Filing Dt:
|
06/26/1997
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Title:
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ACYLATED ENOL DERIVATIVES AS PRODRUGS OF ELASTASE INHIBITORS
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Patent #:
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|
Issue Dt:
|
03/09/1999
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Application #:
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08910053
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Filing Dt:
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08/12/1997
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Title:
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NOVEL MERCAPTOACETYLAMINO 1,3,4,5-TETRAHYDRO-BENZO(C)AZEPIN-2-ONE DISULEFIDE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE
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Patent #:
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Issue Dt:
|
06/08/1999
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Application #:
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08921956
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Filing Dt:
|
08/26/1997
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Title:
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USE OF CERTAIN ESTERS OF HEXAHYDRO-8-HYDROXY-2,6-METHAN0-2H- QUINOLOZIN-3(4H)-ONE AND RELATED COMPOUNDS FOR TREATING COGNITIVE DISORDERS
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Patent #:
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Issue Dt:
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09/05/2000
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Application #:
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08925943
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Filing Dt:
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09/08/1997
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Title:
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DIFLUORO STATONE ANALOGS
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Patent #:
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Issue Dt:
|
07/13/1999
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Application #:
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09131761
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Filing Dt:
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08/10/1998
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Title:
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ETHYLENIL AND ALLENIC PHOSPHONATE DERIVATIVES OF PURINES
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Patent #:
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Issue Dt:
|
10/10/2000
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Application #:
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09139009
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Filing Dt:
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08/24/1998
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Title:
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NOVEL PEPTIDASE INHIBITORS
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Patent #:
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Issue Dt:
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09/21/1999
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Application #:
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09181888
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Filing Dt:
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10/29/1998
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Title:
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DERIVATIVES OF AMIDE ANALOGS OF CERTAIN METHANO BRIDGED QUINOLIZINES
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Patent #:
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Issue Dt:
|
06/04/2002
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Application #:
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09663343
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Filing Dt:
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09/15/2000
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Title:
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METHOD OF PROVIDING AN ANTIHISTAMINIC EFFECT IN A HEPATICALLY IMPAIRED PATIENT
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Patent #:
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Issue Dt:
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04/22/2003
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Application #:
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09725259
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Filing Dt:
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11/29/2000
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Publication #:
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Pub Dt:
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09/06/2001
| | | | |
Title:
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NOVEL INTERMEDIATES USEFUL FOR THE PREPARATION OF ANTIHISTAMINIC PIPERIDINE DERIVATIVES
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