|
|
Patent #:
|
|
Issue Dt:
|
10/15/2013
|
Application #:
|
13129593
|
Filing Dt:
|
05/17/2011
|
Publication #:
|
|
Pub Dt:
|
09/15/2011
| | | | |
Title:
|
ARYL METHYL BENZOQUINAZOLININE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/10/2013
|
Application #:
|
13130473
|
Filing Dt:
|
05/20/2011
|
Publication #:
|
|
Pub Dt:
|
09/22/2011
| | | | |
Title:
|
NITROOXY CYCLOALKANE DERIVATIVES
|
|
|
Patent #:
|
|
Issue Dt:
|
02/05/2013
|
Application #:
|
13130891
|
Filing Dt:
|
05/24/2011
|
Publication #:
|
|
Pub Dt:
|
09/22/2011
| | | | |
Title:
|
BIARYL CARBOXAMIDES
|
|
|
Patent #:
|
|
Issue Dt:
|
12/31/2013
|
Application #:
|
13133516
|
Filing Dt:
|
06/08/2011
|
Publication #:
|
|
Pub Dt:
|
09/29/2011
| | | | |
Title:
|
NOVEL CRYSTALLINE FORMS OF AN INHIBITOR OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1
|
|
|
Patent #:
|
|
Issue Dt:
|
11/05/2013
|
Application #:
|
13139830
|
Filing Dt:
|
10/13/2011
|
Publication #:
|
|
Pub Dt:
|
01/26/2012
| | | | |
Title:
|
TRIAZOLE DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE
|
|
|
Patent #:
|
|
Issue Dt:
|
05/21/2013
|
Application #:
|
13140260
|
Filing Dt:
|
06/16/2011
|
Publication #:
|
|
Pub Dt:
|
10/13/2011
| | | | |
Title:
|
GLUCAGON RECEPTOR ANTAGONIST COMPOUNDS
|
|
|
Patent #:
|
|
Issue Dt:
|
06/24/2014
|
Application #:
|
13140987
|
Filing Dt:
|
08/02/2011
|
Publication #:
|
|
Pub Dt:
|
12/01/2011
| | | | |
Title:
|
GAMMA SECRETASE MODULATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/13/2014
|
Application #:
|
13141227
|
Filing Dt:
|
07/15/2011
|
Publication #:
|
|
Pub Dt:
|
10/27/2011
| | | | |
Title:
|
PYRIMIDINE DERIVATIVES AS GPCR MODULATORS FOR USE IN THE TREATMENT OF OBESITY AND DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
04/02/2013
|
Application #:
|
13141344
|
Filing Dt:
|
07/15/2011
|
Publication #:
|
|
Pub Dt:
|
10/27/2011
| | | | |
Title:
|
BICYCLIC HETEROCYCLE DERIVATIVES AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
11/26/2013
|
Application #:
|
13144123
|
Filing Dt:
|
09/26/2011
|
Publication #:
|
|
Pub Dt:
|
01/12/2012
| | | | |
Title:
|
IMIDAZO[1,2-A]PYRIDINES AND IMIDAZO[1,2-B]PYRIDAZINES AS MARK INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/17/2013
|
Application #:
|
13145190
|
Filing Dt:
|
07/19/2011
|
Publication #:
|
|
Pub Dt:
|
11/10/2011
| | | | |
Title:
|
TRIFLUOROMETHYLSULFONAMIDE GAMMA SECRETASE INHIBITOR
|
|
|
Patent #:
|
|
Issue Dt:
|
08/19/2014
|
Application #:
|
13148577
|
Filing Dt:
|
08/09/2011
|
Publication #:
|
|
Pub Dt:
|
12/22/2011
| | | | |
Title:
|
GLUCAGON RECEPTOR ANTAGONIST COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE
|
|
|
Patent #:
|
|
Issue Dt:
|
12/04/2012
|
Application #:
|
13148809
|
Filing Dt:
|
08/10/2011
|
Publication #:
|
|
Pub Dt:
|
12/15/2011
| | | | |
Title:
|
GLUCAGON RECEPTOR ANTAGONIST COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE
|
|
|
Patent #:
|
|
Issue Dt:
|
09/16/2014
|
Application #:
|
13151683
|
Filing Dt:
|
06/02/2011
|
Publication #:
|
|
Pub Dt:
|
05/31/2012
| | | | |
Title:
|
DIHYDROFOLATE REDUCTASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/09/2013
|
Application #:
|
13167495
|
Filing Dt:
|
06/23/2011
|
Title:
|
ANTIBIOTIC COMPOSITIONS FOR THE TREATMENT OF GRAM NEGATIVE INFECTIONS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/12/2013
|
Application #:
|
13188520
|
Filing Dt:
|
07/22/2011
|
Publication #:
|
|
Pub Dt:
|
12/08/2011
| | | | |
Title:
|
FUSED RING THROMBIN RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/10/2013
|
Application #:
|
13190137
|
Filing Dt:
|
07/25/2011
|
Publication #:
|
|
Pub Dt:
|
07/26/2012
| | | | |
Title:
|
PROCESS FOR LARGE SCALE PRODUCTION OF PLASMID DNA BY E. COLI FERMENTATION
|
|
|
Patent #:
|
|
Issue Dt:
|
06/19/2012
|
Application #:
|
13191978
|
Filing Dt:
|
07/27/2011
|
Publication #:
|
|
Pub Dt:
|
11/17/2011
| | | | |
Title:
|
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/21/2014
|
Application #:
|
13201570
|
Filing Dt:
|
08/15/2011
|
Publication #:
|
|
Pub Dt:
|
12/15/2011
| | | | |
Title:
|
SPIROPYRROLIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE
|
|
|
Patent #:
|
|
Issue Dt:
|
07/16/2013
|
Application #:
|
13201575
|
Filing Dt:
|
08/15/2011
|
Publication #:
|
|
Pub Dt:
|
12/08/2011
| | | | |
Title:
|
PYRAZOLO [4,3-C] CINNOLIN-3-ONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/27/2012
|
Application #:
|
13202124
|
Filing Dt:
|
08/18/2011
|
Publication #:
|
|
Pub Dt:
|
12/08/2011
| | | | |
Title:
|
GLUCAGON RECEPTOR ANTAGONIST COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE
|
|
|
Patent #:
|
|
Issue Dt:
|
01/28/2014
|
Application #:
|
13203983
|
Filing Dt:
|
08/31/2011
|
Publication #:
|
|
Pub Dt:
|
12/29/2011
| | | | |
Title:
|
BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYLGLYCEROL ACYLTRANSFERASE
|
|
|
Patent #:
|
|
Issue Dt:
|
11/18/2014
|
Application #:
|
13242426
|
Filing Dt:
|
09/23/2011
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
SUBSTITUTED QUINOXALINES AS INHIBITORS OF FATTY ACID BINDING PROTEIN
|
|
|
Patent #:
|
|
Issue Dt:
|
01/01/2013
|
Application #:
|
13242744
|
Filing Dt:
|
09/23/2011
|
Publication #:
|
|
Pub Dt:
|
04/05/2012
| | | | |
Title:
|
ANTAGONISTS OF PCSK9
|
|
|
Patent #:
|
|
Issue Dt:
|
07/22/2014
|
Application #:
|
13247009
|
Filing Dt:
|
09/28/2011
|
Publication #:
|
|
Pub Dt:
|
05/31/2012
| | | | |
Title:
|
ETHER BENZOTRIAZOLE DERIVATIVES
|
|
|
Patent #:
|
|
Issue Dt:
|
02/16/2016
|
Application #:
|
13251410
|
Filing Dt:
|
10/03/2011
|
Publication #:
|
|
Pub Dt:
|
01/26/2012
| | | | |
Title:
|
SURFACE DISPLAY OF WHOLE ANTIBODIES IN EUKARYOTES
|
|
|
Patent #:
|
|
Issue Dt:
|
07/09/2013
|
Application #:
|
13254108
|
Filing Dt:
|
08/31/2011
|
Publication #:
|
|
Pub Dt:
|
12/29/2011
| | | | |
Title:
|
COMBINATION CANCER THERAPY WITH AN AKT INHIBITOR AND OTHER ANTICANCER AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/04/2014
|
Application #:
|
13254363
|
Filing Dt:
|
09/01/2011
|
Publication #:
|
|
Pub Dt:
|
05/10/2012
| | | | |
Title:
|
IMIDAZOLE DERIVATIVES USEFUL AS MODULATORS OF FAAH AND AS FAAH IMAGING AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/24/2013
|
Application #:
|
13255785
|
Filing Dt:
|
09/09/2011
|
Publication #:
|
|
Pub Dt:
|
01/05/2012
| | | | |
Title:
|
INHIBITORS OF AKT ACTIVITY
|
|
|
Patent #:
|
|
Issue Dt:
|
07/15/2014
|
Application #:
|
13256354
|
Filing Dt:
|
09/13/2011
|
Publication #:
|
|
Pub Dt:
|
01/12/2012
| | | | |
Title:
|
CGRP RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/29/2013
|
Application #:
|
13258943
|
Filing Dt:
|
09/22/2011
|
Publication #:
|
|
Pub Dt:
|
01/19/2012
| | | | |
Title:
|
P2X3 RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN
|
|
|
Patent #:
|
|
Issue Dt:
|
01/19/2016
|
Application #:
|
13259040
|
Filing Dt:
|
09/22/2011
|
Publication #:
|
|
Pub Dt:
|
03/15/2012
| | | | |
Title:
|
P2X3 Receptor Antagonists for Treatment of Pain
|
|
|
Patent #:
|
|
Issue Dt:
|
02/03/2015
|
Application #:
|
13259087
|
Filing Dt:
|
09/22/2011
|
Publication #:
|
|
Pub Dt:
|
01/26/2012
| | | | |
Title:
|
P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN
|
|
|
Patent #:
|
|
Issue Dt:
|
11/12/2013
|
Application #:
|
13260673
|
Filing Dt:
|
09/27/2011
|
Publication #:
|
|
Pub Dt:
|
01/26/2012
| | | | |
Title:
|
BICYCLIC PIPERIDINE AND PIPERAZINE DERIVATIVES AS GPCR MODULATORS FOR THE TREATMENT OF OBESITY, DIABETES AND OTHER METABOLIC DISORDERS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/28/2014
|
Application #:
|
13260684
|
Filing Dt:
|
12/19/2011
|
Publication #:
|
|
Pub Dt:
|
04/05/2012
| | | | |
Title:
|
INHIBITORS OF HEPATITIS C VIRUS REPLICATION
|
|
|
Patent #:
|
|
Issue Dt:
|
04/08/2014
|
Application #:
|
13262096
|
Filing Dt:
|
12/13/2011
|
Publication #:
|
|
Pub Dt:
|
03/29/2012
| | | | |
Title:
|
INHIBITORS OF AKT ACTIVITY
|
|
|
Patent #:
|
|
Issue Dt:
|
11/26/2013
|
Application #:
|
13263193
|
Filing Dt:
|
01/25/2012
|
Publication #:
|
|
Pub Dt:
|
05/10/2012
| | | | |
Title:
|
PYRAZOLO[1,5-A]PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/23/2012
|
Application #:
|
13264267
|
Filing Dt:
|
10/13/2011
|
Publication #:
|
|
Pub Dt:
|
02/16/2012
| | | | |
Title:
|
HETEROCYCLIC FUSED CINNOLINE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
08/20/2013
|
Application #:
|
13266043
|
Filing Dt:
|
10/24/2011
|
Publication #:
|
|
Pub Dt:
|
02/16/2012
| | | | |
Title:
|
P38 KINASE INHIBITING AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/29/2013
|
Application #:
|
13267324
|
Filing Dt:
|
10/06/2011
|
Publication #:
|
|
Pub Dt:
|
10/18/2012
| | | | |
Title:
|
BENZENESULFONYL-CHROMANE, THIOCHROMANE, TETRAHYDRONAPHTHALENE AND RELATED GAMMA SECRETASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/10/2013
|
Application #:
|
13273043
|
Filing Dt:
|
10/13/2011
|
Publication #:
|
|
Pub Dt:
|
02/23/2012
| | | | |
Title:
|
CYTOSKELETAL ACTIVE RHO KINASE INHIBITOR COMPOUNDS, COMPOSITION AND USE
|
|
|
Patent #:
|
|
Issue Dt:
|
05/21/2013
|
Application #:
|
13280148
|
Filing Dt:
|
10/24/2011
|
Publication #:
|
|
Pub Dt:
|
02/16/2012
| | | | |
Title:
|
ANTIBIOTIC MACROCYCLE COMPOUNDS AND METHODS OF MANUFACTURE AND USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
10/13/2015
|
Application #:
|
13285433
|
Filing Dt:
|
10/31/2011
|
Title:
|
CHROMATOGRAPHY MEDIA
|
|
|
Patent #:
|
|
Issue Dt:
|
01/07/2014
|
Application #:
|
13290251
|
Filing Dt:
|
11/07/2011
|
Publication #:
|
|
Pub Dt:
|
03/01/2012
| | | | |
Title:
|
PROCESSES OF MAKING AND USING PHARMACEUTICAL FORMULATIONS OF ANTINEOPLASTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
06/17/2014
|
Application #:
|
13293166
|
Filing Dt:
|
11/10/2011
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
PIPERIDINONE CARBOXAMIDE AZAINDANE CGRP RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/16/2014
|
Application #:
|
13293177
|
Filing Dt:
|
11/10/2011
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
PIPERIDINONE CARBOXAMIDE AZAINDANE CGRP RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/16/2014
|
Application #:
|
13293177
|
Filing Dt:
|
11/10/2011
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
PIPERIDINONE CARBOXAMIDE AZAINDANE CGRP RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/09/2013
|
Application #:
|
13293186
|
Filing Dt:
|
11/10/2011
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
PIPERIDINONE CARBOXAMIDE AZAINDANE CGRP RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/31/2013
|
Application #:
|
13319250
|
Filing Dt:
|
11/07/2011
|
Publication #:
|
|
Pub Dt:
|
03/01/2012
| | | | |
Title:
|
PYRROLIDINE-DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/22/2015
|
Application #:
|
13320427
|
Filing Dt:
|
06/11/2012
|
Publication #:
|
|
Pub Dt:
|
10/04/2012
| | | | |
Title:
|
FUSED TRICYCLIC ARYL COMPOUNDS USEFUL FOR THE TREATMENT OF VIRAL DISEASES
|
|
|
Patent #:
|
|
Issue Dt:
|
09/30/2014
|
Application #:
|
13320816
|
Filing Dt:
|
11/16/2011
|
Publication #:
|
|
Pub Dt:
|
03/15/2012
| | | | |
Title:
|
RADIOLABELED PDE10 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/30/2013
|
Application #:
|
13322184
|
Filing Dt:
|
11/23/2011
|
Publication #:
|
|
Pub Dt:
|
06/07/2012
| | | | |
Title:
|
HIV PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/26/2013
|
Application #:
|
13323366
|
Filing Dt:
|
12/12/2011
|
Publication #:
|
|
Pub Dt:
|
04/05/2012
| | | | |
Title:
|
PROCESS FOR THE SYNTHESIS OF AZETIDINONES
|
|
|
Patent #:
|
|
Issue Dt:
|
02/10/2015
|
Application #:
|
13344905
|
Filing Dt:
|
01/06/2012
|
Publication #:
|
|
Pub Dt:
|
06/07/2012
| | | | |
Title:
|
MAMMALIAN EXPRESSION VECTOR pUHAB
|
|
|
Patent #:
|
|
Issue Dt:
|
07/08/2014
|
Application #:
|
13375088
|
Filing Dt:
|
06/11/2012
|
Publication #:
|
|
Pub Dt:
|
06/27/2013
| | | | |
Title:
|
Antiviral Compounds Composed of Three Aligned Aryl Moieties to Treat Diseases such as Hepatitis C
|
|
|
Patent #:
|
|
Issue Dt:
|
03/17/2015
|
Application #:
|
13375094
|
Filing Dt:
|
06/11/2012
|
Publication #:
|
|
Pub Dt:
|
10/11/2012
| | | | |
Title:
|
ANTIVIRAL COMPOUNDS OF THREE LINKED ARYL MOIETIES TO TREAT DISEASES SUCH AS HEPATITIS C
|
|
|
Patent #:
|
|
Issue Dt:
|
05/05/2015
|
Application #:
|
13376945
|
Filing Dt:
|
12/08/2011
|
Publication #:
|
|
Pub Dt:
|
04/05/2012
| | | | |
Title:
|
3-Substituted-8-Substituted-3H-Imidazo[5,1-d][1,2,3,5]tetrazin-4-one Compounds and Their Use
|
|
|
Patent #:
|
|
Issue Dt:
|
06/25/2013
|
Application #:
|
13377707
|
Filing Dt:
|
12/12/2011
|
Publication #:
|
|
Pub Dt:
|
05/03/2012
| | | | |
Title:
|
THIOPHENES AS GLUCAGON RECEPTOR ANTAGONISTS, COMPOSITIONS, AND METHODS FOR THEIR USE
|
|
|
Patent #:
|
|
Issue Dt:
|
12/30/2014
|
Application #:
|
13378237
|
Filing Dt:
|
12/14/2011
|
Publication #:
|
|
Pub Dt:
|
04/19/2012
| | | | |
Title:
|
SUBSTITUTED-1,3,8-TRIAZASPIRO[4.5]DECANE-2,4-DIONES
|
|
|
Patent #:
|
|
Issue Dt:
|
08/26/2014
|
Application #:
|
13379536
|
Filing Dt:
|
12/20/2011
|
Publication #:
|
|
Pub Dt:
|
05/03/2012
| | | | |
Title:
|
SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES
|
|
|
Patent #:
|
|
Issue Dt:
|
12/17/2013
|
Application #:
|
13379685
|
Filing Dt:
|
03/22/2012
|
Publication #:
|
|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
FUSED TRICYCLIC COMPOUNDS AS NOVEL mTOR INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/12/2013
|
Application #:
|
13379701
|
Filing Dt:
|
12/21/2011
|
Publication #:
|
|
Pub Dt:
|
06/07/2012
| | | | |
Title:
|
SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES
|
|
|
Patent #:
|
|
Issue Dt:
|
05/12/2015
|
Application #:
|
13382469
|
Filing Dt:
|
01/05/2012
|
Publication #:
|
|
Pub Dt:
|
05/03/2012
| | | | |
Title:
|
PLATELET-ACTIVATING FACTOR RECEPTOR ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/25/2014
|
Application #:
|
13384946
|
Filing Dt:
|
01/19/2012
|
Publication #:
|
|
Pub Dt:
|
05/10/2012
| | | | |
Title:
|
QUINOLINONE PDE2 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/09/2014
|
Application #:
|
13387542
|
Filing Dt:
|
01/27/2012
|
Publication #:
|
|
Pub Dt:
|
05/17/2012
| | | | |
Title:
|
HEPATITIS C VIRUS NS3 PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/25/2014
|
Application #:
|
13387619
|
Filing Dt:
|
03/30/2012
|
Publication #:
|
|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
ENANTIO- AND STEREO-SPECIFIC SYNTHESES OF BETA-AMINO-ALPHA- HYDROXY AMIDES
|
|
|
Patent #:
|
|
Issue Dt:
|
04/29/2014
|
Application #:
|
13388270
|
Filing Dt:
|
04/10/2012
|
Publication #:
|
|
Pub Dt:
|
07/26/2012
| | | | |
Title:
|
ANTI-GITR ANTIBODIES
|
|
|
Patent #:
|
|
Issue Dt:
|
12/17/2013
|
Application #:
|
13388628
|
Filing Dt:
|
02/02/2012
|
Publication #:
|
|
Pub Dt:
|
05/31/2012
| | | | |
Title:
|
4, 5, 6-TRISUBSTITUTED PYRIMIDINE DERIVATIVES AS FACTOR IXA INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/03/2013
|
Application #:
|
13389029
|
Filing Dt:
|
05/16/2012
|
Publication #:
|
|
Pub Dt:
|
08/30/2012
| | | | |
Title:
|
PROCESS FOR PREPARING A 2-ALKYNYL SUBSTITUTED 5-AMINO-PYRAZOLO-[4,3-E]-1,2,4-TRIAZOLO[1,5-C]PYRIMIDINE
|
|
|
Patent #:
|
|
Issue Dt:
|
10/08/2013
|
Application #:
|
13390147
|
Filing Dt:
|
02/13/2012
|
Publication #:
|
|
Pub Dt:
|
06/07/2012
| | | | |
Title:
|
SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT
|
|
|
Patent #:
|
|
Issue Dt:
|
06/04/2013
|
Application #:
|
13390538
|
Filing Dt:
|
02/15/2012
|
Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
AMINOTETRAHYDROPYRANS AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
05/06/2014
|
Application #:
|
13390708
|
Filing Dt:
|
02/16/2012
|
Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
SUBSTITUTED AMINOPIPERIDINES AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
10/15/2013
|
Application #:
|
13390856
|
Filing Dt:
|
02/16/2012
|
Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
PENTAFLUOROSULFUR IMINO HETEROCYCLIC COMPOUNDS AS BACE-1 INHIBITORS, COMPOSITIONS, AND THEIR USE
|
|
|
Patent #:
|
|
Issue Dt:
|
03/10/2015
|
Application #:
|
13391315
|
Filing Dt:
|
02/20/2012
|
Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
ETHER BENZOTRIAZOLE DERIVATIVES
|
|
|
Patent #:
|
|
Issue Dt:
|
03/11/2014
|
Application #:
|
13391402
|
Filing Dt:
|
04/12/2012
|
Publication #:
|
|
Pub Dt:
|
08/16/2012
| | | | |
Title:
|
HETEROCYCLIC AMIDE COMPOUNDS AS PROTEIN KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/29/2013
|
Application #:
|
13391441
|
Filing Dt:
|
02/21/2012
|
Publication #:
|
|
Pub Dt:
|
08/02/2012
| | | | |
Title:
|
PENTAFLUOROSULFUR IMINO HETEROCYCLIC COMPOUNDS AS BACE-1 INHIBITORS, COMPOSITIONS AND THEIR USE
|
|
|
Patent #:
|
|
Issue Dt:
|
12/10/2013
|
Application #:
|
13392282
|
Filing Dt:
|
05/14/2012
|
Publication #:
|
|
Pub Dt:
|
09/06/2012
| | | | |
Title:
|
NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/20/2014
|
Application #:
|
13392297
|
Filing Dt:
|
03/16/2012
|
Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
IMINOTHIADIAZINE DIOXIDE COMPOUNDS AS BACE INHIBITORS, COMPOSITIONS AND THEIR USE
|
|
|
Patent #:
|
|
Issue Dt:
|
09/30/2014
|
Application #:
|
13392647
|
Filing Dt:
|
02/27/2012
|
Publication #:
|
|
Pub Dt:
|
06/21/2012
| | | | |
Title:
|
PYRANYL ARYL METHYL BENZOQUINAZOLINONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/15/2013
|
Application #:
|
13392662
|
Filing Dt:
|
02/27/2012
|
Publication #:
|
|
Pub Dt:
|
06/21/2012
| | | | |
Title:
|
NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/22/2013
|
Application #:
|
13392955
|
Filing Dt:
|
03/20/2012
|
Publication #:
|
|
Pub Dt:
|
07/26/2012
| | | | |
Title:
|
IMINOTHIADIAZINE DIOXIDE COMPOUNDS AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE
|
|
|
Patent #:
|
|
Issue Dt:
|
03/31/2015
|
Application #:
|
13393571
|
Filing Dt:
|
04/04/2012
|
Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
MODULATORS OF CELL CYCLE CHECKPOINTS AND THEIR USE IN COMBINATION WITH CHECKPOINT KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/01/2016
|
Application #:
|
13394985
|
Filing Dt:
|
07/30/2012
|
Publication #:
|
|
Pub Dt:
|
03/28/2013
| | | | |
Title:
|
GYRASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/23/2013
|
Application #:
|
13395992
|
Filing Dt:
|
03/14/2012
|
Publication #:
|
|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
HETEROCYCLIC-FUSED PYRAZOLO[4,3-C] PYRIDIN-3-ONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/09/2013
|
Application #:
|
13398887
|
Filing Dt:
|
02/17/2012
|
Publication #:
|
|
Pub Dt:
|
06/14/2012
| | | | |
Title:
|
AMINOTETRAHYDROPYRANS AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
01/20/2015
|
Application #:
|
13402521
|
Filing Dt:
|
02/22/2012
|
Publication #:
|
|
Pub Dt:
|
02/27/2014
| | | | |
Title:
|
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/29/2013
|
Application #:
|
13412032
|
Filing Dt:
|
03/05/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
PRIMARY AMINE DIAZENIUMDIOLATE HETEROCYCLIC DERIVATIVES
|
|
|
Patent #:
|
|
Issue Dt:
|
04/08/2014
|
Application #:
|
13415404
|
Filing Dt:
|
03/08/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/08/2014
|
Application #:
|
13416140
|
Filing Dt:
|
03/09/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/09/2014
|
Application #:
|
13420007
|
Filing Dt:
|
03/14/2012
|
Publication #:
|
|
Pub Dt:
|
11/01/2012
| | | | |
Title:
|
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/14/2014
|
Application #:
|
13421396
|
Filing Dt:
|
03/15/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/03/2013
|
Application #:
|
13435130
|
Filing Dt:
|
03/30/2012
|
Publication #:
|
|
Pub Dt:
|
07/26/2012
| | | | |
Title:
|
METHOD OF TREATMENT USING FATTY ACID SYNTHESIS INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/03/2013
|
Application #:
|
13477742
|
Filing Dt:
|
05/22/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
COMPOSITIONS CONTAINING OPIOID ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/12/2013
|
Application #:
|
13479622
|
Filing Dt:
|
05/24/2012
|
Publication #:
|
|
Pub Dt:
|
09/13/2012
| | | | |
Title:
|
NOVEL OPIOID ANTAGONISTS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/20/2014
|
Application #:
|
13494887
|
Filing Dt:
|
06/12/2012
|
Publication #:
|
|
Pub Dt:
|
05/16/2013
| | | | |
Title:
|
Tiacumicin Production
|
|
|
Patent #:
|
|
Issue Dt:
|
04/22/2014
|
Application #:
|
13496014
|
Filing Dt:
|
03/14/2012
|
Publication #:
|
|
Pub Dt:
|
07/05/2012
| | | | |
Title:
|
PREPARATION OF CRYSTALLINE FORMS OF DIHYDROPYRAZOLOPYRIMIDINONE
|
|
|
Patent #:
|
|
Issue Dt:
|
08/15/2017
|
Application #:
|
13496188
|
Filing Dt:
|
03/14/2012
|
Publication #:
|
|
Pub Dt:
|
09/20/2012
| | | | |
Title:
|
TRICYCLIC GYRASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/27/2014
|
Application #:
|
13496236
|
Filing Dt:
|
03/15/2012
|
Publication #:
|
|
Pub Dt:
|
07/12/2012
| | | | |
Title:
|
NOVEL PYRROLIDINES AS GLUCAGON RECEPTOR ANTAGONISTS, COMPOSITIONS, AND METHODS FOR THEIR USE
|
|
|
Patent #:
|
|
Issue Dt:
|
02/25/2014
|
Application #:
|
13496964
|
Filing Dt:
|
05/04/2012
|
Publication #:
|
|
Pub Dt:
|
08/23/2012
| | | | |
Title:
|
NOVEL COMPOUNDS THAT ARE ERK INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/18/2014
|
Application #:
|
13498605
|
Filing Dt:
|
03/28/2012
|
Publication #:
|
|
Pub Dt:
|
07/19/2012
| | | | |
Title:
|
CRYSTALLINE HYDROCHLORIDE SALTS OF C-MET KINASE INHIBITORS
|
|