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Patent #:
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Issue Dt:
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05/12/1987
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Application #:
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06590820
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Filing Dt:
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03/19/1984
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Title:
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2-(2-FUROYL)-4(5)-28FURANYL)-IH-IMIDAZOLE
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Patent #:
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Issue Dt:
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07/19/1988
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Application #:
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06798032
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Filing Dt:
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11/14/1985
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Title:
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METHOD AND AGENTS FOR INHIBITING PROTEIN AGING
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Patent #:
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Issue Dt:
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02/13/1990
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Application #:
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07091534
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Filing Dt:
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09/03/1987
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Title:
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METHOD AND AGENTS FOR REMOVING ADVANCED GLYCOSYLATION ENDPRODUCTS
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Patent #:
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Issue Dt:
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03/13/1990
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Application #:
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07119958
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Filing Dt:
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11/13/1987
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Title:
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INHIBITORS OF NONENZYMATIC CROSS-LINKING
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Patent #:
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Issue Dt:
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01/08/1991
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Application #:
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07264930
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Filing Dt:
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11/02/1988
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Title:
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INHIBITORS OF NONENZYMATIC CROSS-LINKING
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Patent #:
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Issue Dt:
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07/07/1992
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Application #:
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07481869
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Filing Dt:
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02/20/1990
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Title:
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METHOD AND AGENTS FOR INHIBITING PROTEIN AGING
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Patent #:
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Issue Dt:
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12/29/1992
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Application #:
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07503804
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Filing Dt:
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04/03/1990
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Title:
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INHIBITORS OF THE ADVANCED GLYCOSYLATION OF PROTEINS AND METHODS OF USE THEREFOR
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Patent #:
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Issue Dt:
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03/31/1992
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Application #:
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07606425
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Filing Dt:
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10/31/1990
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Title:
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BIGUANIDES AND DERIVATIVES THEREOF AS INHIBITORS OF ADVANCED GLYCOSYLATION OF A TARGET PROTEIN
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Patent #:
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Issue Dt:
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05/19/1992
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Application #:
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07640271
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Filing Dt:
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01/11/1991
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Title:
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AMINO-SUBSTITUTED PYRIMIDINES, DERIVATIVES AND METHODS OF USE THEREFOR
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Patent #:
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Issue Dt:
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11/02/1993
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Application #:
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07652575
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Filing Dt:
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02/08/1991
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Title:
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2-SUBSTITUTED-2-IMIDAZOLINES
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Patent #:
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Issue Dt:
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06/08/1993
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Application #:
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07672946
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Filing Dt:
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03/25/1991
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Title:
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INHIBITORS OF THE ADVANCED GLYCOSYLATION OF PROTEINS AND METHODS OF USE THEREFOR
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Patent #:
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Issue Dt:
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07/14/1992
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Application #:
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07697212
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Filing Dt:
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05/07/1991
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Title:
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2-ALKYLIDENE-AMINOGUANIDINES AND METHODS OF USE THEREFOR
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Patent #:
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Issue Dt:
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07/14/1992
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Application #:
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07697213
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Filing Dt:
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05/07/1991
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Title:
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AMIDRAZONES AND DERIVATIVES THEREOF
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Patent #:
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Issue Dt:
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12/17/1996
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Application #:
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07749438
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Filing Dt:
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08/23/1991
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Title:
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LIVER-DERIVED RECEPTORS FOR ADVANCED GLYCOSYLATION ENDPRODUCTS AND USES THEREOF
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Patent #:
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Issue Dt:
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04/13/1993
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Application #:
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07749444
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Filing Dt:
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08/23/1991
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Title:
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MESANGIAL CELL-DERIVED RECEPTORS FOR ADVANCED GLYCOSYLATION ENDPRODUCTS AND USES THEREOF
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Patent #:
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Issue Dt:
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08/24/1993
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Application #:
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07805200
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Filing Dt:
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12/10/1991
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Title:
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METHOD AND AGENTS FOR INHIBITING PROTEIN AGING
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Patent #:
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Issue Dt:
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10/19/1993
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Application #:
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07807609
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Filing Dt:
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12/16/1991
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Title:
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COMPOSITIONS CONTAINING BIGUANIDES AND DERIVATIVES THEREOF AS INHIBITORS OF NONENZYMATIC CROSS-LINKING
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Patent #:
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Issue Dt:
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08/02/1994
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Application #:
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07825598
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Filing Dt:
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01/27/1992
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Title:
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AMINO ACIDS USEFUL AS INHIBITORS OF THE ADVANCED GLYCOSYLATION OF PROTEINS
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Patent #:
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Issue Dt:
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10/18/1994
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Application #:
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07889141
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Filing Dt:
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05/27/1992
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Title:
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1,4 PIPERIZINO INHIBITORS OF NON-ENZYMATIC CROSS-LINKING OF PROTEEINS
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Patent #:
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Issue Dt:
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09/07/1993
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Application #:
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07890556
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Filing Dt:
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05/28/1992
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Title:
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2-ALKYLIDENE-AMINOGUANIDINES AND METHODS OF USE THEREFOR
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Patent #:
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Issue Dt:
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03/21/1995
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Application #:
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07956722
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Filing Dt:
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10/01/1992
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Title:
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1,2,4-TRIAZINE PRODUCTS RESULTING FROM THE INHIBITION OF ADVANCED GLY- COSYLATION
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Patent #:
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Issue Dt:
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04/29/1997
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Application #:
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07956849
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Filing Dt:
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10/01/1992
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Title:
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IMMUNOCHEMICAL DETECTION OF IN VIVO ADVANCED GLYCOSYLATION ENDPRODUCTS
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Patent #:
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Issue Dt:
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06/07/1994
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Application #:
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07986661
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Filing Dt:
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12/08/1992
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Title:
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INHIBITION OF THE ADVANCED GLYCOSYLATION OF PROTEINS USING SUBSTITUTED-1,2,4-TRIAZOLES
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Patent #:
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Issue Dt:
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10/25/1994
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Application #:
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07986662
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Filing Dt:
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12/08/1992
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Title:
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METHOD FOR INHIBITING ADVANCED GLYCOSYLATION OF PROTEINS USING AMINOSUBSTITUTED IMIDAZOLES
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Patent #:
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Issue Dt:
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07/05/1994
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Application #:
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07986673
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Filing Dt:
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12/08/1992
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Title:
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METHOD OF INHIBITING THE ADVANCED GLYCOSYLATION OF PROTEINS USING 1,2- DISIBSTITUTED-BENZIMIDAZLOES
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Patent #:
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Issue Dt:
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12/21/1993
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Application #:
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07998539
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Filing Dt:
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12/30/1992
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Title:
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2-ALKYLIDENE-AMINOGUANIDINES AND METHODS OF USE THEREFOR
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Patent #:
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Issue Dt:
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02/09/1999
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Application #:
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08029417
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Filing Dt:
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03/11/1993
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Title:
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GLYCOSYLATION OF LIPIDS AND LIPID-CONTAINING PARTICLES, AND DIAGNOSTIC AND THERAPEUTIC METHODS AND MATERIALS DERIVED THEREFROM
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Patent #:
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Issue Dt:
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12/19/1995
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Application #:
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08162538
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Filing Dt:
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12/03/1993
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Title:
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METHODS FOR GLYCOSYLATION INHIBITION USING AMINO-BENZOIC ACIDS AND DERIVATIVES
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Patent #:
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Issue Dt:
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03/11/1997
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Application #:
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08236416
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Filing Dt:
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04/29/1994
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Title:
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METHOD FOR DETECTING HEMOGLOBIN ADVANCED GLYCOSYLATION ENDPRODUCTS
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Patent #:
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Issue Dt:
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07/09/1996
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08318754
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Filing Dt:
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12/22/1994
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Title:
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AMINOGUANIDINE SPRAY DRYING PROCESS
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Patent #:
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Issue Dt:
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12/23/1997
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08319747
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10/07/1994
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Title:
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METHODS AND MATERIALS FOR THE DIAGNOSIS AND TREATMENT OF CONDITIONS SUCH AS STROKE
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Patent #:
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04/28/1998
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08367507
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12/30/1994
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Title:
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MONOCLONAL ANTIBODY FOR THE DETECTION ADVANCED GLYCOSYLATION ENDPRO- DUCTS IN BIOLOGICAL
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Patent #:
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Issue Dt:
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12/16/1997
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Application #:
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08372672
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Filing Dt:
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01/13/1995
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Title:
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BIS-[HYDRAZONES]
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Patent #:
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Issue Dt:
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08/12/1997
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08375155
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01/18/1995
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Title:
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PREVENTING AND REVERSING ADVANCED GLYCOSYLATION ENDPRODUCTS
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Patent #:
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Issue Dt:
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05/07/1996
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Application #:
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08383764
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02/03/1995
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Title:
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AMINO-BENZOIC ACIDS AND DERIVATIVES, AND METHODS OF USE
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Patent #:
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Issue Dt:
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09/01/1998
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08418525
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04/07/1995
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Title:
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METHODS AND MATERIALS FOR THE DIAGNOSIS AND TREATMENT OF CONDITIONS SUCH AS STROKE
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Patent #:
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02/25/1997
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08437064
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05/09/1995
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Title:
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METHOD AND AGENTS FOR REMOVING ADVANCED GLYCOSYLATION ENDPRODUCTS
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Patent #:
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Issue Dt:
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01/27/1998
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Application #:
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08472398
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Filing Dt:
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06/07/1995
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Title:
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IMMUNOCHEMICAL DETECTION OF IN VIVO ADVANCED GLYCOSYLATION ENDPRODUCTS
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Patent #:
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Issue Dt:
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03/31/1998
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08473009
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06/07/1995
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Title:
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METHODS AND MATERIALS FOR THE DIAGNOSIS AND TREATMENT OF CONDITIONS SUCH AS STROKE
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Patent #:
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05/13/1997
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08476381
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06/07/1995
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Title:
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IMMUNOCHEMICAL ISOLATION OF IN VIVO ADVANCED GLYCOSYLATION ENDPRODUCTS
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06/25/2002
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08477364
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06/07/1995
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Title:
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COMPOSITIONS AND METHODS FOR ADVANCED GLYCOSYLATION ENDPRODUCT-MEDIATED MODULATION OF AMYLOIDOSIS
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12/22/1998
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08479149
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06/07/1995
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Title:
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ANTIBODIES TO LIVER DERIVED RECEPTORS FOR ADVANCED GLYCOSYLATION END- PRODUCTS AND USES THEREFOR
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03/31/1998
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08479673
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06/07/1995
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Title:
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METHODS AND MATERIALS FOR THE DIAGNOSIS AND TREATMENT OF CONDITIONS SUCH AS STROKE
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06/16/1998
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08483184
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06/07/1995
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Title:
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THERAPEUTIC METHODS AND PHARMACEUTICAL COMPOSITIONS
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12/16/1997
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08483186
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06/07/1995
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Title:
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MONOCLONAL ANTIBODY SPECIFIC FOR ADVANCED GLYCOSYLATION ENDPRODUCTS IN BIOLOGICAL SAMPLES
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03/31/1998
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08484869
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06/07/1995
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Title:
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IMMUNOCHEMICAL DETECTION OF IN VIVO ADVANCED GLYCOSYLATION ENDPRODUCTS
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08/26/1997
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08485387
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06/07/1995
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BIS-(2-ARYL) HYDRAZONES
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01/05/1999
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08485948
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06/07/1995
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Title:
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METHODS FOR INHIBITING THE CROSS-LINKING OF ADVANCED GLYCOSYLATION ENDPRODUCTS
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12/30/1997
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08486513
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06/07/1995
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ANTIBODIES TO IN VIVO ADVANCED GLYCOSYLATION ENDPRODUCTS
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07/14/1998
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08486605
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06/07/1995
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Title:
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GLYCOSYLATION OF LIPIDS AND LIPID-CONTAINING PARTICLES AND DIAGNOSTIC AND THERAPEUTIC METHODS AND MATERIALS DERIVED THEREFROM
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11/04/1997
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08487055
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06/07/1995
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Title:
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IMMUNOCHEMICAL DETECTION OF IN VIVO ADVANCED GLYCOSYLATION ENDPRODUCTS
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01/19/1999
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08487058
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06/07/1995
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Title:
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METHODS FOR PARTITIONING ADVANCED GLYCOSYLATION ENDDPRODUCTS
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09/22/1998
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08487398
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06/07/1995
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METHOD AND AGENTS FOR REMOVING ADVANCED GLYCOSYLATION ENDPRODUCTS
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08/10/1999
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08501127
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08/10/1996
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Title:
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COMPOSITIONS AND METHODS FOR STIMULATING AMYLOID REMOVAL IN AMYLOIDOGENIC DISEASES USING ADVANCED ENDPRODUCTS
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04/06/1999
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08581724
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12/29/1995
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Title:
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MONOCLONAL ANTIBODIES SPECIFIC FOR ADVANCED GLYCOSYLATION ENDPRODUCTS IN BIOLOGICAL SAMPLES
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12/29/1998
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08588249
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01/18/1996
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Title:
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PREVENTING AND REVERSING THE FORMATION OF ADVANCED GLYCOSYLATION ENDPRODUCTS
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04/06/1999
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08628380
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04/05/1996
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COMPOSITIONS AND DEVICES FOR PARTITIONING ADVANCED GLYCOSYLATION ENDPRODUCTS, AND METHODS OF THEIR USE
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11/18/1997
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08673217
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06/27/1996
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3-ALKYLAMINO-2-HYDROXY-4-HYDROXYMETHYL-2-CYCLOPENTEN-1-ONE ADVANCED GLYCOSYLATION ENDPRODUCTS AND METHODS OF USE THEREFOR
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06/23/1998
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11/15/1996
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METHOD AND AGENTS FOR INHIBITING PROTEIN AGING
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02/09/1999
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08771958
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12/23/1996
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6-(N-CARBOXYMETHYLAMINO)CAPROATE, SALTS THEREOF AND METHODS OF USE THEREFOR
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03/02/1999
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08771959
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12/23/1996
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N-ACYLAMINOALKYL-HYDRAZINECARBOXIMIDAMIDES
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12/22/1998
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01/16/1997
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COMPOSTIONS, INCLUDING PHARMAEUTICAL COMPOSITIONS, FOR INHIBITING THE ADVANCED GLYCOSYLATION OF PROTEINS, AND THERAPEUTIC METHODS BASED THEREON
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08/03/1999
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03/27/1997
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TRIAZINE COMPOUNDS AND METHODS OF USE THEREFOR
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12/28/1999
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11/19/1997
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PREVENTING AND REVERSING THE FORMATION OF ADVANCED GLYCOSYLATION ENDPRODUCTS
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02/15/2000
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04/17/1998
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08/29/2000
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11/10/1998
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METHODS FOR TREATMENT PREDICATED ON THE PRESENCE OF ADVANCED GLYCOSYLATION ENDPRODUCTS IN TOBACCO AND ITS COMBUSTION BYPRODUCTS
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09/19/2000
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11/10/1998
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REVERSING ADVANCED GLYCOSYLATION CROSS-LINKS USING HETEROCYCLIC-SUBSTITUTED THIAZOLIUM SALTS
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05/09/2000
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01/20/1999
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TRIAZINE COMPOUNDS AND METHODS OF USE THEREFOR
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11/25/2003
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09373345
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08/12/1999
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PREVENTING AND REVERSING ADVANCED GLYCOSYLATION ENDPRODUCTS
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12/04/2001
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11/12/1999
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GLUCOSE AND LIPID LOWERING COMPOUNDS
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06/20/2006
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12/16/1999
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MONOCLONAL ANTIBODY SPECIFIC FOR ADVANCED GLYCOSYLATION ENDPRODUCTS IN BIOLOGICAL SAMPLES
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08/27/2002
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12/22/1999
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04/30/2002
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Triazine compounds and method of use therefor
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11/20/2001
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Filing Dt:
|
08/23/2000
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Title:
|
Reversing advanced Glycosylation cross-links using Heterocyclic-substituted Thiazolium compounds
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|
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Patent #:
|
|
Issue Dt:
|
11/01/2005
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Application #:
|
09766547
|
Filing Dt:
|
01/19/2001
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Publication #:
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Pub Dt:
|
02/21/2002
| | | | |
Title:
|
THIAZOLE, IMIDAZOLE AND OXAZOLE COMPOUNDS AND TREATMENTS OF DISORDERS ASSOCIATED WITH PROTEIN AGING
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|
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Patent #:
|
|
Issue Dt:
|
10/01/2002
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Application #:
|
09792422
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Filing Dt:
|
02/23/2001
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Publication #:
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Pub Dt:
|
05/09/2002
| | | | |
Title:
|
THIAZOLIUM COMPOUNDS AND TREATMENTS OF DISORDERS ASSOCIATED WITH PROTEIN AGING
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|
|
Patent #:
|
|
Issue Dt:
|
01/14/2003
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Application #:
|
09821846
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Filing Dt:
|
03/29/2001
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Publication #:
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Pub Dt:
|
01/31/2002
| | | | |
Title:
|
SYNTHESIS OF THIAZOLIUM COMPOUNDS
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|
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Patent #:
|
|
Issue Dt:
|
08/26/2003
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Application #:
|
09905035
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Filing Dt:
|
07/13/2001
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Publication #:
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Pub Dt:
|
08/01/2002
| | | | |
Title:
|
CYANOMETHYL SUBSTITUTED THIAZOLIUMS AND IMIDAZOLIUMS AND TREATMENTS OF DISORDERS ASSOCIATED WITH PROTEIN AGING
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|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
09905188
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Filing Dt:
|
07/13/2001
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Publication #:
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Pub Dt:
|
06/06/2002
| | | | |
Title:
|
Method for treating fibrotic diseases or other indications IC
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|
Patent #:
|
NONE
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Issue Dt:
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|
Application #:
|
10036856
|
Filing Dt:
|
12/31/2001
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Publication #:
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|
Pub Dt:
|
08/29/2002
| | | | |
Title:
|
Method for treating glaucoma IIB
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|
|
Patent #:
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|
Issue Dt:
|
01/23/2007
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Application #:
|
10037447
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Filing Dt:
|
12/31/2001
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Publication #:
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|
Pub Dt:
|
11/28/2002
| | | | |
Title:
|
METHOD FOR TREATING FIBROTIC DISEASES AND OTHER INDICATIONS
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|
|
Patent #:
|
|
Issue Dt:
|
10/07/2008
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Application #:
|
10038112
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Filing Dt:
|
12/31/2001
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Publication #:
|
|
Pub Dt:
|
10/31/2002
| | | | |
Title:
|
METHOD FOR TREATING GLAUCOMA IC
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|
|
Patent #:
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|
Issue Dt:
|
07/22/2003
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Application #:
|
10038116
|
Filing Dt:
|
12/31/2001
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Publication #:
|
|
Pub Dt:
|
12/05/2002
| | | | |
Title:
|
METHOD FOR TREATING FIBROTIC DISEASES OR OTHER INDICATIONS UTILIZING THIAZOLE OXAZOLE AND IMIDAZOLE COMPOUNDS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/21/2003
|
Application #:
|
10047182
|
Filing Dt:
|
10/23/2001
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Publication #:
|
|
Pub Dt:
|
10/17/2002
| | | | |
Title:
|
GLUCOSE AND LIPID LOWERING COMPOUNDS
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|
|
Patent #:
|
|
Issue Dt:
|
07/22/2003
|
Application #:
|
10158344
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Filing Dt:
|
05/30/2002
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Publication #:
|
|
Pub Dt:
|
01/02/2003
| | | | |
Title:
|
METHOD FOR TREATING FIBROTIC DISEASES WITH AZOLIUM CHROMAN COMPOUNDS
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|
|
Patent #:
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|
Issue Dt:
|
10/19/2004
|
Application #:
|
10158683
|
Filing Dt:
|
05/30/2002
|
Publication #:
|
|
Pub Dt:
|
12/19/2002
| | | | |
Title:
|
METHOD FOR TREATING GLAUCOMA V
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|
|
Patent #:
|
|
Issue Dt:
|
03/30/2004
|
Application #:
|
10158685
|
Filing Dt:
|
05/30/2002
|
Publication #:
|
|
Pub Dt:
|
01/02/2003
| | | | |
Title:
|
METHOD FOR TREATING GLAUCOMA VI
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|
|
Patent #:
|
|
Issue Dt:
|
09/14/2004
|
Application #:
|
10348378
|
Filing Dt:
|
01/21/2003
|
Publication #:
|
|
Pub Dt:
|
09/18/2003
| | | | |
Title:
|
REVERSING ADVANCED GLYCOSYLATION CROSS-LINKS USING HETEROCYCLIC-SUBSTITUTED THIAZOLIUM COMPOUNDS
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|
|
Patent #:
|
|
Issue Dt:
|
04/04/2006
|
Application #:
|
10418398
|
Filing Dt:
|
04/18/2003
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Publication #:
|
|
Pub Dt:
|
02/19/2004
| | | | |
Title:
|
PREVENTING AND REVERSING THE FORMATION OF ADVANCE GLYCOSYLATION ENDPRODUCTS
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|
|
Patent #:
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|
Issue Dt:
|
08/03/2004
|
Application #:
|
10440896
|
Filing Dt:
|
05/19/2003
|
Publication #:
|
|
Pub Dt:
|
12/04/2003
| | | | |
Title:
|
METHOD FOR TREATING FIBROTIC DISEASES OR OTHER INDICATIONS UTILIZING THIAZOLE, OXAZOLE AND IMIDAZOLE COMPOUNDS
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|
|
Patent #:
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|
Issue Dt:
|
12/05/2006
|
Application #:
|
10444356
|
Filing Dt:
|
05/22/2003
|
Publication #:
|
|
Pub Dt:
|
06/24/2004
| | | | |
Title:
|
SUNSCREEN COMPOSITIONS AND METHODS OF USE THEREOF
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|
|
Patent #:
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|
Issue Dt:
|
07/18/2006
|
Application #:
|
10805757
|
Filing Dt:
|
03/22/2004
|
Publication #:
|
|
Pub Dt:
|
03/24/2005
| | | | |
Title:
|
SUNSCREEN COMPOSITIONS AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
10828051
|
Filing Dt:
|
04/20/2004
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Publication #:
|
|
Pub Dt:
|
10/07/2004
| | | | |
Title:
|
Substituted imidazoliums and methods of use therefor
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|
|
Patent #:
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|
Issue Dt:
|
04/11/2006
|
Application #:
|
10852859
|
Filing Dt:
|
05/24/2004
|
Publication #:
|
|
Pub Dt:
|
02/10/2005
| | | | |
Title:
|
METHOD FOR TREATING FIBROTIC DISEASES OR OTHER INDICATIONS UTILIZING THIAZOLE, OXAZOLE AND IMIDAZOLE COMPOUNDS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
10873056
|
Filing Dt:
|
06/21/2004
|
Publication #:
|
|
Pub Dt:
|
11/25/2004
| | | | |
Title:
|
Method for treating fibrotic diseases or other indications IE
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|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
11204231
|
Filing Dt:
|
08/15/2005
|
Publication #:
|
|
Pub Dt:
|
01/19/2006
| | | | |
Title:
|
Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging
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|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
11295213
|
Filing Dt:
|
12/05/2005
|
Publication #:
|
|
Pub Dt:
|
12/21/2006
| | | | |
Title:
|
Method for treating glaucoma III B
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
11296544
|
Filing Dt:
|
12/06/2005
|
Publication #:
|
|
Pub Dt:
|
12/14/2006
| | | | |
Title:
|
Method for treating glaucoma IV B
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
11351390
|
Filing Dt:
|
02/09/2006
|
Publication #:
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|
Pub Dt:
|
02/22/2007
| | | | |
Title:
|
Method of treating fibrotic diseases or other indications with imidazolium agents
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
11351655
|
Filing Dt:
|
02/09/2006
|
Publication #:
|
|
Pub Dt:
|
02/01/2007
| | | | |
Title:
|
Preventing and reversing the formation of advance glycosylation endproducts
|
|