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10/12/2010
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10590848
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07/03/2007
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Pub Dt:
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02/14/2008
| | | | |
Title:
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STEROID AGONIST FOR FXR
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11/22/2016
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11081002
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03/14/2005
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03/30/2006
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Title:
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08/31/2010
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11602307
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11/21/2006
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06/21/2007
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Title:
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STEROIDS AS AGONISTS FOR FXR
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04/26/2011
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11819517
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06/27/2007
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07/31/2008
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Title:
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BILE ACID DERIVATIVES AS FXR LIGANDS FOR THE PREVENTION OR TREATMENT OF FXR-MEDIATED DISEASES OR CONDITIONS
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08/09/2011
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11914559
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11/16/2007
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09/04/2008
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Title:
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PROCESS FOR PREPARING 3A(BETA)-7A(BETA)-DIHYDROXY-6A(BETA)-ALKYL-5BETA-CHOLANIC ACID
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12/28/2010
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12435063
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05/04/2009
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Pub Dt:
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03/11/2010
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Title:
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BILE ACID DERIVATIVES AS FXR LIGANDS FOR THE PREVENTION OR TREATMENT OF FXR-MEDIATED DISEASES OR CONDITIONS
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04/02/2013
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12523670
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04/30/2010
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Pub Dt:
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01/06/2011
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Title:
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23-SUBSTITUTED BILE ACIDS AS TGR5 MODULATORS AND METHODS OF USE THEREOF
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11/15/2011
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12547147
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08/25/2009
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01/28/2010
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Title:
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STEROIDS AS AGONISTS FOR FXR
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02/14/2012
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12622123
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11/19/2009
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06/17/2010
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Title:
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TGR5 MODULATORS AND METHODS OF USE THEROF
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08/05/2014
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13056797
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03/22/2011
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07/14/2011
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Title:
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TGR5 Modulators And Methods Of Use Thereof
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10/01/2013
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13082261
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04/07/2011
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11/08/2012
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Title:
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Bile Acid Derivatives As FXR Ligands For The Prevention Or Treatment Of FXR-Mediated Diseases Or Conditions
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04/07/2015
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13129947
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07/18/2011
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10/27/2011
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Title:
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TGR5 Modulators and Methods of Use Thereof
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02/19/2013
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13288558
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11/03/2011
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03/01/2012
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Title:
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STEROIDS AS AGONISTS FOR FXR
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05/21/2013
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13313689
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12/07/2011
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05/10/2012
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Title:
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TGR5 MODULATORS AND METHODS OF USE THEREOF
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03/03/2015
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13761889
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02/07/2013
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01/23/2014
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Title:
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STEROIDS AS AGONISTS FOR FXR
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01/26/2016
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13854579
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04/03/2014
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TGR5 Modulators and Methods of Use Thereof
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05/16/2017
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13871492
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04/26/2013
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04/10/2014
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TGR5 Modulators and Methods of Use Thereof
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01/19/2016
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13919734
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06/17/2013
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12/26/2013
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Title:
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Preparation and Uses of Obeticholic Acid
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07/28/2015
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14012401
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08/28/2013
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Pub Dt:
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02/27/2014
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Title:
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04/04/2017
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14120366
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05/14/2014
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12/18/2014
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Title:
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10/03/2017
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14438323
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04/24/2015
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10/15/2015
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Title:
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01/10/2017
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14449995
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08/01/2014
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02/25/2016
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Title:
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TGR5 MODULATORS AND METHODS OF USE THEREOF
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09/19/2017
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14743295
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06/18/2015
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12/17/2015
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Title:
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Bile Acid Derivatives as FXR Ligands for the Prevention or Treatment of FXR-Mediated Diseases or Conditions
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08/15/2017
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14947492
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11/20/2015
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06/23/2016
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Preparation and Uses of Obeticholic Acid
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08/14/2018
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14947658
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11/20/2015
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03/17/2016
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Preparation and Uses of Obeticholic Acid
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12/18/2018
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14947680
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11/20/2015
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07/28/2016
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Title:
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05/29/2018
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14979005
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12/22/2015
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04/21/2016
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Title:
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Preparation and Uses of Obeticholic Acid
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08/15/2017
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15016802
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02/05/2016
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06/02/2016
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STEROIDS AS AGONISTS FOR FXR
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08/21/2018
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15139138
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04/26/2016
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02/09/2017
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Title:
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COMPOSITIONS OF OBETICHOLIC ACID AND METHODS OF USE
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06/15/2021
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15288390
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10/07/2016
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04/13/2017
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FARNESOID X RECEPTOR MODULATORS
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04/16/2019
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15299559
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10/21/2016
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06/15/2017
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Title:
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TREATMENT OF FIBROSIS USING FXR LIGANDS
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10/27/2020
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15451818
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03/07/2017
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09/14/2017
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08/06/2019
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15484379
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04/11/2017
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10/19/2017
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METHODS OF TREATING CANCER
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01/08/2019
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15496398
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04/25/2017
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08/10/2017
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Preparation and Uses of Obeticholic Acid
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04/26/2022
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15548537
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08/03/2017
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01/11/2018
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PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY
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01/19/2021
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15564799
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10/06/2017
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05/03/2018
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09/24/2019
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15645136
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07/10/2017
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10/03/2019
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STEROIDS AS AGONISTS FOR FXR
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02/12/2019
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15681609
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08/21/2017
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03/22/2018
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Title:
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PROCESS FOR PREPARING BILE ACID DERIVATIVES
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NONE
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15711205
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09/21/2017
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09/13/2018
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Title:
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METHODS OF TREATING CANCER
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10/13/2020
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15742595
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09/26/2018
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09/19/2019
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Title:
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TGR5 MODULATORS AND METHODS OF USE THEREOF
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09/17/2019
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15748716
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01/30/2018
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01/10/2019
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Title:
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METHODS FOR PREPARATION OF BILE ACIDS AND DERIVATIVES THEREOF
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03/31/2020
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15750683
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02/06/2018
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08/09/2018
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Title:
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METHODS FOR PREPARATION OF BILE ACIDS AND DERIVATIVES THEREOF
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02/04/2020
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15760769
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03/16/2018
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09/13/2018
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Title:
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07/27/2021
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03/23/2018
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07/30/2020
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Title:
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03/31/2020
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05/04/2018
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02/28/2019
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METHODS FOR THE PREPARATION OF OBETICHOLIC ACID AND DERIVATIVES THEREOF
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07/20/2021
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06/22/2018
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12/27/2018
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METHODS AND INTERMEDIATES FOR THE PREPARATION OF BILE ACID DERIVATIVES
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05/12/2020
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07/09/2018
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03/14/2019
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COMPOSITIONS OF OBETICHOLIC ACID AND METHODS OF USE
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08/23/2022
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09/27/2018
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08/15/2019
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Title:
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Medicine Obtained by Combining FXR Agonist and ARB
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08/16/2022
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16089477
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09/28/2018
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07/18/2019
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05/17/2022
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09/28/2018
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08/27/2020
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02/04/2020
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16094535
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10/18/2018
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07/11/2019
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METHODS FOR THE PREPARATION OF OBETICHOLIC ACID AND DERIVATIVES THEREOF
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01/14/2020
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09/06/2018
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07/11/2019
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FARNESOID X RECEPTOR MODULATORS
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04/27/2021
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16228944
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12/21/2018
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12/24/2020
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Title:
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TREATMENT OF FIBROSIS USING FXR LIGANDS
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08/25/2020
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16248512
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01/15/2019
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08/22/2019
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COMPOSITIONS OF OBETICHOLIC ACID AND METHODS OF USE
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NONE
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16337982
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03/29/2019
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01/23/2020
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CRYSTALLINE FORMS OF A BILE ACID DERIVATIVE
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10/27/2020
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16448503
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06/21/2019
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Title:
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Steroids As Agonists For FXR
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NONE
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16486873
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08/19/2019
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05/28/2020
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Title:
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PHARMACEUTICAL COMPOSITIONS OF A BILE ACID DERIVATIVE AND MICROBIOME AND USES THEREOF
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NONE
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16491798
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09/06/2019
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05/13/2021
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Title:
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CRYSTALLINE FORMS OF OBETICHOLIC ACID
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NONE
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16596741
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10/08/2019
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02/13/2020
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Title:
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COMPOSITIONS OF OBETICHOLIC ACID AND METHODS OF USE
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10/18/2022
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16632093
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01/17/2020
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05/28/2020
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ISOTOPICALLY LABELED BILE ACID DERIVATIVES
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05/11/2021
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16695528
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Filing Dt:
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11/26/2019
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Publication #:
|
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Pub Dt:
|
09/24/2020
| | | | |
Title:
|
FARNESOID X RECEPTOR MODULATORS
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|
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Patent #:
|
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Issue Dt:
|
09/01/2020
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Application #:
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16787796
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Filing Dt:
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02/11/2020
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Publication #:
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Pub Dt:
|
06/04/2020
| | | | |
Title:
|
COMPOSITIONS OF OBETICHOLIC ACID AND METHODS OF USE
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|
|
Patent #:
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NONE
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Issue Dt:
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|
Application #:
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16831365
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Filing Dt:
|
03/26/2020
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Publication #:
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Pub Dt:
|
10/08/2020
| | | | |
Title:
|
METHODS OF DIAGNOSIS AND TREATMENT OF LIVER DISEASES USING OBETICHOLIC ACID
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|
|
Patent #:
|
|
Issue Dt:
|
05/31/2022
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Application #:
|
17010505
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Filing Dt:
|
09/02/2020
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Publication #:
|
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Pub Dt:
|
04/29/2021
| | | | |
Title:
|
TGR5 MODULATORS AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
05/03/2022
|
Application #:
|
17025475
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Filing Dt:
|
09/18/2020
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Publication #:
|
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Pub Dt:
|
04/08/2021
| | | | |
Title:
|
3-DESOXY DERIVATIVE AND PHARMACEUTICAL COMPOSITIONS THEREOF
|
|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
17092612
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Filing Dt:
|
11/09/2020
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Publication #:
|
|
Pub Dt:
|
09/02/2021
| | | | |
Title:
|
TGR5 MODULATORS AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
NONE
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Issue Dt:
|
|
Application #:
|
17142870
|
Filing Dt:
|
01/06/2021
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Publication #:
|
|
Pub Dt:
|
12/23/2021
| | | | |
Title:
|
PREPARATION AND USES OF OBETICHOLIC ACID
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17211033
|
Filing Dt:
|
03/24/2021
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Publication #:
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|
Pub Dt:
|
11/11/2021
| | | | |
Title:
|
TREATMENT OF FIBROSIS USING FXR LIGANDS
|
|
|
Patent #:
|
NONE
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Issue Dt:
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|
Application #:
|
17228819
|
Filing Dt:
|
04/13/2021
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Publication #:
|
|
Pub Dt:
|
07/29/2021
| | | | |
Title:
|
FARNESOID X RECEPTOR MODULATORS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17320286
|
Filing Dt:
|
05/14/2021
|
Publication #:
|
|
Pub Dt:
|
09/02/2021
| | | | |
Title:
|
FARNESOID X RECEPTOR MODULATORS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17342057
|
Filing Dt:
|
06/08/2021
|
Publication #:
|
|
Pub Dt:
|
04/28/2022
| | | | |
Title:
|
METHODS AND INTERMEDIATES FOR THE PREPARATION OF BILE ACID DERIVATIVES
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17384555
|
Filing Dt:
|
07/23/2021
|
Publication #:
|
|
Pub Dt:
|
06/16/2022
| | | | |
Title:
|
METHODS OF USING OBETICHOLIC ACID
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17428029
|
Filing Dt:
|
08/03/2021
|
Publication #:
|
|
Pub Dt:
|
03/31/2022
| | | | |
Title:
|
TREATMENT AND PREVENTION OF INTESTINAL INFLAMMATORY DISEASES WITH A BILE ACID DERIVATIVE
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17542923
|
Filing Dt:
|
12/06/2021
|
Publication #:
|
|
Pub Dt:
|
05/05/2022
| | | | |
Title:
|
COMPOSITIONS OF OBETICHOLIC ACID AND METHODS OF USE
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17615186
|
Filing Dt:
|
11/30/2021
|
Publication #:
|
|
Pub Dt:
|
07/21/2022
| | | | |
Title:
|
PHARMACEUTICAL COMPOSITIONS COMPRISING A FXR AGONIST AND A FIBRATE FOR USE IN THE TREATMENT OF CHOLESTATIC LIVER DISEASE
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17700317
|
Filing Dt:
|
03/21/2022
|
Publication #:
|
|
Pub Dt:
|
09/08/2022
| | | | |
Title:
|
PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17700392
|
Filing Dt:
|
03/21/2022
|
Publication #:
|
|
Pub Dt:
|
09/08/2022
| | | | |
Title:
|
PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY
|
|
|
Patent #:
|
|
Issue Dt:
|
11/07/2023
|
Application #:
|
17720938
|
Filing Dt:
|
04/14/2022
|
Publication #:
|
|
Pub Dt:
|
12/01/2022
| | | | |
Title:
|
TGR5 MODULATORS AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
17939326
|
Filing Dt:
|
09/07/2022
|
Publication #:
|
|
Pub Dt:
|
02/23/2023
| | | | |
Title:
|
ISOTOPICALLY LABELED BILE ACID DERIVATIVES
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
18188341
|
Filing Dt:
|
03/22/2023
|
Publication #:
|
|
Pub Dt:
|
10/26/2023
| | | | |
Title:
|
PREPARATION AND USES OF OBETICHOLIC ACID
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
18295091
|
Filing Dt:
|
04/03/2023
|
Publication #:
|
|
Pub Dt:
|
07/27/2023
| | | | |
Title:
|
FARNESOID X RECEPTOR MODULATORS
|
|