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06/05/2007
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Application #:
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10738965
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Filing Dt:
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12/17/2003
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Publication #:
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Pub Dt:
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09/23/2004
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Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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02/03/2009
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Application #:
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10741164
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Filing Dt:
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12/19/2003
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Publication #:
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Pub Dt:
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09/23/2004
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Title:
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INHIBITORS OF TACE
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Patent #:
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Issue Dt:
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11/03/2009
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Application #:
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10743563
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Filing Dt:
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12/22/2003
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Publication #:
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Pub Dt:
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09/30/2004
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Title:
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CASPASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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10/07/2008
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Application #:
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10749121
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Filing Dt:
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12/30/2003
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Publication #:
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Pub Dt:
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08/26/2004
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Title:
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SULFHYDANTOINS AS PHOSPHATE ISOSTERES
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Patent #:
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Issue Dt:
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10/21/2008
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Application #:
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10750326
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Filing Dt:
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12/31/2003
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Publication #:
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Pub Dt:
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09/23/2004
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Title:
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INHIBITORS OF PHOSPHATASES
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Patent #:
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Issue Dt:
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02/24/2009
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Application #:
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10767638
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Filing Dt:
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01/29/2004
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Publication #:
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Pub Dt:
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11/25/2004
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Title:
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GYRASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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08/07/2007
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Application #:
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10770814
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Filing Dt:
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02/03/2004
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Pub Dt:
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11/18/2004
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Title:
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HETEROCYCLIC INHIBITORS OF ERK2 AND USES THEREOF
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Patent #:
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Issue Dt:
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02/13/2007
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Application #:
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10770861
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Filing Dt:
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02/02/2004
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Publication #:
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Pub Dt:
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09/16/2004
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Title:
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HIGH THROUGHPUT METHOD AND SYSTEM FOR SCREENING CANDIDATE COMPOUNDS FOR ACTIVITY AGAINST TARGET ION CHANNELS
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Patent #:
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Issue Dt:
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08/05/2008
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Application #:
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10771165
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Filing Dt:
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02/03/2004
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Publication #:
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Pub Dt:
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10/28/2004
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Title:
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HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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12/06/2011
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Application #:
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10771283
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Filing Dt:
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02/02/2004
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Publication #:
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Pub Dt:
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09/30/2004
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Title:
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HIGH THROUGHPUT METHOD AND SYSTEM FOR SCREENING CANDIDATE COMPOUNDS FOR ACTIVITY AGAINST TARGET ION CHANNELS
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Patent #:
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Issue Dt:
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10/13/2009
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Application #:
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10772219
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Filing Dt:
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02/04/2004
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Publication #:
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Pub Dt:
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09/30/2004
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Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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10/03/2006
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Application #:
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10775687
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Filing Dt:
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02/10/2004
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Publication #:
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Pub Dt:
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11/18/2004
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Title:
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PROCESSES FOR THE FACILE SYNTHESIS OF DIARYL AMINES AND ANALOGUES THEREOF
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Patent #:
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Issue Dt:
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09/23/2008
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Application #:
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10775699
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Filing Dt:
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02/10/2004
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Publication #:
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Pub Dt:
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08/26/2004
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Title:
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PYRAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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11/02/2010
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Application #:
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10781015
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Filing Dt:
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02/17/2004
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Publication #:
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Pub Dt:
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12/30/2004
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Title:
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METHOD OF MODELING COMPLEX FORMATION BETWEEN A QUERY LIGAN AND A TARGET MOLECULE
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Patent #:
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Issue Dt:
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01/22/2008
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Application #:
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10786997
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Filing Dt:
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02/24/2004
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Publication #:
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Pub Dt:
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08/26/2004
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Title:
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NOVEL SULFONAMIDE INHIBITORS OF ASPARTYL PROTEASE
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Patent #:
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Issue Dt:
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05/11/2010
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Application #:
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10790507
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Filing Dt:
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03/01/2004
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Publication #:
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Pub Dt:
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11/25/2004
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Title:
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TARGET LIGAND GENERATION
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Patent #:
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Issue Dt:
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03/16/2010
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Application #:
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10792688
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Filing Dt:
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03/03/2004
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Publication #:
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Pub Dt:
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12/09/2004
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Title:
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QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS
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Patent #:
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Issue Dt:
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11/25/2008
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Application #:
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10798766
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Filing Dt:
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03/11/2004
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Publication #:
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Pub Dt:
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11/04/2004
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Title:
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COMPOSITIONS USEFUL AS PROTEIN KINASE INHIBITORS
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Patent #:
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Issue Dt:
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05/15/2007
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Application #:
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10799507
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Filing Dt:
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03/12/2004
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Publication #:
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Pub Dt:
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09/23/2004
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Title:
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4-SUBSTITUTED-5-CYANO-1H-PYRIMIDIN-6-(THI) ONES AS GSK-3 INHIBITORS
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Patent #:
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Issue Dt:
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06/16/2009
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Application #:
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10808678
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Filing Dt:
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03/25/2004
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Publication #:
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Pub Dt:
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10/07/2004
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Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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10/02/2007
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Application #:
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10809946
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Filing Dt:
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03/25/2004
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Publication #:
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Pub Dt:
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01/06/2005
| | | | |
Title:
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THIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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04/29/2008
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Application #:
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10821663
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Filing Dt:
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04/09/2004
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Publication #:
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Pub Dt:
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04/14/2005
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Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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Patent #:
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Issue Dt:
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07/18/2006
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Application #:
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10833496
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Filing Dt:
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04/27/2004
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Publication #:
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Pub Dt:
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10/27/2005
| | | | |
Title:
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CLEANABLE VOLUME DISPLACEMENT PIPETTER
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Patent #:
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|
Issue Dt:
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04/15/2008
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Application #:
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10833995
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Filing Dt:
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04/28/2004
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Title:
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GYRASE INHIBITORS AND USES THEREOF
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|
|
Patent #:
|
|
Issue Dt:
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02/27/2007
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Application #:
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10837848
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Filing Dt:
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05/03/2004
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Publication #:
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Pub Dt:
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10/21/2004
| | | | |
Title:
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PYRAZOLE-DERIVED KINASE INHIBITORS AND USES THEREOF
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|
|
Patent #:
|
|
Issue Dt:
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06/30/2009
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Application #:
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10853901
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Filing Dt:
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05/25/2004
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Publication #:
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Pub Dt:
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12/01/2005
| | | | |
Title:
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MODULAR TEST TUBE RACK
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Patent #:
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Issue Dt:
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02/04/2014
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Application #:
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10862909
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Filing Dt:
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06/07/2004
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Publication #:
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Pub Dt:
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03/17/2005
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Title:
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Modulators of ATP-Binding Cassette transporters
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Patent #:
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Issue Dt:
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11/08/2005
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Application #:
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10883305
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Filing Dt:
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07/01/2004
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Publication #:
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Pub Dt:
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12/16/2004
| | | | |
Title:
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INHIBITORS OF P38
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Patent #:
|
|
Issue Dt:
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10/19/2010
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Application #:
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10884865
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Filing Dt:
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07/02/2004
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Publication #:
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Pub Dt:
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03/03/2005
| | | | |
Title:
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PYRIMIDINES USEFUL AS MODULATORS OF VOLTAGE-GATED ION CHANNELS
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Patent #:
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Issue Dt:
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11/02/2010
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Application #:
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10887719
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Filing Dt:
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07/09/2004
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Publication #:
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Pub Dt:
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04/28/2005
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Title:
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POTENTIATORS OF ANTIBACTERIAL ACTIVITY
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Patent #:
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Issue Dt:
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08/14/2007
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Application #:
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10891912
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Filing Dt:
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07/13/2004
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Publication #:
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Pub Dt:
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01/06/2005
| | | | |
Title:
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THIAZOLE COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASE
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|
|
Patent #:
|
|
Issue Dt:
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09/19/2006
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Application #:
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10893748
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Filing Dt:
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07/16/2004
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Publication #:
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|
Pub Dt:
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05/19/2005
| | | | |
Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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|
|
Patent #:
|
|
Issue Dt:
|
05/22/2007
|
Application #:
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10900996
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Filing Dt:
|
07/28/2004
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Publication #:
|
|
Pub Dt:
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02/02/2006
| | | | |
Title:
|
SENSOR FOR LEVELS OF CONDUCTIVE LIQUIDS
|
|
|
Patent #:
|
|
Issue Dt:
|
08/04/2009
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Application #:
|
10901928
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Filing Dt:
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07/29/2004
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Publication #:
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|
Pub Dt:
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02/17/2005
| | | | |
Title:
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GYRASE INHIBITORS AND USES THEREOF
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|
|
Patent #:
|
|
Issue Dt:
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06/28/2011
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Application #:
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10912912
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Filing Dt:
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08/05/2004
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Publication #:
|
|
Pub Dt:
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08/25/2005
| | | | |
Title:
|
COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED ION CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
06/05/2007
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Application #:
|
10914051
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Filing Dt:
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08/06/2004
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Publication #:
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Pub Dt:
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11/24/2005
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Title:
|
AMINOTRIAZOLE COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
06/19/2012
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Application #:
|
10914988
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Filing Dt:
|
08/09/2004
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Publication #:
|
|
Pub Dt:
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06/23/2005
| | | | |
Title:
|
COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
|
|
|
Patent #:
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|
Issue Dt:
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01/02/2007
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Application #:
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10922575
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Filing Dt:
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08/20/2004
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Publication #:
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Pub Dt:
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07/07/2005
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Title:
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AMINOFURAZAN COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
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|
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Patent #:
|
|
Issue Dt:
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05/11/2010
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Application #:
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10935008
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Filing Dt:
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09/02/2004
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Publication #:
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Pub Dt:
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09/28/2006
| | | | |
Title:
|
QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS
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|
|
Patent #:
|
|
Issue Dt:
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07/05/2011
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Application #:
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10936448
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Filing Dt:
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09/07/2004
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Publication #:
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|
Pub Dt:
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08/11/2005
| | | | |
Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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|
|
Patent #:
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|
Issue Dt:
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05/27/2008
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Application #:
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10936450
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Filing Dt:
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09/07/2004
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Publication #:
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|
Pub Dt:
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06/23/2005
| | | | |
Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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|
|
Patent #:
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|
Issue Dt:
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11/04/2008
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Application #:
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10936470
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Filing Dt:
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09/07/2004
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Publication #:
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Pub Dt:
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06/23/2005
| | | | |
Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
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Patent #:
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|
Issue Dt:
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02/24/2009
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Application #:
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10941387
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Filing Dt:
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09/15/2004
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Publication #:
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Pub Dt:
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08/18/2005
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Title:
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CRYSTAL STRUCTURE OF FMS-LIKE TYROSINE KINASE
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Patent #:
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Issue Dt:
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01/30/2007
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Application #:
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10949027
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Filing Dt:
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09/24/2004
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Publication #:
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Pub Dt:
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07/07/2005
| | | | |
Title:
|
IMIDAZOLE COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
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01/26/2010
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Application #:
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10949714
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Filing Dt:
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09/23/2004
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Publication #:
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Pub Dt:
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05/12/2005
| | | | |
Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
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Patent #:
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|
Issue Dt:
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07/21/2009
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Application #:
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10951242
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Filing Dt:
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09/27/2004
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Publication #:
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Pub Dt:
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06/23/2005
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Title:
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PHENYL-PIPERAZINE DERIVATIVES AS MODULATORS OF MUSCARINIC RECEPTORS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/13/2008
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Application #:
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10951382
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Filing Dt:
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09/28/2004
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Publication #:
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Pub Dt:
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04/07/2005
| | | | |
Title:
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COMPOSITIONS COMPRISING IMPDH INHIBITORS AND USES THEREOF FOR TREATING HCV INFECTION
|
|
|
Patent #:
|
|
Issue Dt:
|
12/19/2006
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Application #:
|
10951409
|
Filing Dt:
|
09/27/2004
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Publication #:
|
|
Pub Dt:
|
03/03/2005
| | | | |
Title:
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INHIBITORS OF P38
|
|
|
Patent #:
|
|
Issue Dt:
|
09/22/2009
|
Application #:
|
10958223
|
Filing Dt:
|
10/04/2004
|
Publication #:
|
|
Pub Dt:
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07/07/2005
| | | | |
Title:
|
SULPHONAMIDE DERIVATIVES AS PRODRUGS OF ASPARTYL PROTEASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
10/06/2009
|
Application #:
|
10961485
|
Filing Dt:
|
10/08/2004
|
Publication #:
|
|
Pub Dt:
|
07/07/2005
| | | | |
Title:
|
MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
|
|
|
Patent #:
|
|
Issue Dt:
|
04/24/2007
|
Application #:
|
10964214
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Filing Dt:
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10/12/2004
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Publication #:
|
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Pub Dt:
|
06/23/2005
| | | | |
Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASES
|
|
|
Patent #:
|
|
Issue Dt:
|
04/20/2010
|
Application #:
|
10965695
|
Filing Dt:
|
10/14/2004
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Publication #:
|
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Pub Dt:
|
07/07/2005
| | | | |
Title:
|
COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
11/17/2009
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Application #:
|
10971573
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Filing Dt:
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10/21/2004
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Publication #:
|
|
Pub Dt:
|
06/08/2006
| | | | |
Title:
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GYRASE INHIBITORS AND USES THEREOF
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|
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Patent #:
|
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Issue Dt:
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02/24/2009
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Application #:
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10974558
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Filing Dt:
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10/27/2004
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Publication #:
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Pub Dt:
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06/23/2005
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Title:
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HCV NS3-NS4A PROTEASE RESISTANCE MUTANTS
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Patent #:
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Issue Dt:
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05/29/2012
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Application #:
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10975196
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Filing Dt:
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10/27/2004
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Publication #:
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Pub Dt:
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01/05/2006
| | | | |
Title:
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DRUG DISCOVERY METHOD
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|
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Patent #:
|
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Issue Dt:
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12/18/2007
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Application #:
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10977609
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Filing Dt:
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10/28/2004
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Publication #:
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Pub Dt:
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09/22/2005
| | | | |
Title:
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BENZIMIDAZOLES USEFUL AS MODULATORS OF ION CHANNELS
|
|
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Patent #:
|
|
Issue Dt:
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07/31/2007
|
Application #:
|
10978301
|
Filing Dt:
|
10/28/2004
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Publication #:
|
|
Pub Dt:
|
06/30/2005
| | | | |
Title:
|
PROCESSES FOR PREPARING PYRROLES
|
|
|
Patent #:
|
|
Issue Dt:
|
09/01/2009
|
Application #:
|
10986569
|
Filing Dt:
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11/11/2004
|
Publication #:
|
|
Pub Dt:
|
11/17/2005
| | | | |
Title:
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GYRASE INHIBITORS AND USES THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
08/05/2008
|
Application #:
|
10989218
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Filing Dt:
|
11/15/2004
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Publication #:
|
|
Pub Dt:
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06/16/2005
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Title:
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THIAZOLES AND OXAZOLES USEFUL AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
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10/07/2008
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Application #:
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10997810
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Filing Dt:
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11/24/2004
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Publication #:
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Pub Dt:
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07/07/2005
| | | | |
Title:
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INHIBITORS OF IMPDH ENZYME
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Patent #:
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Issue Dt:
|
07/17/2007
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Application #:
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11001760
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Filing Dt:
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12/02/2004
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Publication #:
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Pub Dt:
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11/03/2005
| | | | |
Title:
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HETEROCYCLIC PROTEIN KINASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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09/22/2009
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Application #:
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11004657
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Filing Dt:
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12/03/2004
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Publication #:
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Pub Dt:
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10/20/2005
| | | | |
Title:
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QUINOXALINES USEFUL AS INHIBITORS OF PROTEIN KINASES
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Patent #:
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Issue Dt:
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11/04/2008
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Application #:
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11005944
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Filing Dt:
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12/07/2004
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Publication #:
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Pub Dt:
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08/04/2005
| | | | |
Title:
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MODULATORS OF MUSCARINIC RECEPTORS
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Patent #:
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Issue Dt:
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10/09/2007
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Application #:
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11030004
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Filing Dt:
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01/05/2005
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Publication #:
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Pub Dt:
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09/29/2005
| | | | |
Title:
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PYRAZOLE-DERIVED KINASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
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03/03/2009
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Application #:
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11033774
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Filing Dt:
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01/12/2005
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Publication #:
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Pub Dt:
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01/26/2006
| | | | |
Title:
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DUAL EXPRESSION VECTOR SYSTEM AND SCREENING METHODS
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Patent #:
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Issue Dt:
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12/21/2010
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Application #:
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11046664
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Filing Dt:
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01/26/2005
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Publication #:
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Pub Dt:
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09/22/2005
| | | | |
Title:
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FUSED CYCLIC SYSTEMS USEFUL AS INHIBITORS OF TEC FAMILY PROTEIN KINASES
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Patent #:
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Issue Dt:
|
06/24/2014
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Application #:
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11047366
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Filing Dt:
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01/31/2005
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Publication #:
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Pub Dt:
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03/09/2006
| | | | |
Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
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Patent #:
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Issue Dt:
|
03/23/2010
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Application #:
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11051977
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Filing Dt:
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02/04/2005
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Publication #:
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Pub Dt:
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09/29/2005
| | | | |
Title:
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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
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Patent #:
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Issue Dt:
|
11/10/2009
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Application #:
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11060719
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Filing Dt:
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02/17/2005
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Publication #:
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Pub Dt:
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02/02/2006
| | | | |
Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
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Patent #:
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Issue Dt:
|
01/26/2010
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Application #:
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11069895
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Filing Dt:
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02/28/2005
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Publication #:
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Pub Dt:
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10/20/2005
| | | | |
Title:
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CASPASE INHIBITORS AND USES THEREOF
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Patent #:
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Issue Dt:
|
03/18/2008
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Application #:
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11077188
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Filing Dt:
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03/10/2005
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Publication #:
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Pub Dt:
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10/20/2005
| | | | |
Title:
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HETEROCYCLIC INHIBITORS OF ERK2 AND USES THEREOF
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|
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Patent #:
|
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Issue Dt:
|
06/03/2008
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Application #:
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11078147
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Filing Dt:
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03/11/2005
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Publication #:
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Pub Dt:
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01/26/2006
| | | | |
Title:
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PROCESSES AND INTERMEDIATES
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|
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Patent #:
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Issue Dt:
|
12/09/2008
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Application #:
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11089701
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Filing Dt:
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03/25/2005
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Publication #:
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Pub Dt:
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01/26/2006
| | | | |
Title:
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PYRIDINE INHIBITORS OF ERK2 AND USES THEREOF
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|
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Patent #:
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Issue Dt:
|
03/24/2009
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Application #:
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11093821
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Filing Dt:
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03/30/2005
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Publication #:
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Pub Dt:
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02/22/2007
| | | | |
Title:
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AZAINDOLES USEFUL AS INHIBITORS OF JAK AND OTHER PROTEIN KINASES
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|
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Patent #:
|
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Issue Dt:
|
04/07/2009
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Application #:
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11098751
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Filing Dt:
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04/04/2005
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Publication #:
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Pub Dt:
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01/05/2006
| | | | |
Title:
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AZAINDOLES USEFUL AS INHIBITORS OF ROCK AND OTHER PROTEIN KINASES
|
|
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Patent #:
|
|
Issue Dt:
|
07/07/2009
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Application #:
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11114979
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Filing Dt:
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04/26/2005
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Publication #:
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Pub Dt:
|
02/09/2006
| | | | |
Title:
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CRYSTAL STRUCTURE OF HUMAN JAK3 KINASE DOMAIN COMPLEX AND BINDING POCKETS THEREOF
|
|
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Patent #:
|
|
Issue Dt:
|
05/12/2009
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Application #:
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11115661
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Filing Dt:
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04/27/2005
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Publication #:
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Pub Dt:
|
01/26/2006
| | | | |
Title:
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COMPOSITIONS USEFUL AS INHIBITORS OF ROCK AND OTHER PROTEIN KINASES
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|
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Patent #:
|
|
Issue Dt:
|
04/08/2008
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Application #:
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11128870
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Filing Dt:
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05/13/2005
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Publication #:
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Pub Dt:
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05/18/2006
| | | | |
Title:
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PYRROLE INHIBITORS OF ERK PROTEIN KINASE, SYNTHESIS THEREOF AND INTERMEDIATES THERETO
|
|
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Patent #:
|
|
Issue Dt:
|
04/15/2008
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Application #:
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11129114
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Filing Dt:
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05/13/2005
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Publication #:
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Pub Dt:
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03/16/2006
| | | | |
Title:
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PRODRUGS OF AN ERK PROTEIN KINASE INHIBITOR
|
|
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Patent #:
|
NONE
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Issue Dt:
|
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Application #:
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11130659
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Filing Dt:
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05/16/2005
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Publication #:
|
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Pub Dt:
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06/15/2006
| | | | |
Title:
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Treating seizures using ice inhibitors
|
|
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Patent #:
|
|
Issue Dt:
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05/12/2009
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Application #:
|
11140649
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Filing Dt:
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05/27/2005
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Publication #:
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Pub Dt:
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12/01/2005
| | | | |
Title:
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TREATMENT OF DISEASES USING ICE INHIBITORS
|
|
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Patent #:
|
|
Issue Dt:
|
10/26/2010
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Application #:
|
11140808
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Filing Dt:
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05/31/2005
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Publication #:
|
|
Pub Dt:
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01/26/2006
| | | | |
Title:
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MODULATORS OF MUSCARINIC RECEPTORS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/18/2008
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Application #:
|
11145356
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Filing Dt:
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06/03/2005
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Publication #:
|
|
Pub Dt:
|
10/06/2005
| | | | |
Title:
|
INHIBITORS OF GSK-3 AND USES THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
08/04/2009
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Application #:
|
11165254
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Filing Dt:
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06/22/2005
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Publication #:
|
|
Pub Dt:
|
04/06/2006
| | | | |
Title:
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HETEROCYCLIC DERIVATIVES FOR MODULATION OF CALCIUM CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/24/2009
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Application #:
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11165818
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Filing Dt:
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06/24/2005
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Publication #:
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Pub Dt:
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04/06/2006
| | | | |
Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
|
|
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Patent #:
|
|
Issue Dt:
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02/12/2008
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Application #:
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11192657
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Filing Dt:
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07/29/2005
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Publication #:
|
|
Pub Dt:
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12/22/2005
| | | | |
Title:
|
INHIBITORS OF IMPDH ENZYME
|
|
|
Patent #:
|
|
Issue Dt:
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07/12/2011
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Application #:
|
11202278
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Filing Dt:
|
08/11/2005
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Publication #:
|
|
Pub Dt:
|
07/24/2008
| | | | |
Title:
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MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/01/2011
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Application #:
|
11208386
|
Filing Dt:
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08/19/2005
|
Publication #:
|
|
Pub Dt:
|
04/13/2006
| | | | |
Title:
|
SPIROINDOLINE MODULATORS OF MUSCARINIC RECEPTORS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/02/2008
|
Application #:
|
11212045
|
Filing Dt:
|
08/25/2005
|
Publication #:
|
|
Pub Dt:
|
08/03/2006
| | | | |
Title:
|
SULFONAMIDE INHIBITORS OF ASPARTYL PROTEASE
|
|
|
Patent #:
|
|
Issue Dt:
|
10/09/2012
|
Application #:
|
11216376
|
Filing Dt:
|
08/31/2005
|
Publication #:
|
|
Pub Dt:
|
08/03/2006
| | | | |
Title:
|
QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/18/2010
|
Application #:
|
11216899
|
Filing Dt:
|
08/31/2005
|
Publication #:
|
|
Pub Dt:
|
07/13/2006
| | | | |
Title:
|
QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/12/2008
|
Application #:
|
11230221
|
Filing Dt:
|
09/19/2005
|
Publication #:
|
|
Pub Dt:
|
03/23/2006
| | | | |
Title:
|
DIAMINOTRIAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/23/2010
|
Application #:
|
11242666
|
Filing Dt:
|
10/04/2005
|
Publication #:
|
|
Pub Dt:
|
02/08/2007
| | | | |
Title:
|
CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE PROTEIN COMPLEXES AND BINDING POCKETS THEREOF, AND USES THEREOF IN DRUG DESIGN
|
|
|
Patent #:
|
|
Issue Dt:
|
01/12/2010
|
Application #:
|
11255569
|
Filing Dt:
|
10/21/2005
|
Publication #:
|
|
Pub Dt:
|
11/22/2007
| | | | |
Title:
|
TRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
04/30/2013
|
Application #:
|
11264746
|
Filing Dt:
|
10/31/2005
|
Publication #:
|
|
Pub Dt:
|
05/18/2006
| | | | |
Title:
|
Dose forms
|
|
|
Patent #:
|
|
Issue Dt:
|
08/03/2010
|
Application #:
|
11266142
|
Filing Dt:
|
11/03/2005
|
Publication #:
|
|
Pub Dt:
|
07/20/2006
| | | | |
Title:
|
ION CHANNEL MODULATORS AND METHODS OF USE
|
|
|
Patent #:
|
|
Issue Dt:
|
05/05/2009
|
Application #:
|
11266935
|
Filing Dt:
|
11/04/2005
|
Publication #:
|
|
Pub Dt:
|
06/22/2006
| | | | |
Title:
|
PYRAZOLO[1,5-A]PYRIMIDINES USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|
|
Patent #:
|
|
Issue Dt:
|
02/17/2015
|
Application #:
|
11280978
|
Filing Dt:
|
11/16/2005
|
Publication #:
|
|
Pub Dt:
|
05/17/2007
| | | | |
Title:
|
WIRELESS DETECTION OF MOTION
|
|
|
Patent #:
|
|
Issue Dt:
|
01/29/2013
|
Application #:
|
11284366
|
Filing Dt:
|
11/21/2005
|
Publication #:
|
|
Pub Dt:
|
07/20/2006
| | | | |
Title:
|
CASPASE INHIBITORS AND USES THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
09/14/2010
|
Application #:
|
11285497
|
Filing Dt:
|
11/22/2005
|
Publication #:
|
|
Pub Dt:
|
11/16/2006
| | | | |
Title:
|
PYRROLOPYRAZINES AND PYRAZOLOPYRAZINES USEFUL AS INHIBITORS OF PROTEIN KINASES
|
|