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05/24/1988
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06858573
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04/24/1986
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Title:
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ANTI-INFLAMMATORY PRODUCTS DERIVED FROM METHYLENE-DIPHOSPHONIC ACID, AND PROCESS FOR THEIR PREPARATION
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07/31/1990
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07036263
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Filing Dt:
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04/09/1987
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Title:
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MICROBIOLOGICAL PROCESS FOR THE PREPARATION OF A PROTEIN BY CULTURING A MUTANT BACTERIAL STRAIN
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10/24/1989
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Application #:
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07165080
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Filing Dt:
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03/07/1988
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Title:
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ANTI-INFLAMMATORY PRODUCTS DERIVED FROM METHYLENE-DIPHOSPHONIC ACID, AND PROCESS FOR THEIR PREPARATION
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05/22/1990
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07230860
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Filing Dt:
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08/11/1988
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Title:
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PROCESS FOR THE 0-ALKYLATION OF N-(HYDROXY)ARALKYLPHENYLETHANOLAMINES
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12/25/1990
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07333966
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Filing Dt:
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04/06/1989
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Title:
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PHARMACEUTICAL COMPOSITION FOR ORAL ADMINISTRATION, BASED ON A DIPHOSPHONIC ACID DERIVATIVE
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Patent #:
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06/25/1991
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07437674
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11/17/1989
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Title:
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METHOD OF TREATMENT OF ANXIETY AND ANXIO-DEPRESSIVE DISORDERS
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08/20/1991
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07488137
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03/05/1990
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Title:
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PROCESS FOR THE O-ALKYLATION OF N-(HYDROXY)ARALKYLPHENYLETHANOLAMINES
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08/17/1993
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07536741
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Filing Dt:
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06/12/1990
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Title:
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PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF OCULAR DISORDERS
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04/28/1992
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07563196
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Filing Dt:
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08/06/1990
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Title:
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TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES FOR THE TREATMENT AND/OR PROPHYLAXIS OF INTESTINAL MOTILITY DISORDERS
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Patent #:
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07/20/1993
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07703835
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05/21/1991
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Title:
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IMPROVED METHOD FOR EVALUATING NEURONAL ACTIVITY OF A DRUG
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01/25/1994
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07705704
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05/23/1991
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Title:
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N-SUBSTITUTED TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES, PROCESS FOR THR PREPARATION THEREOF, INTERMEDIATES IN SAID PROCESS AN PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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10/11/1994
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07707229
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05/24/1991
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Title:
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BENZENE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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07/27/1993
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07714832
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06/13/1991
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Title:
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HEXAHYDROAZEPINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAIN- ING THEM
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08/17/1993
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07755454
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09/05/1991
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Title:
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ARYLALKYLAMINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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12/14/1993
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07789044
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11/07/1991
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Title:
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USE OF A 1-(2-NAPHTHYLETHYL)-4-(3-TRIFLUOROMETHYLPHENYL)-1,2,3,6- TETRAHYDROPYRIDINE FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF CEREBRAL AND NEURONAL DISEASES
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Patent #:
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Issue Dt:
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12/14/1993
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07804580
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12/04/1991
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Title:
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METHOD OF TREATMENT OR PROPHYLAXIS OF DEPRESSION AND STRESS
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Patent #:
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Issue Dt:
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02/08/1994
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07825080
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Filing Dt:
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01/24/1992
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Title:
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SIGNAL PEPTIDE, DNA SEQUENCES CODING FOR THE LATTER, EXPRESSION VECTORS CARRYING ONE OF THESE SEQUENCES, GRAM-NEGATIVE BACTERIA TRANSFORMED BY THESE VECTORS, AND PROCESS FOR THE PERIPLASMIC PRODUCTION OF A POLYPEPTIDE
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Patent #:
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Issue Dt:
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03/08/1994
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07830857
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02/04/1992
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Title:
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USE OF 4-(3-TRIFLUOROMETHYLPHENYL)-1,2,3,6-TETRAHYDROPYRIDINE DERIVATIVES AS FREE RADICAL SCAVENGERS
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Patent #:
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05/02/1995
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07877734
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05/04/1992
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Title:
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N-ALKYLENEPIPERIDINO COMPOUNDS, THEIR ENANTIOMERS AND PHARMACEUTICAL COMPOSITIONS
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08/23/1994
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07878710
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05/04/1992
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Title:
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POLYCYCLIC AMINE COMPOUNDS AND THEIR ENANTIOMERS, THEIR METHOD OF PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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01/18/1994
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07931495
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08/21/1992
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Title:
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DNA SEQUENCE PARTICIPATING IN THE REGULATION OF THE EXPRESSION OF A DNA SEQUENCE CODING FOR A PRECURSOR OF A POLYPEPTIDE, EXPRESSION VECTORS AND PROCESS FOR THE PERIPLASMIC PRODUCTION OF THE POLYPEPTIDE
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Patent #:
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Issue Dt:
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11/30/1993
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08038082
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Filing Dt:
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03/29/1993
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Title:
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TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES FOR THE TREATMENT AND/OR PROPHYLAXIS OF INTESTINAL MOTILITY DISORDERS
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Patent #:
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03/22/1994
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08045722
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04/14/1993
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Title:
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HEXAHYDROAZEPINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION
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Patent #:
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Issue Dt:
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04/18/1995
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08086410
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Filing Dt:
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07/06/1993
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Title:
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ARTIFICIAL PROMOTER FOR THE EXPRESSION OF PROTEINS IN YEAST
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Patent #:
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Issue Dt:
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09/27/1994
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08105677
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08/13/1993
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Title:
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ARYLALKYLAMINES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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09/13/1994
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Application #:
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08114190
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09/01/1993
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Title:
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(RR) AND (RS STEREOISOMERS OF N-(1-ETHOXYCARBONYLMETHOXY-1,2,3,-TETRAHYDRONAPHTH-2-YL)-2-(3-CHLOROPH ENYL)-2-HYDROXYETHANAMINE AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS
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Patent #:
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Issue Dt:
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05/30/1995
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08119830
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09/13/1993
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Title:
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3-AMIDOPYRAZOLE DERIVATIVES, PROCESS FOR PREPARING THESE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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10/31/1995
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08141066
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10/26/1993
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Title:
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N-SUBSTITUTED TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES, PROCESS FOR THE PREPARATION THEREOF, INTERMEDIATES IN SAID PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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11/21/1995
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Application #:
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08142069
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10/20/1993
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Title:
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USE OF A 1-(2-NAPHTHYLETHYL)-4-(3-TRIFLUOROMETHYLPHENYL)-1,2,3,6- TETRAHYDROPYRIDINE FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF CEREBRAL AND NEURONAL DISEASES
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Patent #:
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Issue Dt:
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01/03/1995
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08214307
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03/17/1994
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Title:
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USE OF TETRAHYDROPYRIDINE DERIVATIVES FOR THE PREPARATION OF CARDIOPROTECTIVE DRUGS
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Issue Dt:
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01/30/1996
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08222240
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04/04/1994
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Title:
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METHOD OF PROMOTING BONE REPAIR USING TILUDRONIC DISODIUM SALT
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Issue Dt:
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12/10/1996
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08239417
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05/06/1994
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Title:
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1-AZONIABICYCLO[2.2.2] OCTANES AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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06/23/1998
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08261269
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06/15/1994
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Title:
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POLYCYCLIC AMINE COMPOUNDS AND THEIR ENANTIOMERS, THEIR METHOD OF PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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09/12/1995
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Application #:
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08264064
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Filing Dt:
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06/22/1994
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Title:
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BENZENE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Issue Dt:
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04/30/1996
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08294035
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08/24/1994
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Title:
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PROCESS FOR THE PREPARATION OF AN OPTICALLY PURE AMINOALCOHOL
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Patent #:
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Issue Dt:
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10/07/1997
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08345341
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11/21/1994
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Title:
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QUATERNARY AMMONIUM SALTS OF AROMATIC AMINE COMPOUNDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Issue Dt:
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04/29/1997
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08348881
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11/29/1994
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Title:
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NOVEL PYRAZOLE DERIVATIVES, METHOD OF PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Issue Dt:
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10/31/1995
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Application #:
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08357880
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12/16/1994
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Title:
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NOVEL PYRAZOLE-3-CARBOXAMIDE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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07/29/1997
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08371121
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01/11/1995
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Title:
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PROTEIN HAVING INTERLEUKIN 13 ACTIVITY RECOMBINANT DNA CODING FOR THIS PROTEIN, TRANSFORMED CELLS AND MICROORGANISMS
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Issue Dt:
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06/03/1997
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08393829
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02/24/1995
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Title:
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3-AMIDOPYRAZOLE DERIVATIVES, PROCESS FOR PREPARING THESE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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04/01/1997
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08394756
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02/27/1995
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Title:
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3-AMIDOPYRAZOLE DERIVATIVES, PROCESS FOR PREPARING THESE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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03/04/1997
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08394757
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02/27/1995
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Title:
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3-AMIDOPYRAZOLE DERIVATIVES, PROCESS FOR PREPARING THESE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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02/25/1997
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Application #:
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08410292
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03/24/1995
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Title:
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PROCESS FOR PREPARING N-ALKYLENE PIPERIDINO COMPOUNDS AND THEIR ENANTIOMERS
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Issue Dt:
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02/04/1997
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08455207
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Filing Dt:
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05/31/1995
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Title:
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N-SUBSTITUTED TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES PROCESS FOR THE PREPARATION THEREOF INTERMEDIATES IN SAID PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Issue Dt:
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01/21/1997
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Application #:
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08455210
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Filing Dt:
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05/31/1995
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Title:
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N-SUBSTITUTED TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES,PROCESS FOR THE PREPARATION THEREOF,INTERMEDIATES IN SAID PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Issue Dt:
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04/29/1997
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08463270
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06/05/1995
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Title:
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POLYCYCLIC AMINE COMPOUNDS AND THEIR ENANTIOMERS, THEIR METHOD OF PREPARATION AND PHARMACEUTICAL COMPOSITIONS ON WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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09/10/1996
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08470249
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06/06/1995
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Title:
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1-AZONIABICYCLO[2.2.1] HEPTANES AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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06/30/1998
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08482546
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06/07/1995
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Title:
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QUATERNARY AMMONIUM SALTS OF AROMATIC AMINE COMPOUNDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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09/24/1996
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Application #:
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08482748
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Filing Dt:
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06/07/1995
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Title:
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N-SUBSTITUTED TRIFLUOROMETHYLPHENYLTETRAHYDROPYRIDINES PROCESS FOR THE PREPARATION THEREOF, INTERMEDIATES IN SAID PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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01/14/1997
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08500924
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Filing Dt:
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07/31/1995
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Title:
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1,3-DIHYDROINDOL-2-ONE DERIVATIVES SUBSTITUTED IN THE 3-POSITION BY A NITROGEN-CONTAINING GROUP, THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Issue Dt:
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05/13/1997
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08544027
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Filing Dt:
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10/17/1995
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Title:
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PROCESS FOR THE PREPARATION OF A TETRAZOLE DERIVATIVE IN TWO CRYSTALLINE FORMS AND NOVEL THE CRYSTALLINE FORMS THEREOF
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Issue Dt:
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06/24/1997
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Application #:
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08593938
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Filing Dt:
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01/30/1996
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Title:
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SUBSTITUTED HETEROCYCLIC COMPOUNDS,AND PHARMACEUITICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Issue Dt:
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07/14/1998
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08598001
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02/07/1996
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Title:
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PROCESS FOR THE PREPARATION OF AN OPTICALLY PURE AMINOALCOHOL
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04/21/1998
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08607976
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02/29/1996
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Title:
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COMPOUNDS WHICH ARE SELECTIVE ANTAGONISTS OF THE HUMAN NK3 RECEPTOR AND THEIR USE AS MEDICINAL PRODUCTS AND DIAGNOSTIC TOOLS
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Issue Dt:
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03/03/1998
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08630761
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04/10/1996
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Title:
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SUBSTITUTED 1-PHENYL-3-PYRAZOLECARBOXAMIDES ACTIVE ON NEUROTENSIN RECEPTORS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Issue Dt:
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06/30/1998
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08640080
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04/30/1996
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Title:
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INDOL-2-ONE DERIVATIVES
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Issue Dt:
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10/21/1997
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08685489
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07/24/1996
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Title:
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1-AZONIABICYCLO[2.2.1]HEPTANES, METHOD OF PREPARING THEM AND PHAR- MACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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07/14/1998
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08703729
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08/27/1996
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Title:
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SUBSTITUTED HETEROCYCLIC COMPOUNDS METHOD OF PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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11/03/1998
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08703952
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08/28/1996
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Title:
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PIPERIDINE DERIVATIVES, PROCESS FOR OBTAINING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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01/27/1998
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08734029
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10/18/1996
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Title:
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QUATENARY BASIC AMIDES, METHOD OF PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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04/28/1998
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Application #:
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08775150
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12/31/1996
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Title:
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3-AMIDOPYRAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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04/28/1998
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08778105
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01/02/1997
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Title:
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3-AMIDOPYRAZOLE DERIVATIVES, PROCESS FOR PREPARING THESE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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01/12/1999
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Application #:
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08787910
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01/23/1997
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Title:
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NOVEL HETEROCYCLIC COMPOUNDS METHOD OF PREPARING THEM AND PHARMEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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02/09/1999
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08820716
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03/18/1997
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Title:
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SUBSTITUTED HETEROCYCLIC COMPOUNDS
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Issue Dt:
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05/04/1999
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08913360
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09/17/1997
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Title:
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USE OF FUMAGILLOL AND DERIVATIVES THEREOF FOR PREPARING MEDICAMENTS AGAINST INTESTINAL INFECTIONS
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08/17/1999
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08916952
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08/25/1997
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Title:
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PIPERIDINE DERIVATIVES PROCESS FOR OBTAINING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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11/09/1999
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Application #:
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08973712
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Filing Dt:
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02/24/1998
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Title:
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4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY
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Patent #:
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Issue Dt:
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10/12/1999
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Application #:
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08976309
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Filing Dt:
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11/21/1997
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Title:
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SUBSTITUTED 1-PHENYL1-3-PYRAZOLECARBOXAMIDES ACTIVE ON NEUROTENSIN RECEPTORS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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07/20/1999
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Application #:
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08976691
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Filing Dt:
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11/24/1997
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Title:
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SUBSTITUTED 1-PHENYL-3-PYRAZOLECARBOXAMIDES ACTIVE ON NEUROTENSIN RECEPTORS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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08/10/1999
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Application #:
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08976714
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Filing Dt:
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11/24/1997
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Title:
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HYDRAZINE DERIVATIVE COMPOUNDS AS INTERMEDIATES FOR PREPARING SUBSTITITED 1-PHENYL-3-PYRAZOLECARBOXAMIDES ACTIVE ON NEUROTENSIN RECEPTORS
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Patent #:
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Issue Dt:
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08/17/1999
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Application #:
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08977496
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Filing Dt:
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11/24/1997
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Title:
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SUBSTITUTED 1-PHENYL-3-PYRAZOLECARBOXAMIDES ACTIVE ON NEUROTENSIN RECEPTORS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITONS CONTAINING THEM
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Patent #:
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Issue Dt:
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01/11/2000
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Application #:
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08995902
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Filing Dt:
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12/22/1997
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Title:
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CB2 RECEPTOR AGONIST COMPOUNDS
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Patent #:
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Issue Dt:
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01/04/2000
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Application #:
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09004454
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Filing Dt:
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01/08/1998
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Title:
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SUBSTITUTED HETEROCYCLIC COMPOUNDS, METHOD OF PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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10/12/1999
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Application #:
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09035823
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Filing Dt:
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03/06/1998
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Title:
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NEW PIPERIDINE DERIVATIVES, PROCESS FOR OBTAINING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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Patent #:
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Issue Dt:
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04/17/2001
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Application #:
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09169115
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Filing Dt:
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10/08/1998
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Title:
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USE OF AN ANGIOTENSIN II ANTAGONIST AND A BENZOFURAN DERIVATIVE IN THE TREATMENT OF CARDIOVASCULAR COMPLAINTS
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Patent #:
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Issue Dt:
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11/02/1999
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Application #:
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09175332
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Filing Dt:
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10/20/1998
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Title:
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SUBSTITUTED HETEROCYLIC COMPOUNDS, METHOD OF PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS IN WHICH THEY ARE PRESENT
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Patent #:
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Issue Dt:
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09/26/2000
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Application #:
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09306825
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Filing Dt:
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05/07/1999
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Title:
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COMPOUNDS WHICH ARE SPECIFIC ANTAGONISTS OF THE HUMAN NK3 RECEPTOR AND THEIR USE AS MEDICINAL PRODUCTS AND DIAGNOSTIC TOOLS
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Patent #:
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Issue Dt:
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Application #:
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UNAVAILABLE
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Filing Dt:
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Title:
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