Total properties:
65
|
|
Patent #:
|
|
Issue Dt:
|
04/22/2008
|
Application #:
|
10382203
|
Filing Dt:
|
03/05/2003
|
Publication #:
|
|
Pub Dt:
|
04/29/2004
| | | | |
Title:
|
AZOLE DERIVATIVES AND FUSED BICYCLIC AZOLE DERIVATIVES AS THERAPEUTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
06/10/2008
|
Application #:
|
10679887
|
Filing Dt:
|
10/06/2003
|
Publication #:
|
|
Pub Dt:
|
06/24/2004
| | | | |
Title:
|
ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/08/2011
|
Application #:
|
11197038
|
Filing Dt:
|
08/03/2005
|
Publication #:
|
|
Pub Dt:
|
02/09/2006
| | | | |
Title:
|
RAGE FUSION PROTEINS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/11/2010
|
Application #:
|
11511163
|
Filing Dt:
|
08/28/2006
|
Publication #:
|
|
Pub Dt:
|
01/25/2007
| | | | |
Title:
|
AZOLE DERIVATIVES AND FUSED BICYCLIC AZOLE DERIVATIVES AS THERAPEUTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/19/2011
|
Application #:
|
11629437
|
Filing Dt:
|
04/12/2007
|
Publication #:
|
|
Pub Dt:
|
03/27/2008
| | | | |
Title:
|
RAGE FUSION PROTEINS
|
|
|
Patent #:
|
|
Issue Dt:
|
05/25/2010
|
Application #:
|
11699780
|
Filing Dt:
|
01/30/2007
|
Publication #:
|
|
Pub Dt:
|
08/16/2007
| | | | |
Title:
|
SUBSTITUTED IMIDAZOLE DERIVATIVES, COMPOSITIONS, AND METHODS OF USE AS PTPASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/19/2011
|
Application #:
|
11789637
|
Filing Dt:
|
04/25/2007
|
Publication #:
|
|
Pub Dt:
|
02/21/2008
| | | | |
Title:
|
RAGE FUSION PROTEINS, FORMULATIONS, AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
06/15/2010
|
Application #:
|
11800085
|
Filing Dt:
|
05/03/2007
|
Publication #:
|
|
Pub Dt:
|
09/13/2007
| | | | |
Title:
|
AZOLE DERIVATIVES AND FUSED BICYCLIC AZOLE DERIVATIVES AS THERAPEUTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
11/22/2011
|
Application #:
|
11981997
|
Filing Dt:
|
10/31/2007
|
Publication #:
|
|
Pub Dt:
|
05/22/2008
| | | | |
Title:
|
ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/01/2011
|
Application #:
|
11982248
|
Filing Dt:
|
10/31/2007
|
Publication #:
|
|
Pub Dt:
|
05/22/2008
| | | | |
Title:
|
ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/01/2009
|
Application #:
|
11994728
|
Filing Dt:
|
07/09/2008
|
Publication #:
|
|
Pub Dt:
|
05/07/2009
| | | | |
Title:
|
DICYCLOALKYL UREA GLUCOKINASE ACTIVATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/08/2011
|
Application #:
|
12046872
|
Filing Dt:
|
03/12/2008
|
Publication #:
|
|
Pub Dt:
|
10/09/2008
| | | | |
Title:
|
CRYSTALLINE FORMS OF [3-(4- {2-BUTYL- 1 -[4-(4-CHLORO-PHENOXY)-PHENYL]-1H-IMIDAZOL-4-YL} -PHENOXY)-PROPYL]-DIETHYL-AMINE
|
|
|
Patent #:
|
|
Issue Dt:
|
02/19/2013
|
Application #:
|
12302132
|
Filing Dt:
|
11/24/2008
|
Publication #:
|
|
Pub Dt:
|
07/09/2009
| | | | |
Title:
|
3-(L,3-BENZODIOXOL-5-YL)-6-(4-CYCLOPROPYLPIPERAZIN-L-YL)-PYRIDAZINE, ITS SALTS AND SOLVATES AND ITS USE AS HISTAMINE H3 RECEPTOR ANTAGONIST
|
|
|
Patent #:
|
|
Issue Dt:
|
06/01/2010
|
Application #:
|
12399504
|
Filing Dt:
|
03/06/2009
|
Publication #:
|
|
Pub Dt:
|
12/10/2009
| | | | |
Title:
|
OXADIAZOANTHRACENE COMPOUNDS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
11/27/2012
|
Application #:
|
12522469
|
Filing Dt:
|
09/22/2009
|
Publication #:
|
|
Pub Dt:
|
02/18/2010
| | | | |
Title:
|
UREA GLUCOKINASE ACTIVATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
02/26/2013
|
Application #:
|
12528229
|
Filing Dt:
|
11/01/2010
|
Publication #:
|
|
Pub Dt:
|
02/17/2011
| | | | |
Title:
|
N-ADAMANTYL BENZAMIDES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE
|
|
|
Patent #:
|
|
Issue Dt:
|
06/21/2011
|
Application #:
|
12532861
|
Filing Dt:
|
09/24/2009
|
Publication #:
|
|
Pub Dt:
|
07/29/2010
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/26/2013
|
Application #:
|
12685178
|
Filing Dt:
|
01/11/2010
|
Publication #:
|
|
Pub Dt:
|
05/06/2010
| | | | |
Title:
|
SUBSTITUTED IMIDAZOLE DERIVATIVES, COMPOSITIONS, AND METHODS OF USE AS PTPASE INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
09/07/2010
|
Application #:
|
12759010
|
Filing Dt:
|
04/13/2010
|
Publication #:
|
|
Pub Dt:
|
08/05/2010
| | | | |
Title:
|
OXADIAZOANTHRACENE COMPOUNDS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
02/26/2013
|
Application #:
|
12825631
|
Filing Dt:
|
06/29/2010
|
Publication #:
|
|
Pub Dt:
|
06/30/2011
| | | | |
Title:
|
SUBSTITUTED AZOANTHRACENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
03/15/2011
|
Application #:
|
12849225
|
Filing Dt:
|
08/03/2010
|
Publication #:
|
|
Pub Dt:
|
02/17/2011
| | | | |
Title:
|
OXADIAZOANTHRACENE COMPOUNDS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
09/03/2013
|
Application #:
|
12872580
|
Filing Dt:
|
08/31/2010
|
Publication #:
|
|
Pub Dt:
|
12/23/2010
| | | | |
Title:
|
OXADIAZOANTHRACENE COMPOUNDS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
11/12/2013
|
Application #:
|
12888660
|
Filing Dt:
|
09/23/2010
|
Publication #:
|
|
Pub Dt:
|
05/05/2011
| | | | |
Title:
|
Substituted Imidazole Derivatives And Methods Of Use Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
05/06/2014
|
Application #:
|
12936434
|
Filing Dt:
|
10/05/2010
|
Publication #:
|
|
Pub Dt:
|
02/03/2011
| | | | |
Title:
|
Ligands For The GLP-1 Receptor And Methods For Discovery Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
11/19/2013
|
Application #:
|
12961867
|
Filing Dt:
|
12/07/2010
|
Publication #:
|
|
Pub Dt:
|
03/31/2011
| | | | |
Title:
|
Urea Glucokinase Activators
|
|
|
Patent #:
|
|
Issue Dt:
|
02/12/2013
|
Application #:
|
12982775
|
Filing Dt:
|
12/30/2010
|
Publication #:
|
|
Pub Dt:
|
07/07/2011
| | | | |
Title:
|
CRYSTALLINE FORMS OF [3-(4- {2-BUTYL- 1 -[4-(4-CHLORO-PHENOXY)-PHENYL]-1H-IMIDAZOL-4-YL} -PHENOXY)-PROPYL]-DIETHYL-AMINE
|
|
|
Patent #:
|
|
Issue Dt:
|
11/04/2014
|
Application #:
|
12983604
|
Filing Dt:
|
01/03/2011
|
Publication #:
|
|
Pub Dt:
|
07/05/2012
| | | | |
Title:
|
RAGE FUSION PROTEINS AND METHODS OF USE
|
|
|
Patent #:
|
|
Issue Dt:
|
04/30/2013
|
Application #:
|
13028036
|
Filing Dt:
|
02/15/2011
|
Publication #:
|
|
Pub Dt:
|
09/22/2011
| | | | |
Title:
|
PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
06/24/2014
|
Application #:
|
13028406
|
Filing Dt:
|
02/16/2011
|
Publication #:
|
|
Pub Dt:
|
08/18/2011
| | | | |
Title:
|
SUBSTITUTED FUSED IMIDAZOLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
10/07/2014
|
Application #:
|
13040382
|
Filing Dt:
|
03/04/2011
|
Publication #:
|
|
Pub Dt:
|
06/30/2011
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
06/07/2016
|
Application #:
|
13114964
|
Filing Dt:
|
05/24/2011
|
Publication #:
|
|
Pub Dt:
|
12/22/2011
| | | | |
Title:
|
USE OF METFORMIN IN COMBINATION WITH A GLUCOKINASE ACTIVATOR AND COMPOSITIONS COMPRISING METFORMIN AND A GLUCOKINASE ACTIVATOR
|
|
|
Patent #:
|
|
Issue Dt:
|
01/06/2015
|
Application #:
|
13128045
|
Filing Dt:
|
05/06/2011
|
Publication #:
|
|
Pub Dt:
|
09/15/2011
| | | | |
Title:
|
Adamantyl Benzamide Derivatives
|
|
|
Patent #:
|
|
Issue Dt:
|
05/19/2015
|
Application #:
|
13265132
|
Filing Dt:
|
10/18/2011
|
Publication #:
|
|
Pub Dt:
|
02/16/2012
| | | | |
Title:
|
Control of RAGE Fusion Protein Glycosylation and RAGE Fusion Protein Compositions
|
|
|
Patent #:
|
|
Issue Dt:
|
12/11/2012
|
Application #:
|
13410628
|
Filing Dt:
|
03/02/2012
|
Publication #:
|
|
Pub Dt:
|
07/05/2012
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/29/2013
|
Application #:
|
13415000
|
Filing Dt:
|
03/08/2012
|
Publication #:
|
|
Pub Dt:
|
06/28/2012
| | | | |
Title:
|
UREA GLUCOKINASE ACTIVATORS
|
|
|
Patent #:
|
|
Issue Dt:
|
03/24/2015
|
Application #:
|
13707265
|
Filing Dt:
|
12/06/2012
|
Publication #:
|
|
Pub Dt:
|
04/18/2013
| | | | |
Title:
|
Substituted Azoanthracene Derivatives, Pharmaceutical Compositions, and Methods of Use Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
08/19/2014
|
Application #:
|
13739408
|
Filing Dt:
|
01/11/2013
|
Publication #:
|
|
Pub Dt:
|
09/05/2013
| | | | |
Title:
|
N-ADAMANTYL BENZAMIDES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE
|
|
|
Patent #:
|
|
Issue Dt:
|
06/03/2014
|
Application #:
|
13772685
|
Filing Dt:
|
02/21/2013
|
Publication #:
|
|
Pub Dt:
|
08/01/2013
| | | | |
Title:
|
PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
09/20/2016
|
Application #:
|
13894922
|
Filing Dt:
|
05/15/2013
|
Publication #:
|
|
Pub Dt:
|
09/26/2013
| | | | |
Title:
|
Compounds That Modulate Oxidative Stress
|
|
|
Patent #:
|
|
Issue Dt:
|
10/20/2015
|
Application #:
|
13934491
|
Filing Dt:
|
07/03/2013
|
Publication #:
|
|
Pub Dt:
|
11/07/2013
| | | | |
Title:
|
PHENYLGLYOXYLIC ACID DERIVATIVES AND THEIR PREPARATION AND USE
|
|
|
Patent #:
|
|
Issue Dt:
|
04/22/2014
|
Application #:
|
13956578
|
Filing Dt:
|
08/01/2013
|
Publication #:
|
|
Pub Dt:
|
11/28/2013
| | | | |
Title:
|
OXADIAZOANTHRACENE COMPOUNDS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
03/21/2017
|
Application #:
|
14049261
|
Filing Dt:
|
10/09/2013
|
Publication #:
|
|
Pub Dt:
|
02/06/2014
| | | | |
Title:
|
SUBSTITUTED IMIDAZOLE DERIVATIVES AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
08/01/2017
|
Application #:
|
14059529
|
Filing Dt:
|
10/22/2013
|
Publication #:
|
|
Pub Dt:
|
04/10/2014
| | | | |
Title:
|
TREATMENT OF MILD AND MODERATE ALZHEIMER'S DISEASE
|
|
|
Patent #:
|
|
Issue Dt:
|
06/26/2018
|
Application #:
|
14071976
|
Filing Dt:
|
11/05/2013
|
Publication #:
|
|
Pub Dt:
|
03/06/2014
| | | | |
Title:
|
Glucokinase Activator Compositions for the Treatment of Diabetes
|
|
|
Patent #:
|
|
Issue Dt:
|
01/13/2015
|
Application #:
|
14197771
|
Filing Dt:
|
03/05/2014
|
Publication #:
|
|
Pub Dt:
|
07/03/2014
| | | | |
Title:
|
OXADIAZOANTHRACENE COMPOUNDS FOR THE TREATMENT OF DIABETES
|
|
|
Patent #:
|
|
Issue Dt:
|
07/24/2018
|
Application #:
|
14215873
|
Filing Dt:
|
03/17/2014
|
Publication #:
|
|
Pub Dt:
|
07/17/2014
| | | | |
Title:
|
Substituted Fused Imidazole Derivatives, Pharmaceutical Compositions, and Methods of Use Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
06/02/2015
|
Application #:
|
14225837
|
Filing Dt:
|
03/26/2014
|
Publication #:
|
|
Pub Dt:
|
07/24/2014
| | | | |
Title:
|
PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF
|
|
|
Patent #:
|
|
Issue Dt:
|
12/09/2014
|
Application #:
|
14321884
|
Filing Dt:
|
07/02/2014
|
Publication #:
|
|
Pub Dt:
|
10/23/2014
| | | | |
Title:
|
N-ADAMANTYL BENZAMIDES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE
|
|
|
Patent #:
|
|
Issue Dt:
|
10/20/2015
|
Application #:
|
14477302
|
Filing Dt:
|
09/04/2014
|
Publication #:
|
|
Pub Dt:
|
12/18/2014
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
12/01/2015
|
Application #:
|
14489890
|
Filing Dt:
|
09/18/2014
|
Publication #:
|
|
Pub Dt:
|
01/01/2015
| | | | |
Title:
|
Tris(hydroxymethyl)Aminomethane Salts of a Small-Molecule GLP1R Agonist and Pharmaceutical Compositions and Uses Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
09/01/2015
|
Application #:
|
14556837
|
Filing Dt:
|
12/01/2014
|
Publication #:
|
|
Pub Dt:
|
03/26/2015
| | | | |
Title:
|
Oxadiazoanthracene Compounds for the Treatment of Diabetes
|
|
|
Patent #:
|
|
Issue Dt:
|
11/03/2015
|
Application #:
|
14603556
|
Filing Dt:
|
01/23/2015
|
Publication #:
|
|
Pub Dt:
|
05/28/2015
| | | | |
Title:
|
Substituted Azoanthracene Derivatives and Intermediates for Preparation Thereof
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
14799222
|
Filing Dt:
|
07/14/2015
|
Publication #:
|
|
Pub Dt:
|
11/05/2015
| | | | |
Title:
|
Combinations of a GLP1R Agonist and Metformin and Use Thereof for the Treatment of Type 2 Diabetes and Other Disorders
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
14840657
|
Filing Dt:
|
08/31/2015
|
Publication #:
|
|
Pub Dt:
|
01/21/2016
| | | | |
Title:
|
SOLID COMPOSITIONS COMPRISING A GLUCOKINASE ACTIVATOR AND METHODS OF MAKING AND USING THE SAME
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
14840682
|
Filing Dt:
|
08/31/2015
|
Publication #:
|
|
Pub Dt:
|
01/21/2016
| | | | |
Title:
|
STABLE GLUCOKINASE ACTIVATOR COMPOSITIONS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/19/2016
|
Application #:
|
14850012
|
Filing Dt:
|
09/10/2015
|
Publication #:
|
|
Pub Dt:
|
12/31/2015
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
01/02/2018
|
Application #:
|
14988143
|
Filing Dt:
|
02/11/2016
|
Publication #:
|
|
Pub Dt:
|
06/30/2016
| | | | |
Title:
|
Use of Metformin in Combination with a Glucokinase Activator and Compositions Comprising Metformin and a Glucokinase Activator
|
|
|
Patent #:
|
|
Issue Dt:
|
06/27/2017
|
Application #:
|
15184392
|
Filing Dt:
|
06/16/2016
|
Publication #:
|
|
Pub Dt:
|
10/13/2016
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|
|
Patent #:
|
|
Issue Dt:
|
07/18/2017
|
Application #:
|
15247256
|
Filing Dt:
|
08/25/2016
|
Publication #:
|
|
Pub Dt:
|
07/06/2017
| | | | |
Title:
|
Compounds That Modulate Oxidative Stress
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
15438111
|
Filing Dt:
|
02/21/2017
|
Publication #:
|
|
Pub Dt:
|
06/08/2017
| | | | |
Title:
|
Substituted Imidazole Derivatives and Methods of Use Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
01/08/2019
|
Application #:
|
15584459
|
Filing Dt:
|
05/02/2017
|
Publication #:
|
|
Pub Dt:
|
08/17/2017
| | | | |
Title:
|
Bach1 Inhibitors in Combination with Nrf2 Activators and Pharmaceutical Compositions Thereof
|
|
|
Patent #:
|
|
Issue Dt:
|
12/05/2017
|
Application #:
|
15600942
|
Filing Dt:
|
05/22/2017
|
Publication #:
|
|
Pub Dt:
|
09/07/2017
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|
|
Patent #:
|
NONE
|
Issue Dt:
|
|
Application #:
|
15631203
|
Filing Dt:
|
06/23/2017
|
Publication #:
|
|
Pub Dt:
|
11/16/2017
| | | | |
Title:
|
Treatment of Mild and Moderate Alzheimer's Disease
|
|
|
Patent #:
|
|
Issue Dt:
|
09/04/2018
|
Application #:
|
15687824
|
Filing Dt:
|
08/28/2017
|
Publication #:
|
|
Pub Dt:
|
12/14/2017
| | | | |
Title:
|
USE OF METFORMIN IN COMBINATION WITH A GLUCOKINASE ACTIVATOR AND COMPOSITIONS COMPRISING METFORMIN AND A GLUCOKINASE ACTIVATOR
|
|
|
Patent #:
|
|
Issue Dt:
|
10/02/2018
|
Application #:
|
15800794
|
Filing Dt:
|
11/01/2017
|
Publication #:
|
|
Pub Dt:
|
03/15/2018
| | | | |
Title:
|
TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-ALPHA SYNTHESIS AND AS PDE4 INHIBITORS
|
|