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Patent #:
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Issue Dt:
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08/18/2009
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Application #:
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10452481
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Filing Dt:
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05/30/2003
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Publication #:
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Pub Dt:
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01/15/2004
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Title:
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METHOD AND APPARATUS FOR MOLECULAR MECHANICS ANALYSIS OF MOLECULAR SYSTEMS
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Patent #:
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Issue Dt:
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04/20/2010
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Application #:
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11172215
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Filing Dt:
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06/29/2005
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Publication #:
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Pub Dt:
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12/29/2005
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Title:
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MOLECULAR PROPERTY MODELING USING RANKING
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Patent #:
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Issue Dt:
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03/20/2007
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Application #:
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11172216
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Filing Dt:
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06/29/2005
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Publication #:
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Pub Dt:
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12/29/2005
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Title:
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ESTIMATING THE ACCURACY OF MOLECULAR PROPERTY MODELS AND PREDICTIONS
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Patent #:
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Issue Dt:
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12/21/2010
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Application #:
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11304209
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Filing Dt:
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12/14/2005
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Publication #:
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Pub Dt:
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07/20/2006
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Title:
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MODELING BIOLOGICAL EFFECTS OF MOLECULES USING MOLECULAR PROPERTY MODELS
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Patent #:
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Issue Dt:
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05/28/2013
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Application #:
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11708793
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Filing Dt:
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02/21/2007
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Publication #:
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Pub Dt:
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08/21/2008
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Title:
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DERIVATIVES OF SQUARIC ACID WITH ANTI-PROLIFERATIVE ACTIVITY
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Patent #:
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Issue Dt:
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08/27/2013
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Application #:
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12311843
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Filing Dt:
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11/08/2010
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Publication #:
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Pub Dt:
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08/18/2011
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Title:
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PYRIDO [2,3-D] PYRIMIDINES AND THEIR USE AS KINASE INHIBITORS
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Patent #:
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Issue Dt:
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07/31/2012
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Application #:
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13105957
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Filing Dt:
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05/12/2011
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Publication #:
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Pub Dt:
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10/20/2011
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Title:
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RAF INHIBITORS
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Patent #:
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Issue Dt:
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06/13/2017
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Application #:
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13820489
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Filing Dt:
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07/22/2013
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Publication #:
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Pub Dt:
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11/07/2013
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Title:
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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Patent #:
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Issue Dt:
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10/27/2015
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Application #:
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14115623
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Filing Dt:
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05/15/2014
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Publication #:
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Pub Dt:
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09/18/2014
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Title:
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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Patent #:
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Issue Dt:
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01/31/2017
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Application #:
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14115849
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Filing Dt:
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04/08/2014
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Publication #:
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Pub Dt:
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09/04/2014
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Title:
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PIPERIDINE DERIVATIVES AND COMPOSITIONS FOR THE INHIBITION OF NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE (NAMPT)
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Patent #:
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Issue Dt:
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10/04/2016
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Application #:
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14382123
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Filing Dt:
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08/29/2014
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Publication #:
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Pub Dt:
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06/25/2015
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Title:
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PYRIDINYL AND PYRIMIDINYL SULFOXIDE AND SULFONE DERIVATIVES
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Patent #:
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Issue Dt:
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06/30/2020
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Application #:
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14382141
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Filing Dt:
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08/29/2014
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Publication #:
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Pub Dt:
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04/16/2015
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Title:
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AMIDO-BENZYL SULFONE AND SULFOXIDE DERIVATIVES
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Patent #:
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Issue Dt:
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11/21/2017
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Application #:
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14382210
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Filing Dt:
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08/29/2014
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Publication #:
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Pub Dt:
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01/07/2016
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Title:
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AMIDO SPIROCYCLIC AMIDE AND SULFONAMIDE DERIVATIVES
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Patent #:
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Issue Dt:
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02/27/2018
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Application #:
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14982127
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Filing Dt:
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12/29/2015
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Publication #:
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Pub Dt:
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06/30/2016
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Title:
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PYRROLO AND PYRAZOLOPYRIMIDINES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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Patent #:
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Issue Dt:
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06/19/2018
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Application #:
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14982131
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Filing Dt:
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12/29/2015
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Publication #:
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Pub Dt:
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06/30/2016
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Title:
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PYRROLOTRIAZINONES AND IMIDAZOTRIAZINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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Patent #:
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Issue Dt:
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01/22/2019
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15013811
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Filing Dt:
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02/02/2016
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Publication #:
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Pub Dt:
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08/04/2016
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Title:
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BICYCLIC [4,6,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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02/26/2019
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Application #:
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15013814
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Filing Dt:
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02/02/2016
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Publication #:
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Pub Dt:
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08/04/2016
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Title:
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3-ALKYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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03/26/2019
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Application #:
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15013816
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Filing Dt:
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02/02/2016
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Publication #:
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Pub Dt:
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08/04/2016
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Title:
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3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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02/26/2019
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Application #:
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15013820
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Filing Dt:
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02/02/2016
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Publication #:
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Pub Dt:
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08/04/2016
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Title:
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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10/30/2018
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Application #:
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15013826
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Filing Dt:
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02/02/2016
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Publication #:
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Pub Dt:
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08/04/2016
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Title:
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3-ARYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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04/03/2018
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Application #:
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15015563
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Filing Dt:
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02/04/2016
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Publication #:
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Pub Dt:
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08/11/2016
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Title:
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THIENOPYRIMIDINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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Patent #:
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Issue Dt:
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04/10/2018
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Application #:
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15015566
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Filing Dt:
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02/04/2016
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Publication #:
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Pub Dt:
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08/11/2016
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Title:
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ISOTHIAZOLOPYRIMIDINONES, PYRAZOLOPYRIMIDINONES, AND PYRROLOPYRIMIDINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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Patent #:
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Issue Dt:
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12/12/2017
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15015571
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Filing Dt:
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02/04/2016
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Publication #:
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Pub Dt:
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08/11/2016
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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Patent #:
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Issue Dt:
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08/29/2017
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15067605
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Filing Dt:
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03/11/2016
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Publication #:
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Pub Dt:
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09/15/2016
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Title:
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ALPHA-CINNAMIDE COMPOUNDS AND COMPOSITIONS AS HDAC8 INHIBITORS
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Patent #:
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Issue Dt:
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05/02/2017
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Application #:
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15130603
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Filing Dt:
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04/15/2016
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Publication #:
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Pub Dt:
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10/20/2016
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Title:
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3-SPIROCYCLIC-6-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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04/25/2017
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Application #:
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15130613
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Filing Dt:
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04/15/2016
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Publication #:
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Pub Dt:
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10/20/2016
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Title:
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3-SPIRO-7-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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07/24/2018
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Application #:
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15255817
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Filing Dt:
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09/02/2016
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Publication #:
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Pub Dt:
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03/09/2017
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Title:
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[6,6] FUSED BICYCLIC HDAC8 INHIBITORS
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Patent #:
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Issue Dt:
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04/30/2019
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15352184
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Filing Dt:
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11/15/2016
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Publication #:
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Pub Dt:
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12/28/2017
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Title:
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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Patent #:
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Issue Dt:
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12/24/2019
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15837393
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12/11/2017
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Publication #:
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Pub Dt:
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06/14/2018
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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08/13/2019
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15874163
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01/18/2018
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Pub Dt:
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11/29/2018
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Title:
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PYRROLO AND PYRAZOLOPYRIMIDINES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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08/13/2019
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15907007
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02/27/2018
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Pub Dt:
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12/06/2018
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Title:
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ISOTHIAZOLOPYRIMIDINONES, PYRAZOLOPYRIMIDINONES, AND PYRROLOPYRIMIDINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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08/13/2019
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15909200
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03/01/2018
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Pub Dt:
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12/06/2018
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Title:
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THIENOPYRIMIDINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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04/23/2019
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15925559
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03/19/2018
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Pub Dt:
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10/18/2018
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Title:
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ALPHA-CINNAMIDE COMPOUNDS AND COMPOSITIONS AS HDAC8 INHIBITORS
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08/04/2020
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15936086
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03/26/2018
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Pub Dt:
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11/29/2018
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Title:
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AMIDO SPIROCYCLIC AMIDE AND SULFONAMIDE DERIVATIVES
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07/16/2019
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15988790
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05/24/2018
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Pub Dt:
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11/29/2018
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Title:
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PYRROLOTRIAZINONES AND IMIDAZOTRIAZINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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Patent #:
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08/06/2019
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16003861
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06/08/2018
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Pub Dt:
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12/13/2018
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Title:
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[6,6] FUSED BICYCLIC HDAC8 INHIBITORS
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Patent #:
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06/25/2019
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16008378
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06/14/2018
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Pub Dt:
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10/11/2018
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Title:
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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Patent #:
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01/12/2021
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16077406
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08/10/2018
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Pub Dt:
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11/28/2019
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Title:
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Thienopyrazine Carboxamides as Ubiquitin-Specific Protease Inhibitors
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Patent #:
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02/09/2021
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16077407
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08/10/2018
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Publication #:
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Pub Dt:
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01/16/2020
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Title:
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Thienopyridine Carboxamides as Ubiquitin-Specific Protease Inhibitors
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12/03/2019
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16133918
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09/18/2018
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Pub Dt:
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01/17/2019
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Title:
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3-ARYL-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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Issue Dt:
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12/03/2019
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16133922
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Filing Dt:
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09/18/2018
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Publication #:
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Pub Dt:
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01/17/2019
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Title:
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3-ARYL-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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08/13/2019
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16173871
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Filing Dt:
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10/29/2018
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Publication #:
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Pub Dt:
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02/28/2019
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Title:
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3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/24/2019
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16179061
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11/02/2018
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Pub Dt:
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03/07/2019
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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12/31/2019
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16179071
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11/02/2018
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Publication #:
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Pub Dt:
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03/07/2019
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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12/17/2019
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16179099
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11/02/2018
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Pub Dt:
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03/07/2019
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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12/31/2019
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16179111
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11/02/2018
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Pub Dt:
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03/07/2019
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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12/31/2019
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16179117
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11/02/2018
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Pub Dt:
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03/07/2019
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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12/31/2019
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16179125
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11/02/2018
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Pub Dt:
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03/07/2019
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Title:
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QUINAZOLINONES AND AZAQUINAZOLINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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09/10/2019
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16199489
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11/26/2018
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03/28/2019
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Title:
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BICYCLIC [4,6,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/17/2019
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16202207
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11/28/2018
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03/21/2019
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Title:
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METHODS USING HDAC11 INHIBITORS
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01/21/2020
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16202210
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11/28/2018
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Publication #:
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Pub Dt:
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03/21/2019
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Title:
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METHODS USING HDAC11 INHIBITORS
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10/29/2019
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16212360
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12/06/2018
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04/11/2019
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Title:
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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09/17/2019
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16218108
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12/12/2018
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Pub Dt:
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04/18/2019
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Title:
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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10/01/2019
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16218114
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12/12/2018
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Pub Dt:
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04/18/2019
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Title:
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/24/2019
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16218122
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12/12/2018
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Pub Dt:
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04/18/2019
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Issue Dt:
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09/24/2019
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Application #:
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16218126
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12/12/2018
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Pub Dt:
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04/18/2019
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Title:
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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10/22/2019
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16218132
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12/12/2018
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Pub Dt:
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04/18/2019
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Title:
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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11/05/2019
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16219381
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12/13/2018
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Pub Dt:
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04/25/2019
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Title:
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3-ALKYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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10/15/2019
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16219592
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12/13/2018
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Pub Dt:
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04/25/2019
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Title:
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3-ALKYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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Patent #:
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10/29/2019
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16219648
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12/13/2018
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Pub Dt:
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04/25/2019
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Title:
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3-ALKYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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11/05/2019
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16219669
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12/13/2018
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05/02/2019
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Title:
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3-ALKYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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09/24/2019
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16219685
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12/13/2018
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Pub Dt:
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04/25/2019
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Title:
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3-ALKYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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11/19/2019
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16220035
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12/14/2018
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04/25/2019
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Title:
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3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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10/22/2019
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16220041
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12/14/2018
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04/25/2019
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Title:
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3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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11/12/2019
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16220046
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12/14/2018
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04/25/2019
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Title:
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3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/03/2019
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16220049
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12/14/2018
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04/25/2019
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3-ARYL-4-AMIDO-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/03/2019
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16222868
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12/17/2018
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04/18/2019
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3-ARYL-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/10/2019
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16222871
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12/17/2018
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04/25/2019
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3-ARYL-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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02/11/2020
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16309980
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12/14/2018
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07/04/2019
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2-SPIRO-5- AND 6-HYDROXAMIC ACID INDANES AS HDAC INHIBITORS
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10/13/2020
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16331916
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03/08/2019
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07/04/2019
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MONOCYCLIC COMPOUNDS USEFUL AS GPR120 MODULATORS
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12/15/2020
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16331928
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03/08/2019
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07/18/2019
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BICYCLIC COMPOUNDS USEFUL AS GPR120 MODULATORS
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12/17/2019
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16387937
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04/18/2019
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08/08/2019
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ALPHA-CINNAMIDE COMPOUNDS AND COMPOSITIONS AS HDAC8 INHIBITORS
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05/12/2020
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16419333
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05/22/2019
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09/05/2019
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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04/20/2021
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16449599
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06/24/2019
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10/10/2019
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PYRROLOTRIAZINONES AND IMIDAZOTRIAZINONES AS UBIQUITIN-SPECIFIC PROTEASE 7 INHIBITORS
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11/10/2020
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16449675
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06/24/2019
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10/10/2019
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02/02/2021
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16515194
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07/18/2019
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11/28/2019
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02/23/2021
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16515281
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07/18/2019
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11/28/2019
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03/02/2021
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16517149
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07/19/2019
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12/05/2019
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12/22/2020
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16522082
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07/25/2019
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11/14/2019
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09/15/2020
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08/12/2019
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12/26/2019
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NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT
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04/27/2021
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09/11/2019
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01/02/2020
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11/10/2020
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16654704
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10/16/2019
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02/13/2020
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11/03/2020
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16660015
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10/22/2019
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02/13/2020
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11/10/2020
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02/20/2020
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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03/12/2020
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03/19/2020
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04/23/2020
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09/10/2020
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06/10/2021
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11/19/2020
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05/11/2023
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02/18/2021
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08/12/2021
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10/25/2022
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08/12/2021
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01/14/2021
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03/22/2022
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01/14/2021
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3-ALKYL BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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03/15/2022
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17031815
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09/24/2020
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01/14/2021
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3-ARYL-BICYCLIC [4,5,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
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12/27/2022
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10/20/2020
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08/19/2021
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08/16/2022
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10/08/2020
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05/13/2021
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[6,6] FUSED BICYCLIC HDAC8 INHIBITORS
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